EE9900537A - Karbotsükliline nukleosiidhemisulfaat ja selle kasutamine viirusinfektsioonide raviks - Google Patents

Karbotsükliline nukleosiidhemisulfaat ja selle kasutamine viirusinfektsioonide raviks

Info

Publication number
EE9900537A
EE9900537A EEP199900537A EEP9900537A EE9900537A EE 9900537 A EE9900537 A EE 9900537A EE P199900537 A EEP199900537 A EE P199900537A EE P9900537 A EEP9900537 A EE P9900537A EE 9900537 A EE9900537 A EE 9900537A
Authority
EE
Estonia
Prior art keywords
treatment
viral infections
carbocyclic nucleoside
hemisulfate
nucleoside hemisulfate
Prior art date
Application number
EEP199900537A
Other languages
English (en)
Inventor
Francis Jones Martin
Frederick Seager John
John Wallis Christopher
Couper Brodie Alastair
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10812407&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE9900537(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of EE9900537A publication Critical patent/EE9900537A/et
Publication of EE03924B1 publication Critical patent/EE03924B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/16Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
EEP199900537A 1997-05-17 1998-05-14 Karbotsükliline nukleosiidhemisulfaat ja selle kasutamine viirusinfektsioonide raviks EE03924B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9709945.1A GB9709945D0 (en) 1997-05-17 1997-05-17 A novel salt
PCT/EP1998/002835 WO1998052949A1 (en) 1997-05-17 1998-05-14 Carbocyclic nucleoside hemisulfate and its use in treating viral infections

Publications (2)

Publication Number Publication Date
EE9900537A true EE9900537A (et) 2000-06-15
EE03924B1 EE03924B1 (et) 2002-12-16

Family

ID=10812407

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900537A EE03924B1 (et) 1997-05-17 1998-05-14 Karbotsükliline nukleosiidhemisulfaat ja selle kasutamine viirusinfektsioonide raviks

Country Status (51)

Country Link
US (1) US6294540B1 (et)
EP (1) EP0983271B1 (et)
JP (2) JP3150711B2 (et)
KR (1) KR100521292B1 (et)
CN (2) CN1150194C (et)
AP (1) AP2009A (et)
AR (2) AR015668A1 (et)
AT (1) ATE259811T1 (et)
AU (1) AU739953B2 (et)
BG (1) BG64390B1 (et)
BR (1) BRPI9809126B8 (et)
CA (1) CA2289753C (et)
CO (1) CO4940435A1 (et)
DE (1) DE69821758T2 (et)
DK (1) DK0983271T3 (et)
DZ (1) DZ2493A1 (et)
EA (1) EA001809B1 (et)
EE (1) EE03924B1 (et)
EG (1) EG23836A (et)
ES (1) ES2214712T3 (et)
GB (3) GB9709945D0 (et)
GE (1) GEP20022680B (et)
HK (1) HK1024236A1 (et)
HN (1) HN1998000071A (et)
HR (1) HRP980265B1 (et)
HU (1) HU226563B1 (et)
ID (1) ID24910A (et)
IL (2) IL132793A0 (et)
IS (1) IS2207B (et)
JO (1) JO2032B1 (et)
MA (1) MA26498A1 (et)
MY (1) MY120151A (et)
NO (1) NO324731B1 (et)
NZ (2) NZ510622A (et)
OA (1) OA11304A (et)
PA (1) PA8451301A1 (et)
PE (1) PE78799A1 (et)
PL (1) PL189527B1 (et)
PT (1) PT983271E (et)
RS (1) RS49655B (et)
SA (1) SA98190179B1 (et)
SI (1) SI0983271T1 (et)
SK (1) SK285159B6 (et)
SV (1) SV1998000057A (et)
TN (1) TNSN98065A1 (et)
TR (1) TR199902810T2 (et)
TW (1) TW480259B (et)
UA (1) UA56231C2 (et)
UY (1) UY25004A1 (et)
WO (1) WO1998052949A1 (et)
ZA (2) ZA984085B (et)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9802472D0 (en) * 1998-02-06 1998-04-01 Glaxo Group Ltd Pharmaceutical compositions
HU226998B1 (en) * 2000-11-23 2010-04-28 Richter Gedeon Nyrt Desloratadine hemisulphate, process for the preparation thereof and pharmaceutical compositions containing the same
GB0320738D0 (en) 2003-09-04 2003-10-08 Glaxo Group Ltd Novel process
EP1905772A1 (en) * 2006-09-28 2008-04-02 Esteve Quimica, S.A. Process for the preparation of abacavir
JP5334852B2 (ja) * 2006-09-28 2013-11-06 エステヴェ キミカ, エス.エー. アバカビルの製造方法
EP2085397A1 (en) 2008-01-21 2009-08-05 Esteve Quimica, S.A. Crystalline form of abacavir
EP2218721A1 (en) * 2009-02-11 2010-08-18 LEK Pharmaceuticals d.d. Novel salts of sitagliptin
EP2305680A3 (en) 2009-09-30 2011-05-18 Aurobindo Pharma Limited Novel salts of (1S,4R)-cis-4-[2-amino-6-(cyclopropylamino)-9H-purin-9-yl]-2-cyclopentene-1-methanol
DK3494972T3 (da) 2010-01-27 2024-01-29 Viiv Healthcare Co Kombinationer af dolutegravir og lamivudin til behandling af HIV-infektion
CN103282369A (zh) 2011-04-08 2013-09-04 劳乐斯实验室私营有限公司 抗逆转录病毒化合物与抗氧化酸的固体形式、其制备方法以及其药物组合物
EP2962693B1 (en) 2013-02-27 2019-01-09 Kyoto University Pharmaceutical composition comprising abacavir for the treatment of cancer
CN104788451A (zh) * 2014-01-21 2015-07-22 浙江九洲药业股份有限公司 一种阿巴卡韦的制备方法
CN105315280A (zh) * 2014-06-06 2016-02-10 上海迪赛诺化学制药有限公司 一种阿巴卡韦结晶体及其制备方法
US10874687B1 (en) 2020-02-27 2020-12-29 Atea Pharmaceuticals, Inc. Highly active compounds against COVID-19

