EA201690219A1 - Агонисты рецептора вазопрессина-2 - Google Patents

Агонисты рецептора вазопрессина-2

Info

Publication number
EA201690219A1
EA201690219A1 EA201690219A EA201690219A EA201690219A1 EA 201690219 A1 EA201690219 A1 EA 201690219A1 EA 201690219 A EA201690219 A EA 201690219A EA 201690219 A EA201690219 A EA 201690219A EA 201690219 A1 EA201690219 A1 EA 201690219A1
Authority
EA
Eurasian Patent Office
Prior art keywords
receptor agonists
vazopressina
nocturia
vasopressin
treatment
Prior art date
Application number
EA201690219A
Other languages
English (en)
Other versions
EA029392B1 (ru
Inventor
Казимеж ВИСНЕВСКИ
Клаудио Штайнгарт
Пьер РИВЬЕР
Original Assignee
Ферринг Б.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ферринг Б.В. filed Critical Ферринг Б.В.
Publication of EA201690219A1 publication Critical patent/EA201690219A1/ru
Publication of EA029392B1 publication Critical patent/EA029392B1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/10Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/16Oxytocins; Vasopressins; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Cell Biology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Epidemiology (AREA)

Abstract

Агонисты рецептора вазопрессина-2, их фармацевтические композиции и способы применения вышеуказанных для лечения несахарного диабета, первичного ночного энуреза и никтурии.
EA201690219A 2013-07-26 2014-07-25 Агонисты рецептора вазопрессина-2 EA029392B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361859024P 2013-07-26 2013-07-26
US201461952073P 2014-03-12 2014-03-12
PCT/US2014/048317 WO2015013690A1 (en) 2013-07-26 2014-07-25 Vasopressin-2 receptor agonists

Publications (2)

Publication Number Publication Date
EA201690219A1 true EA201690219A1 (ru) 2016-11-30
EA029392B1 EA029392B1 (ru) 2018-03-30

Family

ID=51398870

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201690219A EA029392B1 (ru) 2013-07-26 2014-07-25 Агонисты рецептора вазопрессина-2

Country Status (28)

Country Link
US (2) US10131692B2 (ru)
EP (1) EP3024829B1 (ru)
JP (1) JP6387095B2 (ru)
KR (1) KR102198130B1 (ru)
CN (1) CN105492441B (ru)
AU (1) AU2014292860B2 (ru)
BR (1) BR112016000436B1 (ru)
CA (1) CA2919208A1 (ru)
DK (1) DK3024829T3 (ru)
EA (1) EA029392B1 (ru)
ES (1) ES2656039T3 (ru)
HK (1) HK1218647A1 (ru)
HR (1) HRP20180009T1 (ru)
HU (1) HUE035252T2 (ru)
IL (1) IL243730B (ru)
JO (1) JO3371B1 (ru)
LT (1) LT3024829T (ru)
MX (1) MX363355B (ru)
MY (1) MY183429A (ru)
PH (1) PH12016500044A1 (ru)
PL (1) PL3024829T3 (ru)
PT (1) PT3024829T (ru)
RS (1) RS56604B1 (ru)
SG (1) SG11201600031RA (ru)
SI (1) SI3024829T1 (ru)
TW (1) TWI640542B (ru)
WO (1) WO2015013690A1 (ru)
ZA (1) ZA201600145B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2343982B1 (en) 2008-09-17 2017-03-22 Chiasma Inc. Pharmaceutical compositions and related methods of delivery
MA46586A (fr) 2016-10-21 2019-08-28 Chiasma Inc Compositions de terlipressine et leurs procédés d'utilisation

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE399252B (sv) * 1976-05-24 1978-02-06 Ferring Ab Forfarande for framstellnign av antidiuretiskt verkande desamino-asparagin Ÿ4-d-argininŸ8-vasopressin
CA1246055A (en) * 1980-03-24 1988-12-06 Joseph H. Cort N-.omega.-substituted hormonogens of vasopressin and its synthetic analogs
DK153883A (da) 1982-04-20 1983-10-21 Ceskoslovenska Akademie Ved Vasopressin-analoge
SE501677C2 (sv) * 1993-06-18 1995-04-10 Ferring Bv Biologiskt aktiva vasopressinanaloger, farmaceutiska preparat innehållande dem samt deras användning för framställning av läkemedel
US5500413A (en) * 1993-06-29 1996-03-19 Ferring Ab Process for manufacture of 1-deamino-8-D-arginine vasopressin
CZ292131B6 (cs) 2000-02-16 2003-08-13 Ústav organické chemie a biochemie AV ČR Synthetické analogy Desmopressinu chráněné v C-terminální sekvenci proti karboxyamidasovému štěpení

Also Published As

Publication number Publication date
EA029392B1 (ru) 2018-03-30
PL3024829T3 (pl) 2018-04-30
AU2014292860A1 (en) 2016-01-28
IL243730B (en) 2019-09-26
RS56604B1 (sr) 2018-02-28
PH12016500044B1 (en) 2016-03-28
TWI640542B (zh) 2018-11-11
CA2919208A1 (en) 2015-01-29
KR20160034943A (ko) 2016-03-30
WO2015013690A1 (en) 2015-01-29
SG11201600031RA (en) 2016-02-26
MX363355B (es) 2019-03-21
PT3024829T (pt) 2017-12-18
TW201536815A (zh) 2015-10-01
HRP20180009T1 (hr) 2018-02-09
IL243730A0 (en) 2016-04-21
US10131692B2 (en) 2018-11-20
NZ716342A (en) 2021-03-26
US20190194257A1 (en) 2019-06-27
JP6387095B2 (ja) 2018-09-05
EP3024829A1 (en) 2016-06-01
CN105492441A (zh) 2016-04-13
HUE035252T2 (en) 2018-05-02
CN105492441B (zh) 2019-09-10
JP2016527255A (ja) 2016-09-08
KR102198130B1 (ko) 2021-01-05
ZA201600145B (en) 2020-01-29
DK3024829T3 (en) 2017-12-04
JO3371B1 (ar) 2019-03-13
HK1218647A1 (zh) 2017-03-03
MX2016000525A (es) 2016-04-07
LT3024829T (lt) 2017-12-27
US10745443B2 (en) 2020-08-18
SI3024829T1 (en) 2018-01-31
US20150307555A1 (en) 2015-10-29
AU2014292860B2 (en) 2017-10-05
BR112016000436A2 (ru) 2017-07-25
MY183429A (en) 2021-02-18
PH12016500044A1 (en) 2016-03-28
ES2656039T3 (es) 2018-02-22
BR112016000436B1 (pt) 2022-07-05
EP3024829B1 (en) 2017-11-08

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): TJ TM