EA200801875A1 - Антагонист cd 80 - Google Patents
Антагонист cd 80Info
- Publication number
- EA200801875A1 EA200801875A1 EA200801875A EA200801875A EA200801875A1 EA 200801875 A1 EA200801875 A1 EA 200801875A1 EA 200801875 A EA200801875 A EA 200801875A EA 200801875 A EA200801875 A EA 200801875A EA 200801875 A1 EA200801875 A1 EA 200801875A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- antagonist
- cinnolin
- dihydropyrazolo
- difluoroethyl
- benzamide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Transplantation (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
Abstract
Холиновая соль антагониста CD80 - 4-(6-фтор-3-оксо-1,3-дигидропиразоло[4,3-с]циннолин-2-ил)-N-(2,2-дифторэтил)бензамида обладает хорошей растворимостью в воде и поэтому удобна для использования в составе лекарственных средств.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0603522.4A GB0603522D0 (en) | 2006-02-22 | 2006-02-22 | Kinase inhibition |
PCT/GB2007/000550 WO2007096588A1 (en) | 2006-02-22 | 2007-02-19 | Salt of cd 80 antagonist |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200801875A1 true EA200801875A1 (ru) | 2008-12-30 |
EA014101B1 EA014101B1 (ru) | 2010-08-30 |
Family
ID=36178528
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200801875A EA014101B1 (ru) | 2006-02-22 | 2007-02-19 | Антагонист cd80 |
Country Status (20)
Country | Link |
---|---|
US (3) | US20090221590A1 (ru) |
EP (1) | EP1991548B1 (ru) |
JP (1) | JP5102785B2 (ru) |
KR (1) | KR101433738B1 (ru) |
CN (1) | CN101384595B (ru) |
AU (1) | AU2007217170B2 (ru) |
BR (1) | BRPI0708114B8 (ru) |
CA (1) | CA2643668C (ru) |
DK (1) | DK1991548T3 (ru) |
EA (1) | EA014101B1 (ru) |
ES (1) | ES2449569T3 (ru) |
GB (1) | GB0603522D0 (ru) |
HK (1) | HK1125376A1 (ru) |
IL (1) | IL192954A (ru) |
NZ (1) | NZ570055A (ru) |
PL (1) | PL1991548T3 (ru) |
PT (1) | PT1991548E (ru) |
UA (1) | UA91904C2 (ru) |
WO (1) | WO2007096588A1 (ru) |
ZA (1) | ZA200806508B (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA009680B1 (ru) | 2003-03-14 | 2008-02-28 | Эвидекс Лимитед | Иммуномодулирующие гетероциклические соединения |
JP4763697B2 (ja) | 2004-08-09 | 2011-08-31 | メディジーン リミテッド | Cd80抑制剤としての免疫調整性オキソピラゾロシンノリン類 |
AU2009309575B2 (en) | 2008-10-31 | 2015-02-26 | C-A-I-R Biosciences Gmbh | Choline and tromethamine salt of Licofelone |
RU2557237C2 (ru) | 2010-02-10 | 2015-07-20 | Киссеи Фармасьютикал Ко., Лтд. | Соль конденсированного гетероциклического производного и его кристаллы |
UA109287C2 (uk) * | 2010-11-02 | 2015-08-10 | Солі органічного аміну похідних амінобензойної кислоти і спосіб їх одержання | |
EP4119128A1 (en) | 2021-07-13 | 2023-01-18 | Dr. Falk Pharma Gmbh | Pharmaceutical composition for the oral administration of poorly soluble drugs comprising an amorphous solid dispersion |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2670350A (en) * | 1952-08-08 | 1954-02-23 | Nepera Chemical Co Inc | Method of preparing choline salt of theophylline |
US3576637A (en) * | 1967-04-20 | 1971-04-27 | Konishiroku Photo Ind | Lith-type of emulsion containing pyrozolone |
US3778150A (en) * | 1971-10-27 | 1973-12-11 | K Aston | Printing of photographic colour negatives |
JPS523818A (en) * | 1975-06-26 | 1977-01-12 | Hoffmann La Roche | Salt of penicillanic acid |
US4591589A (en) * | 1985-01-16 | 1986-05-27 | Roussel Uclaf | 2-aryl pyrazolo[4,3-c]cinnolin-3-ones |
DE3903993A1 (de) * | 1989-02-10 | 1990-08-16 | Basf Ag | Diarylsubstituierte heterocyclische verbindungen, ihre herstellung und arzneimittel daraus |
