EA201290165A1 - Способ получения производного фенилаланина - Google Patents

Способ получения производного фенилаланина

Info

Publication number
EA201290165A1
EA201290165A1 EA201290165A EA201290165A EA201290165A1 EA 201290165 A1 EA201290165 A1 EA 201290165A1 EA 201290165 A EA201290165 A EA 201290165A EA 201290165 A EA201290165 A EA 201290165A EA 201290165 A1 EA201290165 A1 EA 201290165A1
Authority
EA
Eurasian Patent Office
Prior art keywords
fenilalanine
derivatives
producing
obtaining
formula
Prior art date
Application number
EA201290165A
Other languages
English (en)
Inventor
Джозеф Пол Адамс
Тору Курода
Хироаки Мацумае
Джон Брайс Страчан
Нобухиро Яги
Original Assignee
Глаксо Груп Лимитед
Мицубиси Танабе Фарма Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глаксо Груп Лимитед, Мицубиси Танабе Фарма Корпорейшн filed Critical Глаксо Груп Лимитед
Publication of EA201290165A1 publication Critical patent/EA201290165A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/22—Separation; Purification; Stabilisation; Use of additives
    • C07C231/24—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Новый способ получения производного фенилаланина формулы (I)
EA201290165A 2009-10-21 2010-10-19 Способ получения производного фенилаланина EA201290165A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25363809P 2009-10-21 2009-10-21
PCT/EP2010/065710 WO2011048091A1 (en) 2009-10-21 2010-10-19 Process for preparing a phenylalanine derivative

Publications (1)

Publication Number Publication Date
EA201290165A1 true EA201290165A1 (ru) 2012-11-30

Family

ID=43094582

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201290165A EA201290165A1 (ru) 2009-10-21 2010-10-19 Способ получения производного фенилаланина

Country Status (13)

Country Link
US (1) US20120203023A1 (ru)
EP (1) EP2491006A1 (ru)
JP (1) JP2013508333A (ru)
KR (1) KR20120107461A (ru)
CN (1) CN102686557A (ru)
AU (1) AU2010309891A1 (ru)
BR (1) BR112012009292A2 (ru)
CA (1) CA2777158A1 (ru)
EA (1) EA201290165A1 (ru)
IL (1) IL218932A0 (ru)
MX (1) MX2012004707A (ru)
WO (1) WO2011048091A1 (ru)
ZA (1) ZA201202722B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013010679A1 (en) 2011-07-15 2013-01-24 Novartis Ag Salts of aza-bicyclic di-aryl ethers and methods to make them or their precursors
JP6254088B2 (ja) 2011-10-17 2017-12-27 バイオセリックス， インコーポレイテッド 置換ビアリールアルキルアミド
US11224600B2 (en) 2018-10-30 2022-01-18 Gilead Sciences, Inc. Compounds for inhibition of alpha 4 beta 7 integrin
CA3114240C (en) 2018-10-30 2023-09-05 Gilead Sciences, Inc. Imidazopyridine derivatives as alpha4beta7 integrin inhibitors
WO2020092401A1 (en) 2018-10-30 2020-05-07 Gilead Sciences, Inc. COMPOUNDS FOR INHIBITION OF ALPHA 4β7 INTEGRIN
EP3873884A1 (en) 2018-10-30 2021-09-08 Gilead Sciences, Inc. Quinoline derivatives as alpha4beta7 integrin inhibitors
JP7491996B2 (ja) 2019-08-14 2024-05-28 ギリアード サイエンシーズ， インコーポレイテッド α４β７インテグリンの阻害のための化合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20020169157A1 (en) 2000-08-29 2002-11-14 Gang Liu Selective protein tyrosine phosphatatase inhibitors
MY129000A (en) * 2000-08-31 2007-03-30 Tanabe Seiyaku Co INHIBITORS OF a4 MEDIATED CELL ADHESION
MY140707A (en) * 2002-02-28 2010-01-15 Mitsubishi Tanabe Pharma Corp Process for preparing a phenylalanine derivative and intermediates thereof
JP4258227B2 (ja) * 2002-02-28 2009-04-30 田辺三菱製薬株式会社 フェニルアラニン誘導体の製法およびその合成中間体

Also Published As

Publication number Publication date
MX2012004707A (es) 2012-06-08
US20120203023A1 (en) 2012-08-09
ZA201202722B (en) 2013-09-25
KR20120107461A (ko) 2012-10-02
WO2011048091A1 (en) 2011-04-28
EP2491006A1 (en) 2012-08-29
JP2013508333A (ja) 2013-03-07
CN102686557A (zh) 2012-09-19
BR112012009292A2 (pt) 2017-06-06
CA2777158A1 (en) 2011-04-28
AU2010309891A1 (en) 2012-05-17
IL218932A0 (en) 2012-07-31

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