EA201270826A1 - Стабилизированное активное соединение - Google Patents
Стабилизированное активное соединениеInfo
- Publication number
- EA201270826A1 EA201270826A1 EA201270826A EA201270826A EA201270826A1 EA 201270826 A1 EA201270826 A1 EA 201270826A1 EA 201270826 A EA201270826 A EA 201270826A EA 201270826 A EA201270826 A EA 201270826A EA 201270826 A1 EA201270826 A1 EA 201270826A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- active connection
- stabilized active
- carrier
- vitamin
- solubility
- Prior art date
Links
- 239000004480 active ingredient Substances 0.000 abstract 1
- 229910000389 calcium phosphate Inorganic materials 0.000 abstract 1
- 239000001506 calcium phosphate Substances 0.000 abstract 1
- 235000011010 calcium phosphates Nutrition 0.000 abstract 1
- 230000002209 hydrophobic effect Effects 0.000 abstract 1
- 239000008247 solid mixture Substances 0.000 abstract 1
- 239000003381 stabilizer Substances 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical group [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 abstract 1
- 150000003710 vitamin D derivatives Chemical class 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/158—Fatty acids; Fats; Products containing oils or fats
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/10—Organic substances
- A23K20/174—Vitamins
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/20—Inorganic substances, e.g. oligoelements
- A23K20/24—Compounds of alkaline earth metals, e.g. magnesium
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K20/00—Accessory food factors for animal feeding-stuffs
- A23K20/20—Inorganic substances, e.g. oligoelements
- A23K20/26—Compounds containing phosphorus
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23K—FODDER
- A23K40/00—Shaping or working-up of animal feeding-stuffs
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23L—FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
- A23L33/00—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
- A23L33/10—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
- A23L33/15—Vitamins
- A23L33/155—Vitamins A or D
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/59—Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
- A61K31/593—9,10-Secocholestane derivatives, e.g. cholecalciferol, i.e. vitamin D3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/143—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23V—INDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
- A23V2002/00—Food compositions, function of food ingredients or processes for food or foodstuffs
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Polymers & Plastics (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- Zoology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Animal Husbandry (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Physical Education & Sports Medicine (AREA)
- Nutrition Science (AREA)
- Mycology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fodder In General (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Настоящее изобретение относится к стабильным твердым композициям, содержащим первый носитель и адсорбируемое вещество, содержащее по меньшей мере один активный компонент, такой как производное витамина D, и его гидрофобный стабилизатор, отличающимся тем, что указанный первый носитель представляет собой кальция фосфат или его производные с растворимостью в воде меньше чем 0,1 вес.% при комнатной температуре.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP2010059014 | 2010-06-24 | ||
PCT/EP2011/060618 WO2011161236A1 (en) | 2010-06-24 | 2011-06-24 | Stabilized active compound |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201270826A1 true EA201270826A1 (ru) | 2013-05-30 |
EA022768B1 EA022768B1 (ru) | 2016-02-29 |
Family
ID=42537837
