EA202191478A1 - Гетероароматические соединения в качестве ингибиторов ванина - Google Patents
Гетероароматические соединения в качестве ингибиторов ванинаInfo
- Publication number
- EA202191478A1 EA202191478A1 EA202191478A EA202191478A EA202191478A1 EA 202191478 A1 EA202191478 A1 EA 202191478A1 EA 202191478 A EA202191478 A EA 202191478A EA 202191478 A EA202191478 A EA 202191478A EA 202191478 A1 EA202191478 A1 EA 202191478A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- heteroaromatic compounds
- vanin
- compounds
- inhibitors
- vanin inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
- C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862774412P | 2018-12-03 | 2018-12-03 | |
PCT/EP2019/083259 WO2020114947A1 (en) | 2018-12-03 | 2019-12-02 | Heteroaromatic compounds as vanin inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
EA202191478A1 true EA202191478A1 (ru) | 2021-10-26 |
Family
ID=68766765
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202191478A EA202191478A1 (ru) | 2018-12-03 | 2019-12-02 | Гетероароматические соединения в качестве ингибиторов ванина |
Country Status (11)
Country | Link |
---|---|
US (1) | US20220048889A1 (ko) |
EP (1) | EP3890828A1 (ko) |
JP (1) | JP7195436B2 (ko) |
KR (1) | KR20210099093A (ko) |
CN (1) | CN113226462A (ko) |
AU (1) | AU2019392524A1 (ko) |
BR (1) | BR112021010823A2 (ko) |
CA (1) | CA3120037A1 (ko) |
EA (1) | EA202191478A1 (ko) |
MX (1) | MX2021006489A (ko) |
WO (1) | WO2020114947A1 (ko) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA202191476A1 (ru) * | 2018-12-03 | 2021-10-26 | Бёрингер Ингельхайм Интернациональ Гмбх | Гетероароматические соединения в качестве ингибиторов ванина |
CN113412113A (zh) * | 2018-12-11 | 2021-09-17 | 豪夫迈·罗氏有限公司 | 氨基嗪酰胺 |
IL301556A (en) * | 2020-09-25 | 2023-05-01 | Shanghai Meiyue Biotech Dev Co Ltd | Pyrimidine carboxamide compound and its use |
TWI811901B (zh) * | 2020-12-17 | 2023-08-11 | 大陸商上海美悅生物科技發展有限公司 | 一種嘧啶甲醯胺類化合物及其應用 |
WO2023174409A1 (zh) * | 2022-03-18 | 2023-09-21 | 上海美悦生物科技发展有限公司 | Vanin酶抑制剂的盐型、晶型及其制备方法和应用 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2987179C (en) * | 2015-05-29 | 2020-08-25 | Pfizer Inc. | Heterocyclic compounds as inhibitors of vanin-1 enzyme |
EP3484876A1 (en) * | 2016-07-14 | 2019-05-22 | Pfizer Inc | Novel pyrimidine carboxamides as inhibitors of vanin-1 enzyme |
EA202191476A1 (ru) * | 2018-12-03 | 2021-10-26 | Бёрингер Ингельхайм Интернациональ Гмбх | Гетероароматические соединения в качестве ингибиторов ванина |
-
2019
- 2019-12-02 US US17/299,148 patent/US20220048889A1/en active Pending
- 2019-12-02 EP EP19813499.1A patent/EP3890828A1/en active Pending
- 2019-12-02 JP JP2021531394A patent/JP7195436B2/ja active Active
- 2019-12-02 CA CA3120037A patent/CA3120037A1/en active Pending
- 2019-12-02 BR BR112021010823-8A patent/BR112021010823A2/pt unknown
- 2019-12-02 CN CN201980079064.6A patent/CN113226462A/zh active Pending
- 2019-12-02 WO PCT/EP2019/083259 patent/WO2020114947A1/en unknown
- 2019-12-02 MX MX2021006489A patent/MX2021006489A/es unknown
- 2019-12-02 EA EA202191478A patent/EA202191478A1/ru unknown
- 2019-12-02 KR KR1020217020909A patent/KR20210099093A/ko unknown
- 2019-12-02 AU AU2019392524A patent/AU2019392524A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
MX2021006489A (es) | 2021-07-06 |
CN113226462A (zh) | 2021-08-06 |
BR112021010823A2 (pt) | 2021-08-24 |
US20220048889A1 (en) | 2022-02-17 |
EP3890828A1 (en) | 2021-10-13 |
CA3120037A1 (en) | 2020-06-11 |
JP7195436B2 (ja) | 2022-12-23 |
KR20210099093A (ko) | 2021-08-11 |
WO2020114947A1 (en) | 2020-06-11 |
JP2022510351A (ja) | 2022-01-26 |
AU2019392524A1 (en) | 2021-07-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PH12021551065A1 (en) | Fused ring compounds | |
EA201792047A1 (ru) | Новые соединения | |
EA201891494A1 (ru) | Гетероциклические соединения в качестве иммуномодуляторов | |
EA201790492A1 (ru) | СОЕДИНЕНИЯ, КОТОРЫЕ ИНГИБИРУЮТ БЕЛОК Mcl-1 | |
EA202191478A1 (ru) | Гетероароматические соединения в качестве ингибиторов ванина | |
EA202190588A1 (ru) | Гетероароматические соединения в качестве ингибиторов ванина | |
TR201819138T4 (tr) | FGFR Kinaz Modülatörleri Olarak Faydalı Kinoksalin Türevleri | |
EA201592068A1 (ru) | Ингибиторы энхансера zeste гомолога 2 | |
EA201891063A1 (ru) | Производные дигидроимидазопиразинона, применимые в лечении рака | |
EA201792421A1 (ru) | Амидозамещенные производные циклогексана | |
MY197440A (en) | Heteroamatic compounds as btk inhibitors | |
EA202191476A1 (ru) | Гетероароматические соединения в качестве ингибиторов ванина | |
EA202090014A1 (ru) | Гетероароматические соединения в качестве ингибиторов ванина | |
EA201790949A1 (ru) | Замещенные 2,4-диаминохинолины в качестве новых противораковых средств | |
EA201990400A1 (ru) | Соединения и композиции и их применение | |
EA201692481A1 (ru) | Комбинация, содержащая глюкокортикоид и edo-s101 | |
EA202090414A1 (ru) | Соединения и их применение | |
EA201790070A1 (ru) | Бифениламиды, содержащие модифицированные простые эфирные группы, в качестве ингибиторов hsp90 и стимуляторов hsp70 | |
EA202090448A1 (ru) | Дигидрооксадиазиноны | |
EA201792341A1 (ru) | Производные пиразола, пригодные в качестве ингибиторов белка, активирующего 5-липоксигеназу (flap) | |
EA201501187A1 (ru) | Новые химические соединения (варианты) и их применение для лечения онкологических заболеваний | |
EA201791432A1 (ru) | Композиции на основе пролекарства монометилфумарата | |
EA202091003A1 (ru) | Новые производные пиразолопирролопиримидиндиона в качестве ингибиторов p2x3 | |
EA202191477A1 (ru) | Гетероароматические соединения в качестве ингибиторов ванина | |
EA201990947A1 (ru) | Замещенные производные 6-(1h-пиразол-1-ил)пиримидин-4-амина и их применение |