EE9900147A - Oksadiasoolid, nende saamismeetodid ja kasutamine ravimitena - Google Patents

Oksadiasoolid, nende saamismeetodid ja kasutamine ravimitena

Info

Publication number
EE9900147A
EE9900147A EEP199900147A EE9900147A EE9900147A EE 9900147 A EE9900147 A EE 9900147A EE P199900147 A EEP199900147 A EE P199900147A EE 9900147 A EE9900147 A EE 9900147A EE 9900147 A EE9900147 A EE 9900147A
Authority
EE
Estonia
Prior art keywords
oxadiazoles
pharmaceuticals
preparation
methods
Prior art date
Application number
EEP199900147A
Other languages
English (en)
Estonian (et)
Inventor
Brenner Michael
Maier Roland
Wienrich Marion
Weiser Thomas
Palluk Rainer
Bechtel Wolf-Dietrich
Sagrada Angelo
Ensinger Helmut
Pschorn Uwe
Cesana Raffaele
Original Assignee
Boehringer Ingelheim Pharma Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma Kg filed Critical Boehringer Ingelheim Pharma Kg
Publication of EE9900147A publication Critical patent/EE9900147A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
EEP199900147A 1996-10-18 1997-10-15 Oksadiasoolid, nende saamismeetodid ja kasutamine ravimitena EE9900147A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19643037A DE19643037A1 (de) 1996-10-18 1996-10-18 Neue Oxadiazole, Verfahren zu ihrer Herstellung sowie deren Verwendung als Arzneimittel
PCT/EP1997/005693 WO1998017652A1 (de) 1996-10-18 1997-10-15 Oxadiazole, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
EE9900147A true EE9900147A (et) 1999-12-15

Family

ID=7809114

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900147A EE9900147A (et) 1996-10-18 1997-10-15 Oksadiasoolid, nende saamismeetodid ja kasutamine ravimitena

Country Status (32)

Country Link
US (1) US6277872B1 (bg)
EP (1) EP0934288B1 (bg)
JP (1) JP3333523B2 (bg)
KR (1) KR20000049253A (bg)
CN (1) CN1086698C (bg)
AR (1) AR008496A1 (bg)
AT (1) ATE315034T1 (bg)
AU (1) AU737552B2 (bg)
BG (1) BG103251A (bg)
BR (1) BR9714354A (bg)
CA (1) CA2268954C (bg)
CO (1) CO4920253A1 (bg)
CZ (1) CZ138099A3 (bg)
DE (2) DE19643037A1 (bg)
EE (1) EE9900147A (bg)
ES (1) ES2256880T3 (bg)
HK (1) HK1020956A1 (bg)
HR (1) HRP970553A2 (bg)
HU (1) HUP0001652A3 (bg)
ID (1) ID18613A (bg)
IL (1) IL129315A0 (bg)
NO (1) NO312512B1 (bg)
NZ (1) NZ335598A (bg)
PE (1) PE11199A1 (bg)
PL (1) PL332432A1 (bg)
RU (1) RU2182905C2 (bg)
SK (1) SK49999A3 (bg)
TR (1) TR199900848T2 (bg)
TW (1) TW413678B (bg)
WO (1) WO1998017652A1 (bg)
YU (1) YU40997A (bg)
ZA (1) ZA979220B (bg)

