DZ3055A1 - Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant. - Google Patents

Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant.

Info

Publication number
DZ3055A1
DZ3055A1 DZ000113A DZ000113A DZ3055A1 DZ 3055 A1 DZ3055 A1 DZ 3055A1 DZ 000113 A DZ000113 A DZ 000113A DZ 000113 A DZ000113 A DZ 000113A DZ 3055 A1 DZ3055 A1 DZ 3055A1
Authority
DZ
Algeria
Prior art keywords
polymorphs
bicyclo
oct
pharmaceutical compositions
compositions containing
Prior art date
Application number
DZ000113A
Other languages
English (en)
Inventor
Douglas John Meldrum Allen
Troy Anthony Appleton
Michael John Gumkoswki
David Joseph Muehlbauer
Timothy Norris
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DZ3055A1 publication Critical patent/DZ3055A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/02Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DZ000113A 1999-06-22 2000-06-21 Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant. DZ3055A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14023399P 1999-06-22 1999-06-22

Publications (1)

Publication Number Publication Date
DZ3055A1 true DZ3055A1 (fr) 2004-03-27

Family

ID=22490317

Family Applications (1)

Application Number Title Priority Date Filing Date
DZ000113A DZ3055A1 (fr) 1999-06-22 2000-06-21 Polymorphes d'un chlorhydrate d'azo-bicyclo-2,2,2-oct-3-ylamine cristallins et compositions pharmaceutiques les contenant.

Country Status (35)

Country Link
US (1) US6262067B1 (fr)
EP (1) EP1187834A1 (fr)
JP (1) JP2003502425A (fr)
KR (1) KR20020030280A (fr)
CN (1) CN1390216A (fr)
AP (1) AP2001002367A0 (fr)
AR (1) AR024411A1 (fr)
AU (1) AU767336B2 (fr)
BG (1) BG106205A (fr)
BR (1) BR0011835A (fr)
CA (1) CA2375265A1 (fr)
CO (1) CO5190663A1 (fr)
CZ (1) CZ20014458A3 (fr)
DZ (1) DZ3055A1 (fr)
EA (1) EA004264B1 (fr)
EC (1) ECSP003538A (fr)
EE (1) EE200100698A (fr)
HR (1) HRP20010920A2 (fr)
HU (1) HUP0201694A3 (fr)
IL (1) IL146410A0 (fr)
IS (1) IS6161A (fr)
MA (1) MA26744A1 (fr)
MX (1) MXPA02000033A (fr)
NO (1) NO20016187L (fr)
NZ (1) NZ515348A (fr)
OA (1) OA11952A (fr)
PA (1) PA8496701A1 (fr)
PE (1) PE20010322A1 (fr)
PL (1) PL352899A1 (fr)
SK (1) SK18672001A3 (fr)
TN (1) TNSN00137A1 (fr)
TR (1) TR200103688T2 (fr)
UY (1) UY26211A1 (fr)
WO (1) WO2000078759A1 (fr)
ZA (1) ZA200110387B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6387925B1 (en) * 1999-06-01 2002-05-14 Pfizer Inc. Polymorphs of a crystalline azo-bicyclo (2.2.2) oct-3-yl amine citrate and their pharmaceutical compositions
US6939873B2 (en) * 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
US6756379B2 (en) 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
WO2004031191A1 (fr) * 2002-10-04 2004-04-15 Merck Sharp & Dohme Limited Derives de spiroether azabicyclique utilises en tant qu'antagonistes du recepteur nk-1
EP1569627B1 (fr) * 2002-12-11 2008-11-12 Taro Pharmaceutical Industries Ltd. Methode de traitement de troubles moteurs a l'aide de derives de l'acide barbiturique
EP1781624A4 (fr) * 2004-07-02 2010-06-23 Taro Pharma Ind Procede de preparation d'acide 1-methoxymethyl-5,5-diphenylbarbiturique
EP2081576A4 (fr) * 2006-11-14 2010-06-30 Taro Pharmaceuticals North Ame Procédé d'amélioration de la biodisponibilité pour les barbituriques non sédatifs
UA102128C2 (en) * 2008-12-05 2013-06-10 Х. Луннбек А/С Nalmefene hydrochloride dihydrate

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX18467A (es) * 1988-11-23 1993-07-01 Pfizer Agentes terapeuticos de quinuclidinas
CA2102179C (fr) * 1991-05-31 1998-10-27 Fumitaka Ito Derives quinuclidine
EP0668863B1 (fr) * 1992-11-12 1997-01-08 Pfizer Inc. Derive de quinuclidine utilise en tant qu'antagoniste de la substance p
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis

Also Published As

Publication number Publication date
HRP20010920A2 (en) 2003-02-28
EA004264B1 (ru) 2004-02-26
CA2375265A1 (fr) 2000-12-28
KR20020030280A (ko) 2002-04-24
PE20010322A1 (es) 2001-03-14
TR200103688T2 (tr) 2002-12-23
HUP0201694A2 (en) 2002-09-28
SK18672001A3 (sk) 2002-08-06
TNSN00137A1 (fr) 2002-05-30
NZ515348A (en) 2003-07-25
CO5190663A1 (es) 2002-08-29
IL146410A0 (en) 2002-07-25
UY26211A1 (es) 2001-01-31
AR024411A1 (es) 2002-10-02
JP2003502425A (ja) 2003-01-21
CZ20014458A3 (cs) 2002-03-13
BR0011835A (pt) 2002-03-05
BG106205A (bg) 2002-07-31
OA11952A (en) 2006-04-13
HUP0201694A3 (en) 2002-10-28
NO20016187D0 (no) 2001-12-18
AU4774500A (en) 2001-01-09
US6262067B1 (en) 2001-07-17
MXPA02000033A (es) 2002-07-02
AP2001002367A0 (en) 2001-12-31
MA26744A1 (fr) 2004-12-20
WO2000078759A1 (fr) 2000-12-28
ZA200110387B (en) 2002-12-19
PL352899A1 (en) 2003-09-22
EE200100698A (et) 2003-02-17
ECSP003538A (es) 2002-01-25
CN1390216A (zh) 2003-01-08
EP1187834A1 (fr) 2002-03-20
EA200101179A1 (ru) 2002-06-27
IS6161A (is) 2001-11-13
PA8496701A1 (es) 2002-07-30
NO20016187L (no) 2001-12-18
AU767336B2 (en) 2003-11-06

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