EA015073B1 - Комбинированные препараты, содержащие slv308 и l-dopa - Google Patents
Комбинированные препараты, содержащие slv308 и l-dopa Download PDFInfo
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- EA015073B1 EA015073B1 EA200970021A EA200970021A EA015073B1 EA 015073 B1 EA015073 B1 EA 015073B1 EA 200970021 A EA200970021 A EA 200970021A EA 200970021 A EA200970021 A EA 200970021A EA 015073 B1 EA015073 B1 EA 015073B1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
- A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US81405106P | 2006-06-16 | 2006-06-16 | |
| EP06115583 | 2006-06-16 | ||
| PCT/EP2007/055955 WO2007144421A1 (fr) | 2006-06-16 | 2007-06-15 | Préparations combinées contenant le slv308 et de la l-dopa |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200970021A1 EA200970021A1 (ru) | 2009-06-30 |
| EA015073B1 true EA015073B1 (ru) | 2011-04-29 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200970021A EA015073B1 (ru) | 2006-06-16 | 2007-06-15 | Комбинированные препараты, содержащие slv308 и l-dopa |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP2035002A1 (fr) |
| JP (1) | JP2009539941A (fr) |
| KR (1) | KR20090031908A (fr) |
| AU (1) | AU2007259255A1 (fr) |
| CA (1) | CA2654719A1 (fr) |
| EA (1) | EA015073B1 (fr) |
| IL (1) | IL195532A0 (fr) |
| MY (1) | MY148457A (fr) |
| NO (1) | NO20090164L (fr) |
| WO (1) | WO2007144421A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0027020D0 (en) | 2000-11-03 | 2000-12-20 | Univ Manchester | Treatment of movement disorders |
| US20090247537A1 (en) * | 2008-03-25 | 2009-10-01 | William Dale Overfield | Methods for preventing or treating bruxism using dopaminergic agents |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050234389A1 (en) * | 2004-03-26 | 2005-10-20 | Bouwstra Johanna A | Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds |
| WO2006032202A1 (fr) * | 2004-09-21 | 2006-03-30 | Shandong Luye Pharmaceutical Co., Ltd. | Formulation à libération lente et prolongée contenant un agoniste du récepteur de la dopamine et son procédé de préparation |
| WO2007023141A1 (fr) * | 2005-08-22 | 2007-03-01 | Solvay Pharmaceuticals B.V. | N-oxydes utilises en tant que promedicaments de derives de piperazine et de piperidine |
-
2007
- 2007-06-15 EA EA200970021A patent/EA015073B1/ru not_active IP Right Cessation
- 2007-06-15 AU AU2007259255A patent/AU2007259255A1/en not_active Abandoned
- 2007-06-15 CA CA002654719A patent/CA2654719A1/fr not_active Abandoned
- 2007-06-15 JP JP2009514809A patent/JP2009539941A/ja active Pending
- 2007-06-15 EP EP07730193A patent/EP2035002A1/fr not_active Withdrawn
- 2007-06-15 KR KR1020097001024A patent/KR20090031908A/ko not_active Application Discontinuation
- 2007-06-15 WO PCT/EP2007/055955 patent/WO2007144421A1/fr active Search and Examination
- 2007-06-15 MY MYPI20085078A patent/MY148457A/en unknown
-
2008
- 2008-11-26 IL IL195532A patent/IL195532A0/en unknown
-
2009
- 2009-01-12 NO NO20090164A patent/NO20090164L/no not_active Application Discontinuation
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050234389A1 (en) * | 2004-03-26 | 2005-10-20 | Bouwstra Johanna A | Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds |
| WO2006032202A1 (fr) * | 2004-09-21 | 2006-03-30 | Shandong Luye Pharmaceutical Co., Ltd. | Formulation à libération lente et prolongée contenant un agoniste du récepteur de la dopamine et son procédé de préparation |
