EA200401169A1 - Аминометилзамещенные тетрациклиновые соединения - Google Patents

Аминометилзамещенные тетрациклиновые соединения

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Publication number
EA200401169A1
EA200401169A1 EA200401169A EA200401169A EA200401169A1 EA 200401169 A1 EA200401169 A1 EA 200401169A1 EA 200401169 A EA200401169 A EA 200401169A EA 200401169 A EA200401169 A EA 200401169A EA 200401169 A1 EA200401169 A1 EA 200401169A1
Authority
EA
Eurasian Patent Office
Prior art keywords
tetracycline compounds
substituted tetracycline
aminomethyl substituted
aminomethyl
compounds
Prior art date
Application number
EA200401169A
Other languages
English (en)
Other versions
EA013819B1 (ru
Inventor
Марк Л. Нельсон
Квази Охеменг
Роджер Фречетт
Мохамед И. Исмаил
Лора Макинтайр
Тодд Баузер
Original Assignee
Паратек Фармасьютикалс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Паратек Фармасьютикалс, Инк. filed Critical Паратек Фармасьютикалс, Инк.
Publication of EA200401169A1 publication Critical patent/EA200401169A1/ru
Publication of EA013819B1 publication Critical patent/EA013819B1/ru

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    • C07C235/66—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems and singly-bound oxygen atoms, bound to the same carbon skeleton
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    • C07C2603/40—Ortho- or ortho- and peri-condensed systems containing four condensed rings
    • C07C2603/42—Ortho- or ortho- and peri-condensed systems containing four condensed rings containing only six-membered rings
    • C07C2603/44—Naphthacenes; Hydrogenated naphthacenes
    • C07C2603/46—1,4,4a,5,5a,6,11,12a- Octahydronaphthacenes, e.g. tetracyclines

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Abstract

Рассмотрены аминометилзамещенные тетрациклиновые соединения, фармацевтические композиции и способы их применения.Отчет о международном поиске был опубликован 2004.02.05.
EA200401169A 2002-03-08 2003-03-10 Аминометилзамещенные тетрациклиновые соединения EA013819B1 (ru)

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US39549502P 2002-07-12 2002-07-12
PCT/US2003/007229 WO2003075857A2 (en) 2002-03-08 2003-03-10 Amino-methyl substituted tetracycline compounds

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EA200401169A1 true EA200401169A1 (ru) 2005-04-28
EA013819B1 EA013819B1 (ru) 2010-08-30

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EA200802365A EA200802365A1 (ru) 2002-03-08 2003-03-10 Аминометилзамещенные тетрациклиновые соединения
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JP2011102296A (ja) 2011-05-26
KR20040097160A (ko) 2004-11-17
CA2478335A1 (en) 2003-09-18
CN102531948A (zh) 2012-07-04
AU2009208042A1 (en) 2009-08-27
KR101093842B1 (ko) 2011-12-13
CN1649582A (zh) 2005-08-03
EP2301534A1 (en) 2011-03-30
KR101163937B1 (ko) 2012-07-09
IL213220A0 (en) 2011-07-31
AU2003220123B2 (en) 2009-05-07
US20050026875A1 (en) 2005-02-03
JP2010195796A (ja) 2010-09-09
EA201000491A1 (ru) 2010-08-30
EP2316450A1 (en) 2011-05-04
AU2003220123A1 (en) 2003-09-22
US7326696B2 (en) 2008-02-05
IL163931A (en) 2013-06-27
US20080015169A1 (en) 2008-01-17
IL163931A0 (en) 2005-12-18
CA2478335C (en) 2011-05-10
WO2003075857A3 (en) 2004-02-05
KR20110038186A (ko) 2011-04-13
CN101307017A (zh) 2008-11-19
EP1482926A4 (en) 2006-04-12
EA013819B1 (ru) 2010-08-30
AU2009208042B2 (en) 2013-02-14
JP2008266330A (ja) 2008-11-06
WO2003075857A2 (en) 2003-09-18
KR20100090310A (ko) 2010-08-13
EP2311451A1 (en) 2011-04-20
KR101014918B1 (ko) 2011-02-15
EA200802365A1 (ru) 2009-08-28
EP1482926A2 (en) 2004-12-08

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