DK539980A - Fremgangsmaade til fremstilling af 2-metyl-6-substituerede-4-i (2,3-diklorfenyl-1,4-dihydropyridin)-3,5-dikarboxylsyre-3,5-destere - Google Patents
Fremgangsmaade til fremstilling af 2-metyl-6-substituerede-4-i (2,3-diklorfenyl-1,4-dihydropyridin)-3,5-dikarboxylsyre-3,5-destereInfo
- Publication number
- DK539980A DK539980A DK539980A DK539980A DK539980A DK 539980 A DK539980 A DK 539980A DK 539980 A DK539980 A DK 539980A DK 539980 A DK539980 A DK 539980A DK 539980 A DK539980 A DK 539980A
- Authority
- DK
- Denmark
- Prior art keywords
- desters
- dichlorphenyl
- dihydropyridine
- substituted
- methyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- General Health & Medical Sciences (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE7910521A SE7910521L (sv) | 1979-12-20 | 1979-12-20 | Nya 2-metyl-6-substituerade-4-(2,3-disubstituerad fenyl)-1,4-dihydropyridin-3,5-diestrar med hypotesiva egenskaper, samt forfarande for deras framstellning, och farmaceutiska beredningar innehallande desamma |
Publications (1)
Publication Number | Publication Date |
---|---|
DK539980A true DK539980A (da) | 1981-06-21 |
Family
ID=20339605
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK539980A DK539980A (da) | 1979-12-20 | 1980-12-18 | Fremgangsmaade til fremstilling af 2-metyl-6-substituerede-4-i (2,3-diklorfenyl-1,4-dihydropyridin)-3,5-dikarboxylsyre-3,5-destere |
Country Status (11)
Country | Link |
---|---|
EP (1) | EP0031801A3 (da) |
JP (1) | JPS56127356A (da) |
AU (1) | AU6542380A (da) |
DD (1) | DD155519A5 (da) |
DK (1) | DK539980A (da) |
ES (4) | ES8204720A1 (da) |
FI (1) | FI803984L (da) |
MY (1) | MY8500404A (da) |
NO (1) | NO803856L (da) |
SE (1) | SE7910521L (da) |
ZA (1) | ZA807634B (da) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3018259A1 (de) * | 1980-05-13 | 1981-11-19 | Bayer Ag, 5090 Leverkusen | 1,4-dihydropyridine mit unterschiedlichen substituenten in 2- und 6-position, verfahren zu ihrer herstellung und ihre verwendung in arzneimitteln |
DK161312C (da) * | 1982-03-11 | 1991-12-09 | Pfizer | Analogifremgangsmaade til fremstilling af 2-aminoalkoxymethyl-4-phenyl-6-methyl-1,4-dihydropyridin-3,5-dicarboxylsyreestere eller syreadditionssalte deraf samt phthalimidoderivater til anvendelse som udgangsmateriale ved fremgangsmaaden |
IL68604A0 (en) * | 1982-05-21 | 1983-09-30 | Haessle Ab | Processes for preparing therapeutically active dihydropyridines and intermediates for the processes |
EP0100189B1 (en) * | 1982-07-22 | 1986-05-28 | Pfizer Limited | Dihydropyridine anti-ischaemic and antihypertensive agents |
HU192166B (en) * | 1982-08-06 | 1987-05-28 | Banyu Pharma Co Ltd | Process for producing 2-carbamoyl-oxy-alkyl-1,4-dihydro-pyridine derivatives |
EP0107293A3 (en) * | 1982-09-04 | 1984-06-06 | Pfizer Limited | Dihydropyridines |
PH19166A (en) * | 1982-09-04 | 1986-01-16 | Pfizer | Dihydropyridined,pharmaceutical compositions and method of use |
PL140573B1 (en) * | 1982-12-21 | 1987-05-30 | Pfizer | Method of obtaining new dihydropyridine derivatives |
US4515799A (en) * | 1983-02-02 | 1985-05-07 | Pfizer Inc. | Dihydropyridine anti-ischaemic and antihypertensive agents |
GB8306666D0 (en) * | 1983-03-10 | 1983-04-13 | Pfizer Ltd | Therapeutic agents |
GB8412208D0 (en) * | 1984-05-12 | 1984-06-20 | Pfizer Ltd | Quinolone inotropic agents |
GB8415386D0 (en) * | 1984-06-15 | 1984-07-18 | Pfizer Ltd | Therapeutic agents |
GB8526411D0 (en) * | 1985-10-25 | 1985-11-27 | Pfizer Ltd | Dihydropyridines |
GB8527698D0 (en) * | 1985-11-09 | 1985-12-11 | Pfizer Ltd | Dihydropyridine antiischaemic & antihypertensive agents |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2117572C3 (de) * | 1971-04-10 | 1980-03-20 | Bayer Ag, 5090 Leverkusen | Unsymmetrische 1,4-Dihydropyridin ^-dicarbonsäureester, Verfahren zu ihrer Herstellung sowie ihre Verwendung als Arzneimittel |
SE429652B (sv) * | 1978-06-30 | 1983-09-19 | Haessle Ab | 2.6-dimetyl-4-(2.3-diklorfenyl)-1.4-dihydropyridin-3.5-dikarboxylsyra-3-metylester-5-etylester |
CA1117117A (en) * | 1978-10-10 | 1982-01-26 | Fujisawa Pharmaceutical Co., Ltd. | 2-methyl-dihydropyridine compound, processes for preparation thereof and pharmaceutical composition comprising the same |