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IT1300056B1 (it) 1998-04-17 2000-04-05 Boehringer Ingelheim Italia Eterocicli con anello a 6 termini difenil-sostituiti loro procedimento di preparazione e loro impiego come farmaci
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WO2000047567A1 (fr) 1999-02-15 2000-08-17 Eisai Co., Ltd. Derives d'heterodiazinone
ATE257827T1 (de) 1999-07-21 2004-01-15 Hoffmann La Roche Triazolderivate
CZ2002599A3 (cs) * 1999-08-19 2002-06-12 Nps Pharmaceuticals Inc. Heteropolycyklické sloučeniny a jejich pouľití jako antagonistů metabotropního receptoru glutamátu
US6660753B2 (en) 1999-08-19 2003-12-09 Nps Pharmaceuticals, Inc. Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
EP1582519A3 (en) * 1999-08-19 2005-12-21 Nps Pharmaceuticals, Inc. Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
US6579880B2 (en) * 2000-06-06 2003-06-17 Ortho-Mcneil Pharmaceutical, Inc. Isoxazoles and oxadiazoles as anti-inflammatory inhibitors of IL-8
BRPI0111596B8 (pt) 2000-06-12 2022-07-26 Eisai Co Ltd Composto piridona, processo de produção do composto, composição farmacêutica, e uso do dito composto
CN100473647C (zh) * 2000-09-18 2009-04-01 卫材R&D管理有限公司 哒嗪酮和三嗪酮化合物及其作为药物制剂的用途
PT1379525E (pt) * 2001-02-21 2007-12-04 Astrazeneca Ab Compostos heteropolicíclicos e sua utilização como antagonistas dos receptores metabotrópicos de glutamato
AU2002341921B2 (en) * 2001-10-04 2007-05-31 Merck Sharp & Dohme Corp. Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
MY151199A (en) 2001-11-02 2014-04-30 Rigel Pharmaceuticals Inc Substituted diphenyl heterocycles useful for treating hcv infection
GB0129260D0 (en) 2001-12-06 2002-01-23 Eisai London Res Lab Ltd Pharmaceutical compositions and their uses
NZ537980A (en) 2002-08-23 2007-08-31 Rigel Pharmaceuticals Inc Pyridyl substituted heterocycles useful for treating or preventing HCV infection
GB0303503D0 (en) * 2003-02-14 2003-03-19 Novartis Ag Organic compounds
WO2004099165A2 (en) 2003-05-02 2004-11-18 Rigel Pharmaceuticals, Inc. Heterocyclic compounds and hydro isomers thereof
WO2004099164A1 (en) * 2003-05-02 2004-11-18 Rigel Pharmaceuticals, Inc. Substituted diphenyl isoxazoles, pyrazoles and oxadiazoles useful for treating hcv infection
US7220745B2 (en) 2003-05-15 2007-05-22 Rigel Pharmaceuticals Heterocyclic compounds useful to treat HCV
WO2005049065A2 (en) 2003-11-19 2005-06-02 Rigel Pharmaceuticals, Inc. Synergistic combinations of dihaloacetamide with interferon or ribavirin for treatment hcv infections
KR101154830B1 (ko) * 2003-12-24 2012-06-18 프로시디온 리미티드 Gpcr 수용체 효능제로서의 헤테로사이클릭 유도체
US7514434B2 (en) 2004-02-23 2009-04-07 Rigel Pharmaceuticals, Inc. Heterocyclic compounds having an oxadiazole moiety and hydro isomers thereof
MY148809A (en) 2004-07-06 2013-05-31 Eisai R&D Man Co Ltd Crystals of 1,2-dihydropyridine compound and their production process
EP1875912A4 (en) * 2005-04-08 2008-06-04 Eisai R&D Man Co Ltd MEANS OF TREATING UNWILLING MOVEMENTS
CA2606106A1 (en) 2005-05-02 2007-03-08 Rigel Pharmaceuticals, Inc. Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses
GB0510142D0 (en) * 2005-05-18 2005-06-22 Addex Pharmaceuticals Sa Novel compounds A1
HUP0500920A2 (en) * 2005-10-05 2007-07-30 Richter Gedeon Nyrt Oxadiazole derivatives, process for their preparation and their use
AU2007334436A1 (en) * 2006-12-15 2008-06-26 Abbott Laboratories Novel oxadiazole compounds
US20110207704A1 (en) * 2006-12-15 2011-08-25 Abbott Laboratories Novel Oxadiazole Compounds
JO2701B1 (en) 2006-12-21 2013-03-03 جلاكسو جروب ليميتد Vehicles
EP2193126B1 (en) * 2007-10-04 2015-06-24 Merck Serono S.A. Oxadiazole diaryl compounds
US9045442B2 (en) * 2007-12-21 2015-06-02 University Of Notre Dame Du Lac Antibacterial compounds and methods of using same
TR201904041T4 (tr) 2008-06-09 2019-04-22 Max Planck Gesellschaft Protein agregasyonu ile bağlantılı hastalıklarda ve/veya nörodejeneratif hastalıklarda rol oynayan proteinlerin agregasyonunu inhibe etmeye yönelik ilaçlar.
WO2011047129A1 (en) 2009-10-15 2011-04-21 Southern Research Institute Treatment of neurodegenerative diseases, causation of memory enhancement, and assay for screening compounds for such
CN104768949A (zh) * 2012-08-24 2015-07-08 特温蒂斯公司 苯并呋咱抗淀粉样蛋白化合物和方法
ES2734432T3 (es) 2014-02-27 2019-12-05 Treventis Corp Compuestos antiamiloides que contienen benzofurazano
BR112016022451B1 (pt) 2014-04-24 2021-03-30 Sumitomo Chemical Company, Limited Composto de diaril-azol e agente de controle de peste artrópoda
WO2016049586A2 (en) * 2014-09-25 2016-03-31 University Of Notre Dame Du Lac Non-beta lactam antibiotics
CN107286174B (zh) * 2016-04-11 2020-08-18 上海勋和医药科技有限公司 取代2,4-(1h,3h)嘧啶二酮作为parp抑制剂及其应用
WO2018049404A1 (en) 2016-09-12 2018-03-15 University Of Notre Dame Du Lac Compounds for the treatment of clostridium difficile infection
AU2018265584B2 (en) 2017-05-12 2023-09-28 Ludwig-Maximilians-Universität München Phenyl-heterocycle-phenyl derivatives for use in the treatment or prevention of melanoma
US10676467B2 (en) 2017-06-30 2020-06-09 Washington University Compositions for binding sphingosine-1-phosphate receptor 1 (S1P1), imaging of S1P1, and methods of use thereof
JP7177937B2 (ja) 2018-12-14 2022-11-24 エーザイ・アール・アンド・ディー・マネジメント株式会社 1,2-ジヒドロピリジン化合物の水性医薬製剤
WO2023042888A1 (ja) 2021-09-15 2023-03-23 国立大学法人 琉球大学 認知機能低下、または過体重もしくは肥満症を処置することに用いるための医薬組成物
WO2023042887A1 (ja) 2021-09-15 2023-03-23 国立大学法人 琉球大学 認知機能低下、または過体重もしくは肥満症を処置することに用いるための医薬組成物
EP4173485A1 (en) 2021-10-27 2023-05-03 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Protein aggregation inhibiting compounds for plant disease control