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201270826A EA022768B1 (ru) | 2010-06-24 | 2011-06-24 | Стабильная твердая композиция для пищевых, кормовых, косметических или фармацевтических препаратов и способ ее получения |
Country Status (11)
Country | Link |
---|---|
US (1) | US9757331B2 (ru) |
JP (1) | JP5817067B2 (ru) |
CN (1) | CN102958377A (ru) |
BR (1) | BR112012030239A2 (ru) |
CA (1) | CA2798019A1 (ru) |
EA (1) | EA022768B1 (ru) |
ES (1) | ES2725202T3 (ru) |
MX (1) | MX2012014872A (ru) |
TR (1) | TR201906042T4 (ru) |
UA (1) | UA107599C2 (ru) |
WO (1) | WO2011161236A1 (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP6171333B2 (ja) * | 2012-12-26 | 2017-08-02 | 東ソー株式会社 | 安定化したビタミンd類標準液 |
US9801821B2 (en) | 2013-03-27 | 2017-10-31 | Psm Healthcare Limited | Stabilized vitamin D formulations |
US10336817B2 (en) | 2016-10-14 | 2019-07-02 | Sultan Qaboos University | Therapeutic composition of camel milk |
DK3662761T3 (da) * | 2018-12-04 | 2021-07-26 | Dsm Ip Assets Bv | Opbevaringsstabile adsorbater af nitrooxyforbindelser |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB405791A (en) | 1933-01-14 | 1934-02-15 | Bell And Sons Ltd | Improvements in and relating to the manufacture of food accessories for cattle |
US4389419A (en) | 1980-11-10 | 1983-06-21 | Damon Corporation | Vitamin encapsulation |
JPH085782B2 (ja) * | 1989-04-14 | 1996-01-24 | 株式会社サンギ | ハイドロキシアパタイト抗菌剤及びその製造法 |
DE19710054A1 (de) | 1997-03-12 | 1998-09-17 | Merck Patent Gmbh | Pharmazeutische Zubereitung |
US5820903A (en) | 1997-06-30 | 1998-10-13 | General Mills, Inc. | Calcium fortified yogurt and methods of preparation |
US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
JP2002080358A (ja) * | 2000-09-07 | 2002-03-19 | Noevir Co Ltd | 皮膚外用剤 |
WO2003013270A2 (en) | 2001-08-09 | 2003-02-20 | Rhodia Inc. | Calcium dietary supplement |
US7632518B2 (en) | 2002-01-15 | 2009-12-15 | Dsm Ip Assets B.V. | 25-hydroxy vitamin D3 compositions |
DE10311585A1 (de) * | 2003-03-14 | 2004-09-23 | Basf Ag | Wirkstoffhaltige Adsorbate |
US20100143481A1 (en) * | 2006-11-08 | 2010-06-10 | Dinesh Shenoy | Method of preparing solid dosage forms of multi-phasic pharmaceutical compositions |
US20100204204A1 (en) * | 2007-06-06 | 2010-08-12 | University Of South Florida | Nutraceutical co-crystal compositions |
PL2368440T3 (pl) * | 2007-06-29 | 2014-10-31 | Dsm Ip Assets Bv | Kompozycja dodatku paszowego zawierająca kwas benzoesowy i mieszaninę zaadsorbowanych związków olejków eterycznych |
-
2011
- 2011-06-24 BR BR112012030239A patent/BR112012030239A2/pt not_active IP Right Cessation
- 2011-06-24 WO PCT/EP2011/060618 patent/WO2011161236A1/en active Application Filing
- 2011-06-24 ES ES11727187T patent/ES2725202T3/es active Active
- 2011-06-24 EA EA201270826A patent/EA022768B1/ru not_active IP Right Cessation
- 2011-06-24 JP JP2013515911A patent/JP5817067B2/ja not_active Expired - Fee Related
- 2011-06-24 CA CA2798019A patent/CA2798019A1/en not_active Abandoned
- 2011-06-24 CN CN2011800307067A patent/CN102958377A/zh active Pending
- 2011-06-24 TR TR2019/06042T patent/TR201906042T4/tr unknown
- 2011-06-24 MX MX2012014872A patent/MX2012014872A/es not_active Application Discontinuation
- 2011-06-24 UA UAA201300751A patent/UA107599C2/uk unknown
- 2011-06-24 US US13/701,054 patent/US9757331B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
TR201906042T4 (tr) | 2019-05-21 |
CN102958377A (zh) | 2013-03-06 |
CA2798019A1 (en) | 2011-12-29 |
WO2011161236A1 (en) | 2011-12-29 |
US20130095150A1 (en) | 2013-04-18 |
ES2725202T3 (es) | 2019-09-20 |
EA022768B1 (ru) | 2016-02-29 |
BR112012030239A2 (pt) | 2015-09-08 |
JP2013532157A (ja) | 2013-08-15 |
US9757331B2 (en) | 2017-09-12 |
UA107599C2 (xx) | 2015-01-26 |
MX2012014872A (es) | 2013-01-24 |
JP5817067B2 (ja) | 2015-11-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |