EA200000081A1 - Малеат 5-(2-этил-2h-тетразол-5-ил)-1-метил-1,2,3,6-тетрагидропиридина - Google Patents

Малеат 5-(2-этил-2h-тетразол-5-ил)-1-метил-1,2,3,6-тетрагидропиридина

Info

Publication number
EA200000081A1
EA200000081A1 EA200000081A EA200000081A EA200000081A1 EA 200000081 A1 EA200000081 A1 EA 200000081A1 EA 200000081 A EA200000081 A EA 200000081A EA 200000081 A EA200000081 A EA 200000081A EA 200000081 A1 EA200000081 A1 EA 200000081A1
Authority
EA
Eurasian Patent Office
Prior art keywords
tetrahydropyridine
tetrazol
methyl
ethil
maleat
Prior art date
Application number
EA200000081A
Other languages
English (en)
Inventor
Михаэль Бех Соммер
Оле Нильсен
Original Assignee
Х.Лундбекк А/С
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Х.Лундбекк А/С filed Critical Х.Лундбекк А/С
Publication of EA200000081A1 publication Critical patent/EA200000081A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Настоящее изобретение относится к соли присоединения малеиновой кислоты 5-(2-этил-2H-тетразол-5-ил)-1-метил-1,2,3,6-тетрагидропиридина, фармацевтическим композициям, содержащим соль присоединения кислоты, и к их использованию для лечения расстройств, вызванных дисфункцией ацетилхолиновой (AcCh) или мускариновой системы.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200000081A 1997-07-01 1998-07-01 Малеат 5-(2-этил-2h-тетразол-5-ил)-1-метил-1,2,3,6-тетрагидропиридина EA200000081A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK78197 1997-07-01
PCT/DK1998/000294 WO1999001448A1 (en) 1997-07-01 1998-07-01 5-(2-ethyl-2h-tetrazol-5-y1)-1-methyl-1,2,3,6-tetrahydropyridine maleate

Publications (1)

Publication Number Publication Date
EA200000081A1 true EA200000081A1 (ru) 2000-08-28

Family

ID=8097489

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200000081A EA200000081A1 (ru) 1997-07-01 1998-07-01 Малеат 5-(2-этил-2h-тетразол-5-ил)-1-метил-1,2,3,6-тетрагидропиридина

Country Status (25)

Country Link
EP (1) EP0994869A1 (ru)
JP (1) JP2002507215A (ru)
KR (1) KR20010014297A (ru)
CN (1) CN1261361A (ru)
AR (1) AR013096A1 (ru)
AU (1) AU735751B2 (ru)
BG (1) BG103933A (ru)
BR (1) BR9810331A (ru)
CA (1) CA2293324A1 (ru)
CO (1) CO4940483A1 (ru)
EA (1) EA200000081A1 (ru)
HU (1) HUP0002876A2 (ru)
IL (1) IL133093A0 (ru)
IS (1) IS5278A (ru)
JO (1) JO2031B1 (ru)
MA (1) MA25138A1 (ru)
NO (1) NO996580D0 (ru)
PE (1) PE116099A1 (ru)
PL (1) PL337184A1 (ru)
SK (1) SK187399A3 (ru)
TN (1) TNSN98120A1 (ru)
TR (1) TR199903283T2 (ru)
UY (2) UY25069A1 (ru)
WO (1) WO1999001448A1 (ru)
ZA (1) ZA985498B (ru)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714789D0 (en) * 1987-06-24 1987-07-29 Lundbeck & Co As H Heterocyclic compounds
WO1997017074A1 (en) * 1995-11-06 1997-05-15 H. Lundbeck A/S Treatment of traumatic brain injury

Also Published As

Publication number Publication date
BR9810331A (pt) 2000-09-05
EP0994869A1 (en) 2000-04-26
CN1261361A (zh) 2000-07-26
UY25177A1 (es) 2000-12-29
MA25138A1 (fr) 2001-04-02
HUP0002876A2 (hu) 2001-06-28
IS5278A (is) 1999-11-30
AU735751B2 (en) 2001-07-12
PL337184A1 (en) 2000-08-14
KR20010014297A (ko) 2001-02-26
AU8102098A (en) 1999-01-25
SK187399A3 (en) 2000-06-12
PE116099A1 (es) 1999-11-23
IL133093A0 (en) 2001-03-19
NO996580L (no) 1999-12-30
TNSN98120A1 (fr) 2005-03-15
CA2293324A1 (en) 1999-01-14
ZA985498B (en) 1999-01-20
CO4940483A1 (es) 2000-07-24
AR013096A1 (es) 2000-12-13
WO1999001448A1 (en) 1999-01-14
JP2002507215A (ja) 2002-03-05
UY25069A1 (es) 1998-12-21
JO2031B1 (en) 1999-05-15
NO996580D0 (no) 1999-12-30
TR199903283T2 (xx) 2000-06-21
BG103933A (en) 2000-07-31

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