-
1979
- 1979-12-20 SE SE7910521A patent/SE7910521L/xx not_active Application Discontinuation
-
1980
- 1980-12-05 ZA ZA00807634A patent/ZA807634B/xx unknown
- 1980-12-16 AU AU65423/80A patent/AU6542380A/en not_active Abandoned
- 1980-12-16 EP EP80850190A patent/EP0031801A3/en not_active Withdrawn
- 1980-12-18 DK DK539980A patent/DK539980A/da unknown
- 1980-12-18 NO NO803856A patent/NO803856L/no unknown
- 1980-12-19 DD DD80226363A patent/DD155519A5/de unknown
- 1980-12-19 FI FI803984A patent/FI803984L/fi not_active Application Discontinuation
- 1980-12-19 ES ES497927A patent/ES8204720A1/es not_active Expired
- 1980-12-20 JP JP18180980A patent/JPS56127356A/ja active Pending
-
1981
- 1981-12-16 ES ES508025A patent/ES508025A0/es active Granted
- 1981-12-16 ES ES508024A patent/ES508024A0/es active Granted
- 1981-12-16 ES ES508031A patent/ES508031A0/es active Granted
-
1985
- 1985-12-30 MY MY404/85A patent/MY8500404A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
NO803856L (no) | 1981-06-22 |
EP0031801A3 (en) | 1981-09-16 |
ES497927A0 (es) | 1982-05-01 |
EP0031801A2 (en) | 1981-07-08 |
ES8306109A1 (es) | 1982-10-01 |
ZA807634B (en) | 1981-11-25 |
ES8307221A1 (es) | 1982-11-01 |
JPS56127356A (en) | 1981-10-06 |
DD155519A5 (de) | 1982-06-16 |
MY8500404A (en) | 1985-12-31 |
ES8204720A1 (es) | 1982-05-01 |
ES508031A0 (es) | 1982-10-01 |
ES8307220A1 (es) | 1982-11-16 |
SE7910521L (sv) | 1981-06-21 |
FI803984L (fi) | 1981-06-21 |
ES508024A0 (es) | 1982-11-16 |
ES508025A0 (es) | 1982-11-01 |
AU6542380A (en) | 1981-06-25 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK172182A (da) | Fremgangsmaade til fremstilling af 1,4-dihydropyridinderivater | |
DK143491A (da) | Fremgangsmaade til fremstilling af 3-oen-phenylacetylaminopiperidinaa-2,6-dion | |
DK539980A (da) | Fremgangsmaade til fremstilling af 2-metyl-6-substituerede-4-i (2,3-diklorfenyl-1,4-dihydropyridin)-3,5-dikarboxylsyre-3,5-destere | |
DK379985D0 (da) | Fremgangsmaade til fremstilling af 6-chlor-n-methyl-2,3,4,5-tetrahydro-lh-benzazepin | |
DK149855C (da) | Analogifremgangsmaade til fremstilling af 1,4-dihydropyridinderivater | |
DK364880A (da) | Fremgangsmaade til fremstilling af 6-pyridinyl-3-(2h)-pyridazioner | |
DK157855C (da) | Fremgangsmaade til fremstilling af 2,3-dichlor-5-trichlormethylpyridin | |
DK159787C (da) | Fremgangsmaade til fremstilling af 3',4'-dideoxykanamycin b | |
DK400381A (da) | Fremgansmaade til fremstilling af penicillanoyloxymethyl-penicillanoyloxymethyl-penicillanat-1,1,1!,1!-tetraoxid | |
DK159681A (da) | Fremgangsmaade til fremstilling af 4,5-diaryl-alfa-(polyfluoralkyl)-1h-pyrrol-2-methanaminer | |
DK142080C (da) | Fremgangsmaade til fremstilling af 1-azolyl-3,3-dimethyl-1-phenoxy-butan-2-oner | |
DK174380A (da) | Fremgangsmaade til fremstilling af 2!,6!adialkyl-n-alkoxymethyl-2-chlor-acetanillider | |
DK454579A (da) | Fremgangsmaade til fremstilling af 6-piperidino-2,4-diaminopyrimidin-3-oxid | |
DK154207C (da) | Fremgangsmaade til fremstilling af 1,8-dihydroxy-10-acyl-9-anthroner | |
DK113483A (da) | Fremgangsmaade til fremstilling af 3,4-diphenyl-5-methylpyrazolderivater | |
DK418079A (da) | Fremgangsmaade til fremstilling af 3,3-substituerede spiro-1,2,4-benzothiadiaziner | |
DK313580A (da) | Fremgangsmaade til fremstilling af 1,2-dihydro-2-oxo-5-(pyridinyl) nicotinonitriler | |
DK283381A (da) | Fremgangsmaade til fremstilling af 1,2,4-triazinylthiomethyl-3-cephem-sulfoxid | |
DK154085C (da) | Fremgangsmaade til fremstilling af 1,1-dioxopenicillansyrederivater | |
DK143346C (da) | Fremgangsmaade til fremstilling af 0,0-dialkylthionophosphorsyrechlorider | |
DK513580A (da) | Fremgangsmaade til fremstilling af 4,5-diaryl-alfa (polyhalogenalkyl)-1h-imidazol-2-methanoler | |
DK375480A (da) | Fremgangsmaade til fremstilling af 1,2,4-triazol-3-thioler | |
DK149962C (da) | Fremgangsmaade til fremstilling af 2,5-diketogluconsyre | |
DK393079A (da) | Fremgangsmaade til fremstilling af n,n-dimethylaminoacetonitril | |
DK149197C (da) | Fremgangsmaade til fremstilling af d,1-beta-benzoylamido-isosmoersyre |