EA201692532A1 - Антимикробные композиции с шипучими веществами - Google Patents

Антимикробные композиции с шипучими веществами

Info

Publication number
EA201692532A1
EA201692532A1 EA201692532A EA201692532A EA201692532A1 EA 201692532 A1 EA201692532 A1 EA 201692532A1 EA 201692532 A EA201692532 A EA 201692532A EA 201692532 A EA201692532 A EA 201692532A EA 201692532 A1 EA201692532 A1 EA 201692532A1
Authority
EA
Eurasian Patent Office
Prior art keywords
compositions
substances
pipe
antimicrobial compositions
quinolone
Prior art date
Application number
EA201692532A
Other languages
English (en)
Other versions
EA034152B1 (ru
Inventor
Даньпин Ли
Original Assignee
Мелинта Терапьютикс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54868661&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201692532(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Мелинта Терапьютикс, Инк. filed Critical Мелинта Терапьютикс, Инк.
Publication of EA201692532A1 publication Critical patent/EA201692532A1/ru
Publication of EA034152B1 publication Critical patent/EA034152B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007—Effervescent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/133—Amines having hydroxy groups, e.g. sphingosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Quinoline Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Настоящее изобретение относится к фармацевтическим композициям, включающим антимикробное соединение, представляющее собой производное хинолон-карбоновой кислоты, и шипучее вещество. Эти композиции обладают улучшенной желудочно-кишечной переносимостью и/или пониженным потенциалом индукции желудочно-кишечных побочных эффектов. Эти композиции являются полезными для перорального введения для лечения, профилактики или снижения риска микробных инфекций.
EA201692532A 2014-06-20 2015-06-19 Антимикробные композиции с шипучими веществами EA034152B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462014786P 2014-06-20 2014-06-20
PCT/US2015/036605 WO2015196027A1 (en) 2014-06-20 2015-06-19 Antimicrobial compositions with effervescent agents

Publications (2)

Publication Number Publication Date
EA201692532A1 true EA201692532A1 (ru) 2017-05-31
EA034152B1 EA034152B1 (ru) 2020-01-09

Family

ID=54868661

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201692532A EA034152B1 (ru) 2014-06-20 2015-06-19 Антимикробные композиции с шипучими веществами

Country Status (31)

Country Link
US (2) US20150366857A1 (ru)
EP (3) EP3581180B1 (ru)
JP (2) JP6995479B2 (ru)
CN (2) CN114831955B (ru)
AR (1) AR100920A1 (ru)
AU (3) AU2015276954B2 (ru)
BR (1) BR112016029761B1 (ru)
CA (1) CA2952950C (ru)
CL (2) CL2016003273A1 (ru)
CR (2) CR20160592A (ru)
CY (2) CY1121995T1 (ru)
DK (2) DK3157510T3 (ru)
EA (1) EA034152B1 (ru)
EC (1) ECSP16095540A (ru)
ES (2) ES2732865T3 (ru)
HR (2) HRP20211685T1 (ru)
HU (2) HUE056298T2 (ru)
IL (1) IL249622A0 (ru)
LT (2) LT3581180T (ru)
MX (2) MX368940B (ru)
PE (2) PE20210927A1 (ru)
PH (1) PH12016502548A1 (ru)
PL (2) PL3157510T3 (ru)
PT (2) PT3581180T (ru)
RS (2) RS62538B1 (ru)
SI (2) SI3157510T1 (ru)
SV (1) SV2016005349A (ru)
TR (1) TR201909417T4 (ru)
TW (2) TWI705814B (ru)
UY (1) UY36184A (ru)
WO (1) WO2015196027A1 (ru)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022240897A1 (en) * 2021-05-10 2022-11-17 Sepelo Therapeutics, Llc Pharmaceutical composition comprising delafloxacin for administration into the lung

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GB9402203D0 (en) * 1994-02-04 1994-03-30 Smithkline Beecham Plc Pharmaceutical formulation
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EA004443B1 (ru) 1998-09-14 2004-04-29 Рэнбакси Лабораториз Лимитед Лекарственная форма для контролируемого высвобождения ципрофлоксацина для приема один раз в день
US6187317B1 (en) * 1999-07-14 2001-02-13 Judith Taylor Natural anti-diarrheal composition and method
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Also Published As

Publication number Publication date
PL3157510T3 (pl) 2019-12-31
RS59064B1 (sr) 2019-08-30
NZ727638A (en) 2023-08-25
CA2952950C (en) 2023-11-14
MX368940B (es) 2019-10-21
EP3157510A1 (en) 2017-04-26
AU2015276954A1 (en) 2017-01-12
CN114831955B (zh) 2024-03-12
SI3157510T1 (sl) 2019-09-30
CN106572982B9 (zh) 2022-07-08
BR112016029761A2 (pt) 2017-08-22
DK3581180T3 (da) 2021-11-08
JP2020183415A (ja) 2020-11-12
CR20160592A (es) 2017-02-21
TW201625249A (zh) 2016-07-16
EP3581180A1 (en) 2019-12-18
ES2897576T3 (es) 2022-03-01
PL3581180T3 (pl) 2022-02-07
AU2020256457B2 (en) 2021-09-30
RS62538B1 (sr) 2021-12-31
DK3157510T3 (da) 2019-07-01
SI3581180T1 (sl) 2021-12-31
UY36184A (es) 2016-01-29
US20150366857A1 (en) 2015-12-24
MX2019012608A (es) 2019-12-02
CL2020003153A1 (es) 2021-06-25
CA2952950A1 (en) 2015-12-23
EP3157510A4 (en) 2018-02-21
ES2732865T3 (es) 2019-11-26
CY1121995T1 (el) 2020-10-14
EP3919057A1 (en) 2021-12-08
EA034152B1 (ru) 2020-01-09
AU2015276954B2 (en) 2020-07-23
JP6995479B2 (ja) 2022-01-14
CY1125395T1 (el) 2023-03-24
HRP20191133T1 (hr) 2019-09-20
PT3581180T (pt) 2021-11-09
SV2016005349A (es) 2017-08-31
ECSP16095540A (es) 2017-03-31
CN106572982A (zh) 2017-04-19
HRP20211685T1 (hr) 2022-02-04
AU2021286284A1 (en) 2022-01-06
AU2021286284B2 (en) 2024-02-29
MX2016017350A (es) 2017-04-06
CR20200565A (es) 2021-01-14
HUE056298T2 (hu) 2022-02-28
HUE044764T2 (hu) 2019-11-28
PE20210927A1 (es) 2021-05-19
IL249622A0 (en) 2017-02-28
TWI732337B (zh) 2021-07-01
EP3157510B1 (en) 2019-03-27
EP3581180B1 (en) 2021-08-04
AU2020256457A1 (en) 2020-11-12
CN106572982B (zh) 2022-06-03
TWI705814B (zh) 2020-10-01
CN114831955A (zh) 2022-08-02
JP7149991B2 (ja) 2022-10-07
BR112016029761B1 (pt) 2023-03-07
WO2015196027A1 (en) 2015-12-23
CL2016003273A1 (es) 2017-08-04
JP2017518349A (ja) 2017-07-06
US20200237744A1 (en) 2020-07-30
BR112016029761A8 (pt) 2021-06-29
LT3581180T (lt) 2021-12-27
TW202005650A (zh) 2020-02-01
PT3157510T (pt) 2019-06-21
PE20170304A1 (es) 2017-04-19
TR201909417T4 (tr) 2019-07-22
LT3157510T (lt) 2019-09-25
PH12016502548A1 (en) 2017-04-10
AR100920A1 (es) 2016-11-09

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