DK535781A - Fremgangsmaade til fremstilling af n-pyrimidinyl-carbaminsyreestre - Google Patents
Fremgangsmaade til fremstilling af n-pyrimidinyl-carbaminsyreestreInfo
- Publication number
- DK535781A DK535781A DK535781A DK535781A DK535781A DK 535781 A DK535781 A DK 535781A DK 535781 A DK535781 A DK 535781A DK 535781 A DK535781 A DK 535781A DK 535781 A DK535781 A DK 535781A
- Authority
- DK
- Denmark
- Prior art keywords
- pyrimidinyl
- preparing
- acid esters
- carbamic acid
- carbamic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19803045720 DE3045720A1 (de) | 1980-12-04 | 1980-12-04 | N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK535781A true DK535781A (da) | 1982-06-05 |
Family
ID=6118292
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK535781A DK535781A (da) | 1980-12-04 | 1981-12-03 | Fremgangsmaade til fremstilling af n-pyrimidinyl-carbaminsyreestre |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4386084A (da) |
| EP (1) | EP0053695A3 (da) |
| JP (1) | JPS57122068A (da) |
| AU (1) | AU7821981A (da) |
| DE (1) | DE3045720A1 (da) |
| DK (1) | DK535781A (da) |
| ES (1) | ES8300099A1 (da) |
| FI (1) | FI813845L (da) |
| GR (1) | GR75115B (da) |
| NO (1) | NO814138L (da) |
| PT (1) | PT74077B (da) |
| ZA (1) | ZA818370B (da) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5707996A (en) * | 1995-11-06 | 1998-01-13 | Macleod Pharmaceuticals, Inc. | Pharmaceutical solution and methods for preparation thereof |
| JP4903997B2 (ja) * | 2002-07-02 | 2012-03-28 | サザン リサーチ インスティチュート | ＦｔｓＺの阻害剤およびそれらの用途 |
| KR100822530B1 (ko) | 2004-03-05 | 2008-04-16 | 에프. 호프만-라 로슈 아게 | Ｐ2ｘ3 및 ｐ2ｘ2/3 길항물질로서의 다이아미노피리미딘 |
| JP4850913B2 (ja) * | 2005-09-01 | 2012-01-11 | エフ．ホフマン−ラ ロシュ アーゲー | Ｐ２ｘ３及びｐ２ｘ２／３調節因子としてのジアミノピリジン |
| CN101253159B (zh) * | 2005-09-01 | 2011-12-07 | 弗·哈夫曼-拉罗切有限公司 | 作为p2x3和p2x2/3调节剂的二氨基嘧啶类化合物 |
| EP1924564B1 (en) * | 2005-09-01 | 2016-11-09 | F.Hoffmann-La Roche Ag | Diaminopyrimidines as p2x3 and p2x2/3 modulators |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3919229A (en) * | 1973-07-19 | 1975-11-11 | Labaz | Pyrimidine derivatives and process for preparing the same |
| BE850974A (fr) * | 1977-02-01 | 1977-05-31 | Andreu Sa Dr | Nouveaux imides de trimethoprim et leur obtention |
| DE2709634A1 (de) * | 1977-03-05 | 1978-09-07 | Basf Ag | Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
| DE2730467A1 (de) * | 1977-07-06 | 1979-01-18 | Basf Ag | Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
| DE2730468A1 (de) * | 1977-07-06 | 1979-01-18 | Basf Ag | Neue n-pyrimidinyl-imidsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
| DE2732029A1 (de) * | 1977-07-15 | 1979-02-01 | Basf Ag | Neue amidino-benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel |
-
1980
- 1980-12-04 DE DE19803045720 patent/DE3045720A1/de not_active Withdrawn
-
1981
- 1981-10-23 EP EP81108812A patent/EP0053695A3/de not_active Withdrawn
- 1981-10-29 GR GR66414A patent/GR75115B/el unknown
- 1981-11-18 US US06/322,670 patent/US4386084A/en not_active Expired - Fee Related
- 1981-11-26 JP JP56188504A patent/JPS57122068A/ja active Pending
- 1981-12-01 FI FI813845A patent/FI813845L/fi not_active Application Discontinuation
- 1981-12-03 NO NO814138A patent/NO814138L/no unknown
- 1981-12-03 AU AU78219/81A patent/AU7821981A/en not_active Abandoned
- 1981-12-03 ES ES507682A patent/ES8300099A1/es not_active Expired
- 1981-12-03 PT PT74077A patent/PT74077B/pt unknown
- 1981-12-03 DK DK535781A patent/DK535781A/da unknown
- 1981-12-03 ZA ZA818370A patent/ZA818370B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES507682A0 (es) | 1982-10-01 |
| EP0053695A3 (de) | 1982-12-15 |
| JPS57122068A (en) | 1982-07-29 |
| FI813845L (fi) | 1982-06-05 |
| EP0053695A2 (de) | 1982-06-16 |
| GR75115B (da) | 1984-07-13 |
| PT74077A (de) | 1982-01-01 |
| US4386084A (en) | 1983-05-31 |
| AU7821981A (en) | 1982-06-10 |
| NO814138L (no) | 1982-06-07 |
| DE3045720A1 (de) | 1982-07-08 |
| ES8300099A1 (es) | 1982-10-01 |
| ZA818370B (en) | 1982-11-24 |
| PT74077B (de) | 1983-05-11 |
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