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY104575A (en) * 1989-12-22 1994-04-30 The Wellcome Foundation Ltd Therapeutic nucleosides.
GB9417249D0 (en) * 1994-08-26 1994-10-19 Wellcome Found A novel salt
MY115461A (en) * 1995-03-30 2003-06-30 Wellcome Found Synergistic combinations of zidovudine, 1592u89 and 3tc
TR199802703T2 (xx) * 1996-06-25 1999-03-22 Glaxo Group Limited HIV tedavisinde Vx478, Zidov�din, ve/veya 1592U89 i�eren kombinasyonlar�n kullan�m�.

Also Published As

Publication number Publication date
JP2000327679A (ja) 2000-11-28
BR9809126A (pt) 2000-08-01
RS49655B (sr) 2007-09-21
PT983271E (pt) 2004-07-30
CN1263529A (zh) 2000-08-16
BG64390B1 (bg) 2004-12-30
HK1024236A1 (en) 2000-10-05
AR059120A2 (es) 2008-03-12
GB0010222D0 (en) 2000-06-14
BG103959A (en) 2000-12-29
EE03924B1 (et) 2002-12-16
IS5246A (is) 1999-11-11
WO1998052949A1 (en) 1998-11-26
DE69821758T2 (de) 2005-01-13
HRP980265B1 (en) 2004-10-31
YU59599A (et) 2002-08-12
KR100521292B1 (ko) 2005-10-17
CA2289753C (en) 2007-01-23
GB2340491A (en) 2000-02-23
CN1150194C (zh) 2004-05-19
HRP980265A2 (en) 1999-02-28
JP3150711B2 (ja) 2001-03-26
TNSN98065A1 (fr) 2005-03-15
TR199902810T2 (xx) 2000-02-21
GB2340491B (en) 2000-10-18
SA98190179B1 (ar) 2006-08-15
UY25004A1 (es) 2000-10-31
DK0983271T3 (da) 2004-05-10
AR015668A1 (es) 2001-05-16
ES2214712T3 (es) 2004-09-16
UA56231C2 (uk) 2003-05-15
EG23836A (en) 2007-10-02
TW480259B (en) 2002-03-21
ID24910A (id) 2000-08-31
GB2348202A (en) 2000-09-27
MA26498A1 (fr) 2004-12-20
CN1515572A (zh) 2004-07-28
SK156199A3 (en) 2000-07-11
EA001809B1 (ru) 2001-08-27
HUP0002754A3 (en) 2003-01-28
ZA984083B (en) 1999-11-15
NZ500865A (en) 2001-04-27
ZA984085B (en) 2000-01-26
EP0983271A1 (en) 2000-03-08
CA2289753A1 (en) 1998-11-26
BRPI9809126B8 (pt) 2021-07-06
AP2009A (en) 2009-06-26
HN1998000071A (es) 1999-03-19
GB9709945D0 (en) 1997-07-09
SI0983271T1 (en) 2004-06-30
NO995622L (no) 2000-01-14
JO2032B1 (en) 1999-05-15
HUP0002754A2 (hu) 2001-06-28
US6294540B1 (en) 2001-09-25
EP0983271B1 (en) 2004-02-18
IL132793A0 (en) 2001-03-19
NO324731B1 (no) 2007-12-03
GB2348202B (en) 2001-08-08
NZ510622A (en) 2002-04-26
AP9901688A0 (en) 1999-12-31
IL132793A (en) 2006-10-31
PA8451301A1 (es) 2000-05-24
EA199900944A1 (ru) 2000-06-26
KR20010012623A (ko) 2001-02-26
IS2207B (is) 2007-02-15
OA11304A (en) 2003-10-22
AU7765598A (en) 1998-12-11
DE69821758D1 (de) 2004-03-25
MY120151A (en) 2005-09-30
BRPI9809126B1 (pt) 2018-02-06
CN100408580C (zh) 2008-08-06
PL336888A1 (en) 2000-07-17
SV1998000057A (es) 1999-03-02
CO4940435A1 (es) 2000-07-24
PL189527B1 (pl) 2005-08-31
GEP20022680B (en) 2002-04-25
JP2000514096A (ja) 2000-10-24
DZ2493A1 (fr) 2004-06-20
GB9926839D0 (en) 2000-01-12
PE78799A1 (es) 1999-08-31
SK285159B6 (sk) 2006-07-07
AU739953B2 (en) 2001-10-25
ATE259811T1 (de) 2004-03-15
NO995622D0 (no) 1999-11-16
HU226563B1 (en) 2009-04-28

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