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US4003909A (en) * 1974-07-22 1977-01-18 E. R. Squibb & Sons, Inc. [(1,2,4-Oxadiazol-3-yl)phenyl]carbamic or thiocarbamic acid esters
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Also Published As

Publication number Publication date
ES2256880T3 (es) 2006-07-16
HUP0001652A2 (hu) 2001-01-29
HRP970553A2 (en) 1998-08-31
AU737552B2 (en) 2001-08-23
ATE315034T1 (de) 2006-02-15
IL129315A0 (en) 2000-02-17
DE59712543D1 (de) 2006-03-30
RU2182905C2 (ru) 2002-05-27
SK49999A3 (en) 1999-11-08
TW413678B (en) 2000-12-01
NO991815D0 (no) 1999-04-16
CA2268954C (en) 2006-06-13
NO312512B1 (no) 2002-05-21
PE11199A1 (es) 1999-03-03
WO1998017652A1 (de) 1998-04-30
CN1086698C (zh) 2002-06-26
EP0934288B1 (de) 2006-01-04
AR008496A1 (es) 2000-01-19
TR199900848T2 (xx) 1999-06-21
CO4920253A1 (es) 2000-05-29
ID18613A (id) 1998-04-23
NZ335598A (en) 2001-06-29
HK1020956A1 (en) 2000-05-26
AU4867697A (en) 1998-05-15
US6277872B1 (en) 2001-08-21
KR20000049253A (ko) 2000-07-25
JP3333523B2 (ja) 2002-10-15
PL332432A1 (en) 1999-09-13
CZ138099A3 (cs) 1999-11-17
ZA979220B (en) 1998-04-20
BG103251A (bg) 2000-02-29
HUP0001652A3 (en) 2002-12-28
DE19643037A1 (de) 1998-04-23
NO991815L (no) 1999-04-16
YU40997A (sh) 2000-10-30
CA2268954A1 (en) 1998-04-30
CN1233245A (zh) 1999-10-27
JP2000505089A (ja) 2000-04-25
EP0934288A1 (de) 1999-08-11
BR9714354A (pt) 2000-04-11

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