EP0000300B1 - Estra-1,3,5(10),6-tétraènes substitués, procédé de préparation et application dans la synthèse de stéroides marqués au tritium - Google Patents

Estra-1,3,5(10),6-tétraènes substitués, procédé de préparation et application dans la synthèse de stéroides marqués au tritium Download PDF

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Publication number
EP0000300B1
EP0000300B1 EP78400016A EP78400016A EP0000300B1 EP 0000300 B1 EP0000300 B1 EP 0000300B1 EP 78400016 A EP78400016 A EP 78400016A EP 78400016 A EP78400016 A EP 78400016A EP 0000300 B1 EP0000300 B1 EP 0000300B1
Authority
EP
European Patent Office
Prior art keywords
methoxy
estra
agent
diol
radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
EP78400016A
Other languages
German (de)
English (en)
French (fr)
Other versions
EP0000300A1 (fr
Inventor
Alain Jouquey
Jean-Pierre Raynaud
Jean Salmon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of EP0000300A1 publication Critical patent/EP0000300A1/fr
Application granted granted Critical
Publication of EP0000300B1 publication Critical patent/EP0000300B1/fr
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
EP78400016A 1977-06-27 1978-06-12 Estra-1,3,5(10),6-tétraènes substitués, procédé de préparation et application dans la synthèse de stéroides marqués au tritium Expired EP0000300B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7719613 1977-06-27
FR7719613A FR2401173A1 (fr) 1977-06-27 1977-06-27 Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium

Publications (2)

Publication Number Publication Date
EP0000300A1 EP0000300A1 (fr) 1979-01-10
EP0000300B1 true EP0000300B1 (fr) 1982-01-06

Family

ID=9192607

Family Applications (1)

Application Number Title Priority Date Filing Date
EP78400016A Expired EP0000300B1 (fr) 1977-06-27 1978-06-12 Estra-1,3,5(10),6-tétraènes substitués, procédé de préparation et application dans la synthèse de stéroides marqués au tritium

Country Status (7)

Country Link
US (1) US4191697A (it)
EP (1) EP0000300B1 (it)
JP (2) JPS5412362A (it)
CA (1) CA1130277A (it)
DE (1) DE2861501D1 (it)
FR (1) FR2401173A1 (it)
IT (1) IT1105060B (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3414508A1 (de) * 1984-04-13 1985-10-24 Schering AG, 1000 Berlin und 4709 Bergkamen Mehrfach tritiierte steroid-20.17-spirolactone und ihre verwendung als tracersubstanzen
DE3937412A1 (de) * 1989-11-10 1991-05-16 Hoechst Ag Synthetische vakzine zur spezifischen induktion zytotoxischer t-lymphozyten
US4757062A (en) * 1985-11-01 1988-07-12 E. I. Du Pont De Nemours And Company Substituted benzoate ester prodrugs of estrogens
AU1924701A (en) 1999-12-15 2001-06-25 Dow Global Technologies Inc. Multi-component articles prepared from hydrogenated block copolymers
DE102017119621A1 (de) 2016-12-01 2018-06-07 Pouya Molana Mayonnaise-Pulver-Zusammensetzung und Verfahren zur Herstellung eines Lebensmittelprodukts unter Verwendung eines solchen

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3020294A (en) * 1950-03-28 1962-02-06 Syntex Sa Production of ring a aromatic steroids
FR5519M (it) * 1966-06-07 1967-11-06
FR2115033B1 (it) * 1970-11-24 1974-03-22 Roussel Uclaf

Also Published As

Publication number Publication date
IT7850022A0 (it) 1978-06-26
JPS6360035B2 (it) 1988-11-22
CA1130277A (fr) 1982-08-24
JPS62142196A (ja) 1987-06-25
DE2861501D1 (en) 1982-02-25
FR2401173B1 (it) 1980-04-04
US4191697A (en) 1980-03-04
EP0000300A1 (fr) 1979-01-10
FR2401173A1 (fr) 1979-03-23
JPS5412362A (en) 1979-01-30
IT1105060B (it) 1985-10-28
JPS6220196B2 (it) 1987-05-06

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