| WO2007023141A1 (fr) * | 2005-08-22 | 2007-03-01 | Solvay Pharmaceuticals B.V. | N-oxydes utilises en tant que promedicaments de derives de piperazine et de piperidine |
Non-Patent Citations (8)
| Title |
|---|
| DATABASE BIOSIS [Online] BIOSCIENCES INFORMATION SERVICE, PHILADELPHIA, PA, US; 2001, HESSELINK M. ET AL.: "SLV308, a molecule combining potent partial dopamine D2 receptor agonism with serotonin 5-HT1A receptor agonism: In vitro and in vivo neurochemistry" XP002412435 Database accession no. PREV200100499786 abstract & SOCIETY FOR NEUROSCIENCE ABSTRACTS, vol. 27, no. 1, 2001, page 531, 31ST ANNUAL MEETING OF THE SOCIETY FOR NEUROSCIENCE; SAN DIEGO, CALIFORNIA, USA; NOVEMBER 10-15, 2001 ISSN: 0190-5295 * |
| DATABASE BIOSIS [Online] BIOSCIENCES INFORMATION SERVICE, PHILADELPHIA, PA, US; 2001, JOHNSTON L.C. ET AL.: "SLV308: Antiparkinsonian effects in the MPTP-treated common marmoset (Callithrix jacchus)" XP002412436 Database accession no. PREV200100499785 abstract & SOCIETY FOR NEUROSCIENCE ABSTRACTS, vol. 27, no. 1, 2001, page 531, 31ST ANNUAL MEETING OF THE SOCIETY FOR NEUROSCIENCE; SAN DIEGO, CALIFORNIA, USA; NOVEMBER 10-15, 2001 ISSN: 0190-5295 * |
| DATABASE WPI Week 200626 Derwent Publications Ltd., London, GB; AN 2006-253555 XP002412438 & WO-A1-2006032202 * |
| JOHNSTON L.C. ET AL.: "THE NOVEL DOPAMINE D2 RECEPTOR PARTIAL AGONIST, SLV-308, REVERSES MOTOR DISABILITY IN MPTP-LESIONED COMMON MARMOSETS (CALLITHRIXJACCHUS)" BRITISH JOURNAL OF PHARMACOLOGY, BASINGSTOKE, HANTS, GB, vol. 133, no. SUPPL, May 2001 (2001-05), pages U-70, AN134P, XP001061442 ISSN: 0007-1188 the whole document * |
| JOST W.H. ET AL.: "Efficacy and tolerability of Stalevo (R) 1n patients with Parkinson's disease experiencing wearing-off" AKTUELLE NEUROLOGIE, THIEME, STUTTGART, DE, vol. 32, no. Suppl 6, November 2005 (2005-11), pages S318-S325, XP009074453 ISSN: 0302-4350 abstract * |
| MCCREARY A.C. ET AL.: "SLV308: A NOVEL ANTIPARKINSONIAN AGENT WITH ANTIDEPRESSANT AND ANXIOLYTIC EFFICACY" ABSTRACTS OF THE SOCIETY FOR NEUROSCIENCE, SOCIETY FOR NEUROSCIENCE, WASHINGTON, DC, US, vol. 27, no. 1, 2001, page 531, XP001197381 ISSN: 0190-5295 the whole document * |
| OLBRICH R. ET AL.: "ANTIPARKINSONIAN ANTIDEPRESSANT ANXIOLYTIC DOPAMINE D2 PARTIAL AGONIST 5-HT 1A AGONIST 7-(4-METHYL-l-PIPERAZINYL)BENZOXAZOL-2(3H)-ONE MONOHYDROCHIORIDE AN EVALUATION OF THE PARTIAL DOPAMINE AGONIST TERGURIDE REGARDING POSITIVE SYMPTOMS REDUCTION IN SCH" DRUGS OF THE FUTURE, BARCELONA, ES, vol. 26, no. 2, 2001, pages 128-132, XP001061489 ISSN: 0377-8282 page 128, right-hand column - page 129, left-hand column * |
| WOLF W.A.: "SLV-308 SOLVAY" CURRENT OPINION IN INVESTIGATIONAL DRUGS, PHARMAPRESS, US, vol. 4, no. 7, 1 July 2003 (2003-07-01), pages 878-882, XP008033520 ISSN: 1472-4472 page 879 - page 880 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2035002A1 (fr) | 2009-03-18 |
| WO2007144421A1 (fr) | 2007-12-21 |
| NO20090164L (no) | 2009-01-14 |
| MY148457A (en) | 2013-04-30 |
| JP2009539941A (ja) | 2009-11-19 |
| AU2007259255A1 (en) | 2007-12-21 |
| KR20090031908A (ko) | 2009-03-30 |
| IL195532A0 (en) | 2009-09-01 |
| EA200970021A1 (ru) | 2009-06-30 |
| CA2654719A1 (fr) | 2007-12-21 |
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