EG18484A - Process for preparing 1-tertiary-alkyl-substituted naphthyridine and quinoline carboxylic acid antibacterial agents - Google Patents
Process for preparing 1-tertiary-alkyl-substituted naphthyridine and quinoline carboxylic acid antibacterial agentsInfo
- Publication number
- EG18484A EG18484A EG579/87A EG57987A EG18484A EG 18484 A EG18484 A EG 18484A EG 579/87 A EG579/87 A EG 579/87A EG 57987 A EG57987 A EG 57987A EG 18484 A EG18484 A EG 18484A
- Authority
- EG
- Egypt
- Prior art keywords
- tertiary
- alkyl
- preparing
- carboxylic acid
- antibacterial agents
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91675286A | 1986-10-08 | 1986-10-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EG18484A true EG18484A (en) | 1993-04-30 |
Family
ID=25437769
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EG579/87A EG18484A (en) | 1986-10-08 | 1987-10-07 | Process for preparing 1-tertiary-alkyl-substituted naphthyridine and quinoline carboxylic acid antibacterial agents |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP0288519A4 (xx) |
| AU (2) | AU611400B2 (xx) |
| DD (2) | DD280530A5 (xx) |
| EG (1) | EG18484A (xx) |
| FI (1) | FI883894A0 (xx) |
| HU (3) | HU911136D0 (xx) |
| WO (1) | WO1988002627A1 (xx) |
| ZA (1) | ZA877471B (xx) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS62108878A (ja) * | 1985-11-05 | 1987-05-20 | Kyorin Pharmaceut Co Ltd | キノロンカルボン酸誘導体およびその製造方法 |
| CA1336090C (en) * | 1988-08-31 | 1995-06-27 | Isao Hayakawa | Spiro-substituted cyclic amines of quinolone derivatives |
| US5286723A (en) * | 1988-08-31 | 1994-02-15 | Daiichi Seiyaku Co., Ltd. | Spiro compound |
| CA1332605C (en) * | 1988-10-03 | 1994-10-18 | Yasuhiro Nishitani | Pyridonecarboxylic acids |
| US5262417A (en) * | 1988-12-06 | 1993-11-16 | The Upjohn Company | Antibacterial quinolone compounds |
| US4916141A (en) * | 1989-03-28 | 1990-04-10 | Warner-Lambert Company | (S)-7-(3-amino-1-pyrrolidinyl)-1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid |
| AU618460B2 (en) * | 1989-04-18 | 1991-12-19 | Hokuriku Pharmaceutical Co. Ltd. | Thiazetoquinoline-3-carboxylic acid derivative, method for preparation thereof, and a pharmaceutical composition comprising the same |
| US5342846A (en) * | 1990-12-05 | 1994-08-30 | Synphar Laboratories, Inc. | 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds and 7-(substituted triazolyl pyrrolidin-1-yl) 4-oxoquinoline-3-carboxylic acid derivatives useful as antibacterial agents |
| TW425394B (en) * | 1996-04-24 | 2001-03-11 | Daiichi Seiyaku Co | Antimicrobial quinolone derivatives having 3-(N-cycloalkyl) aminomethylpyrrolidine group |
| US6872742B2 (en) | 1996-08-28 | 2005-03-29 | The Procter & Gamble Company | Substituted cyclic amine metalloprotease inhibitors |
| DE69716449T2 (de) * | 1996-08-28 | 2003-08-07 | Procter & Gamble | Substituierte zyklische amine als metalloproteaseinhibitoren |
| NZ503945A (en) | 1997-07-31 | 2002-11-26 | Procter & Gamble | Metalloprotease-inhibiting amide derivatives |
| CN1349498A (zh) | 1999-03-03 | 2002-05-15 | 宝洁公司 | 含有链烯基和炔基的金属蛋白酶抑制剂 |
