EA028031B1 - Твердая форма производного дигидропиридооксазина - Google Patents

Твердая форма производного дигидропиридооксазина Download PDF

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Publication number
EA028031B1
EA028031B1 EA201591023A EA201591023A EA028031B1 EA 028031 B1 EA028031 B1 EA 028031B1 EA 201591023 A EA201591023 A EA 201591023A EA 201591023 A EA201591023 A EA 201591023A EA 028031 B1 EA028031 B1 EA 028031B1
Authority
EA
Eurasian Patent Office
Prior art keywords
activity
compounds
pyrido
mediated
column
Prior art date
Application number
EA201591023A
Other languages
English (en)
Russian (ru)
Other versions
EA201591023A1 (ru
Inventor
Констанце Хурт
Кристоф Калис
Карен Каммертэн
Николя Солдерманн
Фредерик Зекри
Original Assignee
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Новартис Аг filed Critical Новартис Аг
Priority claimed from PCT/IB2013/060412 external-priority patent/WO2014102630A1/en
Publication of EA201591023A1 publication Critical patent/EA201591023A1/ru
Publication of EA028031B1 publication Critical patent/EA028031B1/ru

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Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
EA201591023A 2012-11-26 2013-11-26 Твердая форма производного дигидропиридооксазина EA028031B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GC201222895 2012-11-26
PCT/IB2013/060412 WO2014102630A1 (en) 2012-11-26 2013-11-26 Solid form of dihydro-pyrido-oxazine derivative

Publications (2)

Publication Number Publication Date
EA201591023A1 EA201591023A1 (ru) 2015-09-30
EA028031B1 true EA028031B1 (ru) 2017-09-29

Family

ID=54198861

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201591023A EA028031B1 (ru) 2012-11-26 2013-11-26 Твердая форма производного дигидропиридооксазина

Country Status (8)

Country Link
JP (1) JP6310474B2 (es)
EA (1) EA028031B1 (es)
ES (1) ES2643902T3 (es)
HR (1) HRP20171573T1 (es)
HU (1) HUE036665T2 (es)
LT (1) LT2928896T (es)
MA (1) MA38100A1 (es)
SI (1) SI2928896T1 (es)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013093849A1 (en) * 2011-12-22 2013-06-27 Novartis Ag Dihydro-benzo-oxazine and dihydro-pyrido-oxazine derivatives

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2010027002A1 (ja) * 2008-09-05 2012-02-02 塩野義製薬株式会社 Ｐｉ３ｋ阻害活性を有する縮環モルホリン誘導体

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013093849A1 (en) * 2011-12-22 2013-06-27 Novartis Ag Dihydro-benzo-oxazine and dihydro-pyrido-oxazine derivatives

Also Published As

Publication number Publication date
JP2016502531A (ja) 2016-01-28
LT2928896T (lt) 2017-09-25
MA38100A1 (fr) 2017-12-29
EA201591023A1 (ru) 2015-09-30
ES2643902T3 (es) 2017-11-27
JP6310474B2 (ja) 2018-04-11
SI2928896T1 (sl) 2017-10-30
HRP20171573T1 (hr) 2017-11-17
HUE036665T2 (hu) 2018-07-30

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KG TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): BY KZ