EA199700247A1 - Прозрачные, быстро высвобождающие активное вещество композиции нестероидных анальгетиков - Google Patents

Прозрачные, быстро высвобождающие активное вещество композиции нестероидных анальгетиков

Info

Publication number
EA199700247A1
EA199700247A1 EA199700247A EA199700247A EA199700247A1 EA 199700247 A1 EA199700247 A1 EA 199700247A1 EA 199700247 A EA199700247 A EA 199700247A EA 199700247 A EA199700247 A EA 199700247A EA 199700247 A1 EA199700247 A1 EA 199700247A1
Authority
EA
Eurasian Patent Office
Prior art keywords
transparent
active substance
nesteroidal
analgetics
substance compositions
Prior art date
Application number
EA199700247A
Other languages
English (en)
Other versions
EA000434B1 (ru
Inventor
Йёрг Брайтенбах
Аксель Заннер
Йёрг Розенберг
Original Assignee
Басф Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Басф Акциенгезельшафт filed Critical Басф Акциенгезельшафт
Publication of EA199700247A1 publication Critical patent/EA199700247A1/ru
Publication of EA000434B1 publication Critical patent/EA000434B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Finger-Pressure Massage (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Прозрачные, быстро высвобождающие активное вещество композиции, получаемые экструзией расплавов, содержащих нестероидные анальгетики, гомополимеры N-винилпирролидона, сахариды или многоатомные спирты, образующие при окислении моносахариды, и натриевые или калиевые соли.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA199700247A 1995-03-21 1996-03-09 Фармацевтическая композиция, получаемая экструзией расплава EA000434B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19509805A DE19509805A1 (de) 1995-03-21 1995-03-21 Transparente, schnell freisetzende Zubereitungen von nichtsteroidalen Analgetica
PCT/EP1996/001021 WO1996029053A1 (de) 1995-03-21 1996-03-09 Transparente, schnell freisetzende zubereitungen von nichtsteroidalen analgetica

Publications (2)

Publication Number Publication Date
EA199700247A1 true EA199700247A1 (ru) 1998-02-26
EA000434B1 EA000434B1 (ru) 1999-08-26

Family

ID=7757016

Family Applications (1)

Application Number Title Priority Date Filing Date
EA199700247A EA000434B1 (ru) 1995-03-21 1996-03-09 Фармацевтическая композиция, получаемая экструзией расплава

Country Status (21)

Country Link
US (1) US6063821A (ru)
EP (1) EP0817612B1 (ru)
JP (1) JPH11502209A (ru)
KR (1) KR19980703160A (ru)
AT (1) ATE196078T1 (ru)
AU (1) AU5105396A (ru)
BR (1) BR9607867A (ru)
CA (1) CA2213719C (ru)
CZ (1) CZ286011B6 (ru)
DE (2) DE19509805A1 (ru)
DK (1) DK0817612T3 (ru)
EA (1) EA000434B1 (ru)
ES (1) ES2151150T3 (ru)
GR (1) GR3034441T3 (ru)
HU (1) HU221614B (ru)
IL (1) IL117531A (ru)
NO (1) NO318236B1 (ru)
PT (1) PT817612E (ru)
TW (1) TW416850B (ru)
WO (1) WO1996029053A1 (ru)
ZA (1) ZA962241B (ru)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19602206A1 (de) 1996-01-23 1997-07-24 Basf Ag Zubereitungen nichtsteroidaler Analgetika
US6274727B1 (en) 1996-11-15 2001-08-14 Merck Patent Gesellschaft Mit Beschrankter Haftung Method for producing shaped and unshaped polyol masses
DE69834255T2 (de) * 1997-07-25 2006-09-28 Alpex Pharma S.A. Verfahren zur herstellung eines granulates, geeignet zur herstellung schnell-freisetzender, im mund löslicher tabletten
US7364752B1 (en) 1999-11-12 2008-04-29 Abbott Laboratories Solid dispersion pharamaceutical formulations
WO2001034119A2 (en) * 1999-11-12 2001-05-17 Abbott Laboratories Inhibitors of crystallization in a solid dispersion
ES2170645B1 (es) * 2000-03-23 2003-10-01 Alcala Farma S L Lab Forma farmaceutica solida de administracion oral de una sal de metamizol soluble en agua, procedimiento para su obtencion y forma de presentacion de dicha forma farmaceutica.
DE10026698A1 (de) * 2000-05-30 2001-12-06 Basf Ag Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
US7842308B2 (en) 2001-01-30 2010-11-30 Smithkline Beecham Limited Pharmaceutical formulation
US7883721B2 (en) 2001-01-30 2011-02-08 Smithkline Beecham Limited Pharmaceutical formulation
GB0102342D0 (en) 2001-01-30 2001-03-14 Smithkline Beecham Plc Pharmaceutical formulation
US20050175687A1 (en) * 2001-01-30 2005-08-11 Mcallister Stephen M. Pharmaceutical formulations
EP1530457B1 (en) 2002-08-12 2009-09-09 Bend Research, Inc. Pharmaceutical compositions of drugs in semi-ordered form and polymers
TW200526274A (en) 2003-07-21 2005-08-16 Smithkline Beecham Plc Pharmaceutical formulations
US8377952B2 (en) 2003-08-28 2013-02-19 Abbott Laboratories Solid pharmaceutical dosage formulation
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
GB0403098D0 (en) 2004-02-12 2004-03-17 Euro Celtique Sa Extrusion
TW201240679A (en) * 2004-03-12 2012-10-16 Capsugel Belgium Nv Pharmaceutical formulations
US20070043097A1 (en) * 2005-07-18 2007-02-22 Horizon Therapeutics, Inc. Medicaments containing famotidine and ibuprofen and administration of same
GB2447898B (en) * 2007-03-24 2011-08-17 Reckitt Benckiser Healthcare A tablet having improved stability with at least two actives
JP2011503048A (ja) 2007-11-08 2011-01-27 グラクソ グループ リミテッド 医薬製剤
US20100074947A1 (en) * 2008-06-13 2010-03-25 Adrian Brown Pharmaceutical Formulations
JP5499703B2 (ja) * 2009-12-28 2014-05-21 ライオン株式会社 イブプロフェン含有製剤
US20110236465A1 (en) * 2010-03-26 2011-09-29 Hall Mark J Melt-extruded film
KR101837927B1 (ko) * 2010-03-26 2018-03-13 다우 글로벌 테크놀로지스 엘엘씨 용융-압출된 필름