| SE0003795D0 (sv) | 2000-10-20 | 2000-10-20 | Astrazeneca Ab | Pharmaceutically useful compounds |
| JP2006504690A (ja) * | 2002-09-10 | 2006-02-09 | ファイザー・プロダクツ・インク | Ｃｎｓ及びその他の障害の治療に有用なジアザ二環式化合物 |
| JP2008528586A (ja) * | 2005-01-25 | 2008-07-31 | グラクソ グループ リミテッド | 抗菌剤 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH404678A (de) * | 1960-02-17 | 1965-12-31 | Lepetit Spa | Verfahren zur Herstellung von neuen 3,8-Diazabicyclo-(3,2,1)-octanen |
| GB937183A (en) * | 1960-02-17 | 1963-09-18 | Lepetit Spa | 3,8-diazabicyclo-[3,2,1]-octanes |
| DE2808070A1 (de) * | 1978-02-24 | 1979-08-30 | Bayer Ag | Verfahren zur herstellung von 4-pyridon-3-carbonsaeuren und/oder deren derivaten |
| GB2093018B (en) * | 1979-08-22 | 1984-09-12 | Kyorin Seiyaku Kk | 6,8-difluoro-quinoline carboxylic acid derivatives |
| JPS5649382A (en) * | 1979-09-28 | 1981-05-02 | Dainippon Pharmaceut Co Ltd | 6-fluoro-7-cyclic amino-1,8-naphthylidine derivative and its salt |
| US4665079A (en) * | 1984-02-17 | 1987-05-12 | Warner-Lambert Company | Antibacterial agents |
| US4571396A (en) * | 1984-04-16 | 1986-02-18 | Warner-Lambert Company | Antibacterial agents |
| DE3509546A1 (de) * | 1985-03-16 | 1986-09-25 | Bayer Ag, 5090 Leverkusen | 7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel |
| US4578473A (en) * | 1985-04-15 | 1986-03-25 | Warner-Lambert Company | Process for quinoline-3-carboxylic acid antibacterial agents |
| US4772706A (en) * | 1986-01-13 | 1988-09-20 | Warner-Lambert Company | Process for quinoline-3-carboxylic acid antibacterial agents |
| DE3601567A1 (de) * | 1986-01-21 | 1987-07-23 | Bayer Ag | 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate |
-
1987
- 1987-10-05 ZA ZA877471A patent/ZA877471B/xx unknown
- 1987-10-06 DD DD87327989A patent/DD280530A5/de not_active IP Right Cessation
- 1987-10-06 DD DD87307706A patent/DD266354A5/de not_active IP Right Cessation
- 1987-10-07 EG EG579/87A patent/EG18484A/xx active
- 1987-10-08 AU AU81581/87A patent/AU611400B2/en not_active Ceased
- 1987-10-08 HU HU911136A patent/HU911136D0/hu not_active IP Right Cessation
- 1987-10-08 EP EP19870907178 patent/EP0288519A4/en active Pending
- 1987-10-08 HU HU875686A patent/HUT52500A/hu unknown
- 1987-10-08 HU HU875686A patent/HU203753B/hu not_active IP Right Cessation
- 1987-10-08 WO PCT/US1987/002556 patent/WO1988002627A1/en not_active Application Discontinuation
-
1988
- 1988-08-23 FI FI883894A patent/FI883894A0/fi not_active Application Discontinuation
-
1991
- 1991-05-01 AU AU76326/91A patent/AU7632691A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU8158187A (en) | 1988-05-06 |
| FI883894A (fi) | 1988-08-23 |
| WO1988002627A1 (en) | 1988-04-21 |
| DD266354A5 (de) | 1989-03-29 |
| FI883894A0 (fi) | 1988-08-23 |
| HU911136D0 (en) | 1991-10-28 |
| DD280530A5 (de) | 1990-07-11 |
| AU7632691A (en) | 1991-08-08 |
| AU611400B2 (en) | 1991-06-13 |
| HUT52500A (en) | 1990-07-28 |
| ZA877471B (en) | 1988-04-05 |
| HU203753B (en) | 1991-09-30 |
| EP0288519A4 (en) | 1992-04-15 |
| EP0288519A1 (en) | 1988-11-02 |
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