EA200700179A1 - Производные пиррола, их получение и их применение в терапии - Google Patents

Производные пиррола, их получение и их применение в терапии

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Publication number
EA200700179A1
EA200700179A1 EA200700179A EA200700179A EA200700179A1 EA 200700179 A1 EA200700179 A1 EA 200700179A1 EA 200700179 A EA200700179 A EA 200700179A EA 200700179 A EA200700179 A EA 200700179A EA 200700179 A1 EA200700179 A1 EA 200700179A1
Authority
EA
Eurasian Patent Office
Prior art keywords
therapy
pyrrola
derivatives
production
application
Prior art date
Application number
EA200700179A
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English (en)
Other versions
EA012726B1 (ru
Inventor
Франсис Барт
Кристиан Конжи
Лоран Ортала
Мюриэлль Ринальди-Кармона
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Санофи-Авентис
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Application filed by Санофи-Авентис filed Critical Санофи-Авентис
Publication of EA200700179A1 publication Critical patent/EA200700179A1/ru
Publication of EA012726B1 publication Critical patent/EA012726B1/ru

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    • A61K31/33Heterocyclic compounds
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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Abstract

Объектом изобретения являются соединения, отвечающие формуле (I), в которой Rозначает водород или (C-C) алкил; Rозначает группу (С-С); неароматический карбоциклический остаток C-C; инданил; 1,2, 3,4-тетрагидронафталенил-1 или -2; гетероциклический остаток; замещенную (C-С)алкиленовую группу; группу NRR; или Rи Rвместе с атомом азота, с которым они связаны, образуют гетероциклический остаток. Способ получения и применение в терапии.
EA200700179A 2004-08-09 2005-08-02 Производные пиррола, их получение и их применение в терапии EA012726B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0408773A FR2874012B1 (fr) 2004-08-09 2004-08-09 Derives de pyrrole, leur preparation et leur utlisation en therapeutique
PCT/FR2005/002015 WO2006024777A1 (fr) 2004-08-09 2005-08-02 Derives de pyrrole, leur preparation et leur utilisation en therapeutique

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EA200700179A1 true EA200700179A1 (ru) 2007-08-31
EA012726B1 EA012726B1 (ru) 2009-12-30

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EA200700179A EA012726B1 (ru) 2004-08-09 2005-08-02 Производные пиррола, их получение и их применение в терапии

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US (2) US7381727B2 (ru)
EP (1) EP1781636A1 (ru)
JP (1) JP2008509202A (ru)
KR (1) KR20070054649A (ru)
CN (1) CN101014588A (ru)
AR (1) AR050447A1 (ru)
AU (1) AU2005279086A1 (ru)
BR (1) BRPI0514235A (ru)
CA (1) CA2576717A1 (ru)
EA (1) EA012726B1 (ru)
FR (1) FR2874012B1 (ru)
IL (1) IL180867A0 (ru)
MA (1) MA28847B1 (ru)
MX (1) MX2007001383A (ru)
NO (1) NO20071209L (ru)
PE (1) PE20060419A1 (ru)
TW (1) TW200616948A (ru)
UY (1) UY29054A1 (ru)
WO (1) WO2006024777A1 (ru)
ZA (1) ZA200700950B (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2005264980A1 (en) * 2004-06-16 2006-01-26 Inotek Pharmaceuticals Corporation Methods for treating or preventing erectile dysfunction or urinary incontinence
FR2874012B1 (fr) * 2004-08-09 2008-08-22 Sanofi Synthelabo Derives de pyrrole, leur preparation et leur utlisation en therapeutique
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KR20070054649A (ko) 2007-05-29
WO2006024777A1 (fr) 2006-03-09
TW200616948A (en) 2006-06-01
US20070149596A1 (en) 2007-06-28
US20080194581A1 (en) 2008-08-14
ZA200700950B (en) 2008-06-25
NO20071209L (no) 2007-03-05
FR2874012A1 (fr) 2006-02-10
FR2874012B1 (fr) 2008-08-22
CN101014588A (zh) 2007-08-08
BRPI0514235A (pt) 2008-06-03
CA2576717A1 (fr) 2006-03-09
MA28847B1 (fr) 2007-09-03
IL180867A0 (en) 2007-07-04
AR050447A1 (es) 2006-10-25
JP2008509202A (ja) 2008-03-27
PE20060419A1 (es) 2006-06-20
AU2005279086A1 (en) 2006-03-09
EA012726B1 (ru) 2009-12-30
EP1781636A1 (fr) 2007-05-09
US7879902B2 (en) 2011-02-01
US7381727B2 (en) 2008-06-03
UY29054A1 (es) 2006-03-31

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