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3612212A1 (de) * 1986-04-11 1987-10-15 Basf Ag Verfahren zur herstellung von festen pharmazeutischen formen
DE3830355A1 (de) * 1988-09-07 1990-03-15 Basf Ag Verfahren zur herstellung von pharmazeutischen tabletten
DK0607467T3 (da) * 1992-12-01 1999-12-13 Spirig Ag Lægemidler, der indeholder S(+)-ibuprofen
GB9302259D0 (en) * 1993-02-05 1993-03-24 Cerestar Holding Bv Starch based material
DE19509807A1 (de) * 1995-03-21 1996-09-26 Basf Ag Verfahren zur Herstellung von Wirkstoffzubereitungen in Form einer festen Lösung des Wirkstoffs in einer Polymermatrix sowie mit diesem Verfahren hergestellte Wirkstoffzubereitungen
DE4418837A1 (de) * 1994-05-30 1995-12-07 Bayer Ag Thermisches Granulierverfahren

Also Published As

Publication number Publication date
NO974338L (no) 1997-09-19
DE19509805A1 (de) 1996-09-26
EA000434B1 (ru) 1999-08-26
KR19980703160A (ko) 1998-10-15
HU221614B (hu) 2002-11-28
ES2151150T3 (es) 2000-12-16
HUP9801152A3 (en) 2000-06-28
CA2213719A1 (en) 1996-09-26
GR3034441T3 (en) 2000-12-29
DK0817612T3 (da) 2000-11-20
IL117531A0 (en) 1996-07-23
CA2213719C (en) 2005-01-11
BR9607867A (pt) 1998-06-30
PT817612E (pt) 2001-03-30
CZ280297A3 (cs) 1998-03-18
IL117531A (en) 2000-01-31
WO1996029053A1 (de) 1996-09-26
CZ286011B6 (cs) 1999-12-15
ZA962241B (en) 1997-09-22
MX9706652A (es) 1997-11-29
JPH11502209A (ja) 1999-02-23
AU5105396A (en) 1996-10-08
EP0817612A1 (de) 1998-01-14
TW416850B (en) 2001-01-01
ATE196078T1 (de) 2000-09-15
NO318236B1 (no) 2005-02-21
US6063821A (en) 2000-05-16
DE59605848D1 (de) 2000-10-12
NO974338D0 (no) 1997-09-19
EP0817612B1 (de) 2000-09-06
HUP9801152A2 (hu) 1998-08-28

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): RU