EA034288B1 - Система доставки лекарственного средства - Google Patents

Info

Publication number

EA034288B1

EA034288B1 EA201391689A EA201391689A EA034288B1 EA 034288 B1 EA034288 B1 EA 034288B1 EA 201391689 A EA201391689 A EA 201391689A EA 201391689 A EA201391689 A EA 201391689A EA 034288 B1 EA034288 B1 EA 034288B1

Authority

EA

Eurasian Patent Office

Prior art keywords

testosterone

shell

active ingredient

drug delivery

core

Prior art date

2011-05-13

Links

• Espacenet
• Global Dossier
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• 238000012377 drug delivery Methods 0.000 title claims abstract description 134
• MUMGGOZAMZWBJJ-DYKIIFRCSA-N Testostosterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 MUMGGOZAMZWBJJ-DYKIIFRCSA-N 0.000 claims abstract description 579
• 229960003604 testosterone Drugs 0.000 claims abstract description 290
• 239000004480 active ingredient Substances 0.000 claims abstract description 146
• ZZSNKZQZMQGXPY-UHFFFAOYSA-N Ethyl cellulose Chemical compound CCOCC1OC(OC)C(OCC)C(OCC)C1OC1C(O)C(O)C(OC)C(CO)O1 ZZSNKZQZMQGXPY-UHFFFAOYSA-N 0.000 claims abstract description 81
• HQKMJHAJHXVSDF-UHFFFAOYSA-L magnesium stearate Chemical compound [Mg+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O HQKMJHAJHXVSDF-UHFFFAOYSA-L 0.000 claims abstract description 42
• 229920000168 Microcrystalline cellulose Polymers 0.000 claims abstract description 41
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• ODLHGICHYURWBS-LKONHMLTSA-N trappsol cyclo Chemical compound CC(O)COC[C@H]([C@H]([C@@H]([C@H]1O)O)O[C@H]2O[C@@H]([C@@H](O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O3)[C@H](O)[C@H]2O)COCC(O)C)O[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@@H]3O[C@@H]1COCC(C)O ODLHGICHYURWBS-LKONHMLTSA-N 0.000 claims abstract description 9
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