EA201270826A1 - Стабилизированное активное соединение - Google Patents

Стабилизированное активное соединение

Info

Publication number
EA201270826A1
EA201270826A1 EA201270826A EA201270826A EA201270826A1 EA 201270826 A1 EA201270826 A1 EA 201270826A1 EA 201270826 A EA201270826 A EA 201270826A EA 201270826 A EA201270826 A EA 201270826A EA 201270826 A1 EA201270826 A1 EA 201270826A1
Authority
EA
Eurasian Patent Office
Prior art keywords
active connection
stabilized active
carrier
vitamin
solubility
Prior art date
Application number
EA201270826A
Other languages
English (en)
Other versions
EA022768B1 (ru
Inventor
Хадижа Тантауи Эльарак
Гай Броуз
Одри Лерюит
Original Assignee
Прэйон С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Прэйон С.А. filed Critical Прэйон С.А.
Publication of EA201270826A1 publication Critical patent/EA201270826A1/ru
Publication of EA022768B1 publication Critical patent/EA022768B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/158Fatty acids; Fats; Products containing oils or fats
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/174Vitamins
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/20Inorganic substances, e.g. oligoelements
    • A23K20/24Compounds of alkaline earth metals, e.g. magnesium
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/20Inorganic substances, e.g. oligoelements
    • A23K20/26Compounds containing phosphorus
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K40/00Shaping or working-up of animal feeding-stuffs
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L33/00Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
    • A23L33/10Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
    • A23L33/15Vitamins
    • A23L33/155Vitamins A or D
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/59Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
    • A61K31/5939,10-Secocholestane derivatives, e.g. cholecalciferol, i.e. vitamin D3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/143Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00Food compositions, function of food ingredients or processes for food or foodstuffs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Zoology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Husbandry (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nutrition Science (AREA)
  • Mycology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Fodder In General (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Настоящее изобретение относится к стабильным твердым композициям, содержащим первый носитель и адсорбируемое вещество, содержащее по меньшей мере один активный компонент, такой как производное витамина D, и его гидрофобный стабилизатор, отличающимся тем, что указанный первый носитель представляет собой кальция фосфат или его производные с растворимостью в воде меньше чем 0,1 вес.% при комнатной температуре.
EA201270826A 2010-06-24 2011-06-24 Стабильная твердая композиция для пищевых, кормовых, косметических или фармацевтических препаратов и способ ее получения EA022768B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP2010059014 2010-06-24
PCT/EP2011/060618 WO2011161236A1 (en) 2010-06-24 2011-06-24 Stabilized active compound

Publications (2)

Publication Number Publication Date
EA201270826A1 true EA201270826A1 (ru) 2013-05-30
EA022768B1 EA022768B1 (ru) 2016-02-29

Family

ID=42537837

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201270826A EA022768B1 (ru) 2010-06-24 2011-06-24 Стабильная твердая композиция для пищевых, кормовых, косметических или фармацевтических препаратов и способ ее получения

Country Status (11)

Country Link
US (1) US9757331B2 (ru)
JP (1) JP5817067B2 (ru)
CN (1) CN102958377A (ru)
BR (1) BR112012030239A2 (ru)
CA (1) CA2798019A1 (ru)
EA (1) EA022768B1 (ru)
ES (1) ES2725202T3 (ru)
MX (1) MX2012014872A (ru)
TR (1) TR201906042T4 (ru)
UA (1) UA107599C2 (ru)
WO (1) WO2011161236A1 (ru)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6171333B2 (ja) * 2012-12-26 2017-08-02 東ソー株式会社 安定化したビタミンd類標準液
US9801821B2 (en) 2013-03-27 2017-10-31 Psm Healthcare Limited Stabilized vitamin D formulations
US10336817B2 (en) 2016-10-14 2019-07-02 Sultan Qaboos University Therapeutic composition of camel milk
DK3662761T3 (da) * 2018-12-04 2021-07-26 Dsm Ip Assets Bv Opbevaringsstabile adsorbater af nitrooxyforbindelser

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB405791A (en) 1933-01-14 1934-02-15 Bell And Sons Ltd Improvements in and relating to the manufacture of food accessories for cattle
US4389419A (en) 1980-11-10 1983-06-21 Damon Corporation Vitamin encapsulation
JPH085782B2 (ja) * 1989-04-14 1996-01-24 株式会社サンギ ハイドロキシアパタイト抗菌剤及びその製造法
DE19710054A1 (de) 1997-03-12 1998-09-17 Merck Patent Gmbh Pharmazeutische Zubereitung
US5820903A (en) 1997-06-30 1998-10-13 General Mills, Inc. Calcium fortified yogurt and methods of preparation
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
JP2002080358A (ja) * 2000-09-07 2002-03-19 Noevir Co Ltd 皮膚外用剤
WO2003013270A2 (en) 2001-08-09 2003-02-20 Rhodia Inc. Calcium dietary supplement
US7632518B2 (en) 2002-01-15 2009-12-15 Dsm Ip Assets B.V. 25-hydroxy vitamin D3 compositions
DE10311585A1 (de) * 2003-03-14 2004-09-23 Basf Ag Wirkstoffhaltige Adsorbate
US20100143481A1 (en) * 2006-11-08 2010-06-10 Dinesh Shenoy Method of preparing solid dosage forms of multi-phasic pharmaceutical compositions
US20100204204A1 (en) * 2007-06-06 2010-08-12 University Of South Florida Nutraceutical co-crystal compositions
PL2368440T3 (pl) * 2007-06-29 2014-10-31 Dsm Ip Assets Bv Kompozycja dodatku paszowego zawierająca kwas benzoesowy i mieszaninę zaadsorbowanych związków olejków eterycznych

Also Published As

Publication number Publication date
TR201906042T4 (tr) 2019-05-21
CN102958377A (zh) 2013-03-06
CA2798019A1 (en) 2011-12-29
WO2011161236A1 (en) 2011-12-29
US20130095150A1 (en) 2013-04-18
ES2725202T3 (es) 2019-09-20
EA022768B1 (ru) 2016-02-29
BR112012030239A2 (pt) 2015-09-08
JP2013532157A (ja) 2013-08-15
US9757331B2 (en) 2017-09-12
UA107599C2 (xx) 2015-01-26
MX2012014872A (es) 2013-01-24
JP5817067B2 (ja) 2015-11-18

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU