EA201070534A1 - Стабилизированная суспензия каризбамата для применения в педиатрии - Google Patents
Стабилизированная суспензия каризбамата для применения в педиатрииInfo
- Publication number
- EA201070534A1 EA201070534A1 EA201070534A EA201070534A EA201070534A1 EA 201070534 A1 EA201070534 A1 EA 201070534A1 EA 201070534 A EA201070534 A EA 201070534A EA 201070534 A EA201070534 A EA 201070534A EA 201070534 A1 EA201070534 A1 EA 201070534A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- pediatrics
- carisbamate
- application
- stabilized suspension
- stabilized
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/325—Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Inorganic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Emergency Medicine (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Psychology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Настоящее изобретение предоставляет стабилизированную суспензию каризбамата для применения в педиатрии и у взрослых. Конкретнее, суспензию стабилизируют гипромеллозой (НРМС) для предупреждения роста кристаллов суспендированных частиц и предупреждения рекристаллизации лекарственного средства в полиморфной форме.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US98414407P | 2007-10-31 | 2007-10-31 | |
PCT/IB2008/003331 WO2009056980A1 (en) | 2007-10-31 | 2008-10-31 | Stabilized pediatric suspension of carisbamate |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201070534A1 true EA201070534A1 (ru) | 2010-12-30 |
EA019881B1 EA019881B1 (ru) | 2014-07-30 |
Family
ID=40386492
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201070534A EA019881B1 (ru) | 2007-10-31 | 2008-10-31 | Стабилизированная суспензия каризбамата для применения в педиатрии |
Country Status (26)
Country | Link |
---|---|
US (4) | US8263652B2 (ru) |
EP (1) | EP2214637B1 (ru) |
JP (3) | JP5841333B2 (ru) |
KR (1) | KR101568681B1 (ru) |
CN (2) | CN104840971A (ru) |
AR (1) | AR069125A1 (ru) |
AU (1) | AU2008320458B2 (ru) |
BR (1) | BRPI0818118B8 (ru) |
CA (1) | CA2703971C (ru) |
CL (1) | CL2008003261A1 (ru) |
CO (1) | CO6270300A2 (ru) |
CR (1) | CR11550A (ru) |
EA (1) | EA019881B1 (ru) |
EC (1) | ECSP10010208A (ru) |
ES (1) | ES2432666T3 (ru) |
IL (1) | IL205352A (ru) |
MX (1) | MX2010004889A (ru) |
MY (1) | MY154063A (ru) |
NI (1) | NI201000076A (ru) |
PA (1) | PA8801901A1 (ru) |
PE (1) | PE20090951A1 (ru) |
PL (1) | PL2214637T3 (ru) |
TW (1) | TW200934531A (ru) |
UY (1) | UY31444A1 (ru) |
WO (1) | WO2009056980A1 (ru) |
ZA (1) | ZA201003848B (ru) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8263652B2 (en) * | 2007-10-31 | 2012-09-11 | Sk Biopharmaceuticals Co., Ltd. | Stabilized pediatric suspension of carisbamate |
WO2011107855A2 (en) | 2010-03-04 | 2011-09-09 | Torrent Pharmaceuticals Limited | Sustained release oral liquid suspension dosage form |
EP2563763B1 (en) * | 2010-04-30 | 2014-12-31 | Bristol-Myers Squibb Company | Pharmaceutical compositions comprising n-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-l-(4-fluorophenyl)-2-oxo- 1,2-dihydropyridine-3 -carboxamide |
US8609849B1 (en) | 2010-11-30 | 2013-12-17 | Fox Chase Chemical Diversity Center, Inc. | Hydroxylated sulfamides exhibiting neuroprotective action and their method of use |
AR088372A1 (es) * | 2011-10-19 | 2014-05-28 | Otsuka Pharma Co Ltd | Solucion para administracion oral |
TWI660748B (zh) * | 2013-03-01 | 2019-06-01 | 日商大塚製藥股份有限公司 | 用於口服投藥之包含非晶型托伐普坦(Tolvaptan)的懸浮液 |
CN103966680A (zh) * | 2014-05-04 | 2014-08-06 | 东华大学 | 一种药物缓释纳米纤维的制备方法 |
TW201717929A (zh) * | 2015-05-22 | 2017-06-01 | 愛思開生物製藥股份有限公司 | 包括卡立胺酯之藥物及其於預防、緩解或治療疼痛或癲癎之用途 |
ITUB20155193A1 (it) * | 2015-11-03 | 2017-05-03 | Italfarmaco Spa | Sospensioni orali di Givinostat fisicamente e chimicamente stabili |
CN105997866B (zh) * | 2016-07-13 | 2019-08-20 | 成都明慈医药科技有限公司 | 一种含地塞米松的混悬剂及其制备方法 |
US10336679B2 (en) * | 2016-10-24 | 2019-07-02 | Syneurx International (Taiwan) Corp. | Polymorphic forms of sodium benzoate and uses thereof |
US11369579B2 (en) | 2016-10-24 | 2022-06-28 | Syneurx International (Taiwan) Corp. | Polymorphic forms of sodium benzoate and uses thereof |
US10098861B1 (en) | 2017-10-24 | 2018-10-16 | Syneurx International (Taiwan) Corp. | Pharmaceutical composition comprising sodium benzoate compound and clozapine, and uses thereof |
KR102369827B1 (ko) | 2020-09-04 | 2022-03-04 | (주)피알지에스앤텍 | 프로게리닌을 포함하는 나노현탁액 및 이의 제조방법 |
US20220213802A1 (en) * | 2021-01-06 | 2022-07-07 | General Electric Company | System for controlling blade clearances within a gas turbine engine |
KR102686558B1 (ko) | 2022-01-25 | 2024-07-22 | (주)피알지에스앤텍 | 프로게리닌을 포함하는 과립제 및 이를 이용한 샤셋제 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3265728A (en) | 1962-07-18 | 1966-08-09 | Armour Pharma | Substituted phenethyl carbamates |
RU2141821C1 (ru) * | 1994-10-14 | 1999-11-27 | Жансен Фармасетика Н.В. | Водная суспензия сабелюзола для орального применения и способ ее изготовления |
US5698588A (en) | 1996-01-16 | 1997-12-16 | Yukong Limited | Halogen substituted carbamate compounds from 2-phenyl-1,2-ethanediol |
WO2001013904A2 (en) * | 1999-08-20 | 2001-03-01 | Ortho-Mcneil Pharmaceutical, Inc. | Composition comprising a tramadol material and an anticonvulsant drug |
RS50505B (sr) * | 2001-02-27 | 2010-03-02 | Ortho-Mcneil Pharmaceutical Inc. | Karbamatna jedinjenja za upotrebu u sprečavanju ili lečenju anksioznih poremećaja |
AP2005003467A0 (en) * | 2003-06-17 | 2006-12-31 | Pfizer | N-pyrrolidin-3-YL-amide derivatives as serotonin and noradrenaline reuptake inhibitors. |
EP2051696A2 (en) * | 2006-08-18 | 2009-04-29 | Morton Grove Pharmaceuticals, Inc. | Stable liquid levetiracetam compositions and methods |
MX2009003929A (es) * | 2006-10-13 | 2009-06-26 | Janssen Pharmaceutica Nv | Composiciones de fenilalquil carbamato. |
US8263652B2 (en) * | 2007-10-31 | 2012-09-11 | Sk Biopharmaceuticals Co., Ltd. | Stabilized pediatric suspension of carisbamate |
-
2008
- 2008-10-27 US US12/258,490 patent/US8263652B2/en active Active
- 2008-10-29 PA PA20088801901A patent/PA8801901A1/es unknown
- 2008-10-30 TW TW097141713A patent/TW200934531A/zh unknown
- 2008-10-30 CL CL2008003261A patent/CL2008003261A1/es unknown
- 2008-10-30 AR ARP080104758A patent/AR069125A1/es unknown
- 2008-10-30 UY UY31444A patent/UY31444A1/es unknown
- 2008-10-31 MX MX2010004889A patent/MX2010004889A/es active IP Right Grant
- 2008-10-31 BR BRPI0818118A patent/BRPI0818118B8/pt active IP Right Grant
- 2008-10-31 AU AU2008320458A patent/AU2008320458B2/en active Active
- 2008-10-31 ES ES08843347T patent/ES2432666T3/es active Active
- 2008-10-31 WO PCT/IB2008/003331 patent/WO2009056980A1/en active Application Filing
- 2008-10-31 CN CN201510170122.XA patent/CN104840971A/zh active Pending
- 2008-10-31 JP JP2010531607A patent/JP5841333B2/ja active Active
- 2008-10-31 CA CA2703971A patent/CA2703971C/en active Active
- 2008-10-31 PE PE2008001876A patent/PE20090951A1/es not_active Application Discontinuation
- 2008-10-31 EP EP08843347.9A patent/EP2214637B1/en active Active
- 2008-10-31 MY MYPI2010001910A patent/MY154063A/en unknown
- 2008-10-31 EA EA201070534A patent/EA019881B1/ru not_active IP Right Cessation
- 2008-10-31 KR KR1020107011813A patent/KR101568681B1/ko active IP Right Grant
- 2008-10-31 PL PL08843347T patent/PL2214637T3/pl unknown
- 2008-10-31 CN CN200880114312A patent/CN101848699A/zh active Pending
-
2010
- 2010-04-26 IL IL205352A patent/IL205352A/en active IP Right Grant
- 2010-04-29 NI NI201000076A patent/NI201000076A/es unknown
- 2010-05-10 CO CO10055401A patent/CO6270300A2/es not_active Application Discontinuation
- 2010-05-28 ZA ZA2010/03848A patent/ZA201003848B/en unknown
- 2010-05-28 EC EC2010010208A patent/ECSP10010208A/es unknown
- 2010-06-30 CR CR11550A patent/CR11550A/es not_active Application Discontinuation
-
2012
- 2012-08-09 US US13/570,853 patent/US9161913B2/en active Active
-
2014
- 2014-06-05 JP JP2014116727A patent/JP2014193913A/ja active Pending
-
2015
- 2015-09-18 US US14/858,583 patent/US20160008476A1/en not_active Abandoned
-
2016
- 2016-07-11 JP JP2016136713A patent/JP6273589B2/ja active Active
-
2017
- 2017-01-06 US US15/400,676 patent/US10201519B2/en active Active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201070534A1 (ru) | Стабилизированная суспензия каризбамата для применения в педиатрии | |
CL2012002771A1 (es) | Compuestos derivados de ariletinilo sustituidos, moduladores de los receptores mglur5; proceso de obtencion; composicion farmaceutica; y su uso en el tratamiento o prevencion de la esquizofrenia, enfermedades cognitivas, sindrome de x fragil o el autismo. | |
EA201291220A1 (ru) | Производные аминопиримидина в качестве модуляторов lrrk2 | |
EA201200174A1 (ru) | Производные оксазина и их применение в качестве ингибиторов bace для лечения неврологических нарушений | |
EA201101709A1 (ru) | Полициклические антагонисты рецепторов лизофосфатидной кислоты | |
MX2013007295A (es) | Quinoxalinas y aza-quinoxalinas como moduladores del receptor de crth2. | |
EA201300200A1 (ru) | N-((6-аминопиридин-3-ил)метил)гетероарилкарбоксамиды в качестве ингибиторов калликреина в плазме | |
MX349556B (es) | Derivados de aminopirimidina como moduladores de proteina cinasa 2 rica en unidades repetitivas de leucina (lrrk2). | |
RS54123B1 (en) | THERAPEUTIC COMBINATION CONTAINING DOLUTEGRAVIR, ABACAVIR AND LAMIVUDINE | |
EA201490569A1 (ru) | Полиморфная форма гидрохлорида придопидина | |
MX2011013016A (es) | Derivados de aminopirrolidinona y usos de los mismos. | |
EA201001243A1 (ru) | Кристаллические формы n-[2-(диэтиламино)этил]-5-[(5-фтор-1,2-дигидро-2-оксо-3н-индол-3-илиден)метил]-2,4-диметил-1н-пиррол-3-карбоксамида и способы их получения | |
PE20090876A1 (es) | Nuevos derivados de 6-aril/heteroalquiloxi benzotiazol y bencimidazol, su procedimiento de preparacion, su aplicacion como medicamentos, composiciones farmaceuticas y nueva utilizacion principalmente como inhibidores de cmet | |
EA201270808A1 (ru) | Новые формы рифаксимина и их применение | |
CY1120435T1 (el) | Φαρμακοτεχνικες μορφες που περιλαμβανουν κρυσταλλικες μορφες του μονοενυδρου υδροχλωρικου (r)-7-χλωρο-ν-(κινουκλιδινο-3-υλο) βενζο(β)θειοφαινο-2-καρβοξαμιδιου | |
EA201300436A1 (ru) | Совместные кристаллы и соли ингибиторов ccr3 | |
EA201300034A1 (ru) | Фармацевтические композиции, содержащие иматиниб или его фармацевтически приемлемую соль, и способы их получения | |
EA201200046A1 (ru) | Новые соединения, фармацевтическая композиция и связанные с ними способы | |
EA201000391A1 (ru) | Соединение, представляющее собой ингибитор гликогенфосфорилазы, и его фармацевтическая композиция | |
CY1118036T1 (el) | Βελτιστοποιημενη συνθεση καθαρων μη-πολυμορφικων, κρυσταλλικων χολικων οξεων με καθορισμενο μεγεθος σωματιδιων | |
MX2010001851A (es) | Derivados de indol-2-ona disustituidos en 3, su preparacion y uso terapeutico. | |
EA201001870A1 (ru) | Новые кристаллические формы рабепразола натрия | |
EA201290229A1 (ru) | Производные спиролактама и их применение | |
MY157425A (en) | Substituted oxindole derivatives and the use thereof for the treatment of vasopressin-dependent illnesses | |
EA201270377A1 (ru) | Стабильные композиции sns-595 и способы их получения |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |
|
PC4A | Registration of transfer of a eurasian patent by assignment |