EP0805145B1 - Effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-Aminosäuren - Google Patents

Effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-Aminosäuren Download PDF

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Publication number
EP0805145B1
EP0805145B1 EP97106550A EP97106550A EP0805145B1 EP 0805145 B1 EP0805145 B1 EP 0805145B1 EP 97106550 A EP97106550 A EP 97106550A EP 97106550 A EP97106550 A EP 97106550A EP 0805145 B1 EP0805145 B1 EP 0805145B1
Authority
EP
European Patent Office
Prior art keywords
general formula
compounds
carbon atoms
chain
straight
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
EP97106550A
Other languages
German (de)
English (en)
French (fr)
Other versions
EP0805145A1 (de
Inventor
Joachim Dr. Mittendorf
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to SI9730164T priority Critical patent/SI0805145T1/xx
Publication of EP0805145A1 publication Critical patent/EP0805145A1/de
Application granted granted Critical
Publication of EP0805145B1 publication Critical patent/EP0805145B1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/24—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/74—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
EP97106550A 1996-05-03 1997-04-21 Effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-Aminosäuren Expired - Lifetime EP0805145B1 (de)

Priority Applications (1)

Application Number Priority Date Filing Date Title
SI9730164T SI0805145T1 (en) 1996-05-03 1997-04-21 Efficient and highly enantioselective process for the preparation of enantiomerically pure cylopentane-beta-amino acids

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19617772 1996-05-03
DE19617772A DE19617772A1 (de) 1996-05-03 1996-05-03 Neues effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-aminosäuren

Publications (2)

Publication Number Publication Date
EP0805145A1 EP0805145A1 (de) 1997-11-05
EP0805145B1 true EP0805145B1 (de) 2001-10-31

Family

ID=7793231

Family Applications (1)

Application Number Title Priority Date Filing Date
EP97106550A Expired - Lifetime EP0805145B1 (de) 1996-05-03 1997-04-21 Effizientes und hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan-beta-Aminosäuren

Country Status (25)

Country Link
US (1) US5877343A (zh)
EP (1) EP0805145B1 (zh)
JP (1) JPH1087586A (zh)
KR (1) KR970074749A (zh)
CN (1) CN1168883A (zh)
AR (2) AR006944A1 (zh)
AT (1) ATE207876T1 (zh)
AU (1) AU1915697A (zh)
BR (1) BR9701983A (zh)
CA (1) CA2204055A1 (zh)
CZ (1) CZ135397A3 (zh)
DE (2) DE19617772A1 (zh)
DK (1) DK0805145T3 (zh)
ES (1) ES2166930T3 (zh)
HR (1) HRP970214A2 (zh)
HU (1) HU9700831D0 (zh)
ID (1) ID16859A (zh)
IL (1) IL120747A0 (zh)
NO (1) NO971983L (zh)
PL (1) PL319775A1 (zh)
PT (1) PT805145E (zh)
SI (1) SI0805145T1 (zh)
SK (1) SK55497A3 (zh)
SV (1) SV1997000031A (zh)
ZA (1) ZA973796B (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002010096A1 (en) * 2000-07-31 2002-02-07 Brandeis University Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
EP1419125A4 (en) * 2001-07-31 2005-03-23 Univ Brandeis KINETIC RACEMAT SPLITS OF CHIRALER 2 AND 3 SUBSTITUTED CARBOXYLIC ACIDS
US7531662B2 (en) * 2003-06-11 2009-05-12 Brandeis University Cinchona-alkaloid-based catalysts, and asymmetric alcoholysis of cyclic anhydrides using them

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3560565A (en) * 1969-06-03 1971-02-02 American Home Prod 1-amino-n-sulfonylcyclopentane-carboxamides
GB8716278D0 (en) * 1987-07-10 1987-08-19 Fujisawa Pharmaceutical Co Antimicrobial agent
AU673824B2 (en) * 1992-05-29 1996-11-28 Bayer Aktiengesellschaft Cyclopentane- and -pentene-beta-amino acids
DE4400749A1 (de) * 1994-01-13 1995-07-20 Bayer Ag Neues hochenantioselektives Verfahren zur Herstellung von enantiomerenreinen Cyclopentan- und -penten-beta-Aminosäuren

Also Published As

Publication number Publication date
ES2166930T3 (es) 2002-05-01
DE19617772A1 (de) 1997-11-13
EP0805145A1 (de) 1997-11-05
SV1997000031A (es) 1997-10-23
PT805145E (pt) 2002-03-28
SK55497A3 (en) 1997-11-05
IL120747A0 (en) 1997-09-30
MX9702768A (es) 1997-11-29
AR006944A1 (es) 1999-09-29
BR9701983A (pt) 1998-09-15
NO971983L (no) 1997-11-04
CN1168883A (zh) 1997-12-31
CZ135397A3 (cs) 1998-05-13
ID16859A (id) 1997-11-20
PL319775A1 (en) 1997-11-10
HU9700831D0 (en) 1997-06-30
SI0805145T1 (en) 2002-02-28
DK0805145T3 (da) 2002-03-04
CA2204055A1 (en) 1997-11-03
US5877343A (en) 1999-03-02
ATE207876T1 (de) 2001-11-15
KR970074749A (ko) 1997-12-10
DE59705135D1 (de) 2001-12-06
JPH1087586A (ja) 1998-04-07
AR013071A2 (es) 2000-12-13
NO971983D0 (no) 1997-04-29
HRP970214A2 (en) 1998-04-30
ZA973796B (en) 1997-12-01
AU1915697A (en) 1997-11-06

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