IT1290448B1 (it) * | 1997-04-01 | 1998-12-03 | Schiena Michele Giuseppe Di | Nimesulide sale di colina,metodo di preparazione e composizioni farmaceutiche che lo contengono |
EA009680B1 (ru) | 2003-03-14 | 2008-02-28 | Эвидекс Лимитед | Иммуномодулирующие гетероциклические соединения |
TW200526638A (en) * | 2003-10-22 | 2005-08-16 | Smithkline Beecham Corp | 2-(3,4-dimethylphenyl)-4-{[2-hydroxy-3'-(1H-tetrazol-5-yl)biphenyl-3-yl]-hydrazono}-5-methyl-2,4-dihydropyrazol-3-one choline |
GB0325644D0 (en) * | 2003-11-04 | 2003-12-10 | Avidex Ltd | Immuno ihibitory pyrazolone compounds |
GB0411770D0 (en) * | 2004-05-26 | 2004-06-30 | Avidex Ltd | Immuno inhibitory heterocyclic compouds |
JP4763697B2 (ja) * | 2004-08-09 | 2011-08-31 | メディジーン リミテッド | Cd80抑制剤としての免疫調整性オキソピラゾロシンノリン類 |
WO2006083687A1 (en) * | 2005-01-28 | 2006-08-10 | Cardiome Pharma Corp. | Crystal salt of xanthine oxidase inhibitors |
-
2006
- 2006-02-22 GB GBGB0603522.4A patent/GB0603522D0/en not_active Ceased
-
2007
- 2007-02-19 JP JP2008555857A patent/JP5102785B2/ja not_active Expired - Fee Related
- 2007-02-19 EP EP07712727.2A patent/EP1991548B1/en active Active
- 2007-02-19 DK DK07712727.2T patent/DK1991548T3/en active
- 2007-02-19 US US12/279,898 patent/US20090221590A1/en not_active Abandoned
- 2007-02-19 NZ NZ570055A patent/NZ570055A/en unknown
- 2007-02-19 UA UAA200811363A patent/UA91904C2/ru unknown
- 2007-02-19 AU AU2007217170A patent/AU2007217170B2/en active Active
- 2007-02-19 EA EA200801875A patent/EA014101B1/ru unknown
- 2007-02-19 PL PL07712727T patent/PL1991548T3/pl unknown
- 2007-02-19 CN CN2007800051162A patent/CN101384595B/zh active Active
- 2007-02-19 KR KR1020087019729A patent/KR101433738B1/ko active IP Right Grant
- 2007-02-19 CA CA2643668A patent/CA2643668C/en active Active
- 2007-02-19 BR BRPI0708114A patent/BRPI0708114B8/pt active IP Right Grant
- 2007-02-19 PT PT77127272T patent/PT1991548E/pt unknown
- 2007-02-19 ES ES07712727.2T patent/ES2449569T3/es active Active
- 2007-02-19 WO PCT/GB2007/000550 patent/WO2007096588A1/en active Application Filing
-
2008
- 2008-07-22 IL IL192954A patent/IL192954A/en active IP Right Grant
- 2008-07-25 ZA ZA200806508A patent/ZA200806508B/xx unknown
-
2009
- 2009-05-07 HK HK09104229.6A patent/HK1125376A1/xx unknown
-
2011
- 2011-09-15 US US13/233,634 patent/US20120004237A1/en not_active Abandoned
-
2017
- 2017-11-20 US US15/817,323 patent/US20180265514A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN101384595A (zh) | 2009-03-11 |
GB0603522D0 (en) | 2006-04-05 |
US20090221590A1 (en) | 2009-09-03 |
BRPI0708114A2 (pt) | 2011-05-17 |
BRPI0708114B1 (pt) | 2020-02-04 |
JP5102785B2 (ja) | 2012-12-19 |
WO2007096588A1 (en) | 2007-08-30 |
US20120004237A1 (en) | 2012-01-05 |
KR101433738B1 (ko) | 2014-08-25 |
EA014101B1 (ru) | 2010-08-30 |
CA2643668A1 (en) | 2007-08-30 |
UA91904C2 (en) | 2010-09-10 |
US20180265514A1 (en) | 2018-09-20 |
IL192954A (en) | 2015-01-29 |
BRPI0708114B8 (pt) | 2021-05-25 |
IL192954A0 (en) | 2009-02-11 |
ZA200806508B (en) | 2009-06-24 |
HK1125376A1 (en) | 2009-08-07 |
DK1991548T3 (en) | 2014-03-10 |
NZ570055A (en) | 2011-08-26 |
PL1991548T3 (pl) | 2014-05-30 |
CN101384595B (zh) | 2011-02-09 |
AU2007217170B2 (en) | 2012-02-02 |
KR20080103523A (ko) | 2008-11-27 |
PT1991548E (pt) | 2014-03-10 |
EP1991548B1 (en) | 2013-12-11 |
JP2009527538A (ja) | 2009-07-30 |
AU2007217170A1 (en) | 2007-08-30 |
CA2643668C (en) | 2014-05-13 |
ES2449569T3 (es) | 2014-03-20 |
EP1991548A1 (en) | 2008-11-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC4A | Registration of transfer of a eurasian patent by assignment |