ES507682A0 - Procedimiento para preparar esteres de acidos n-pirimidinilcarbamicos. - Google Patents

Procedimiento para preparar esteres de acidos n-pirimidinilcarbamicos.

Info

Publication number
ES507682A0
ES507682A0 ES507682A ES507682A ES507682A0 ES 507682 A0 ES507682 A0 ES 507682A0 ES 507682 A ES507682 A ES 507682A ES 507682 A ES507682 A ES 507682A ES 507682 A0 ES507682 A0 ES 507682A0
Authority
ES
Spain
Prior art keywords
pirimidinyl
procedure
carbamic acids
preparing esters
esters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES507682A
Other languages
English (en)
Other versions
ES8300099A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Publication of ES507682A0 publication Critical patent/ES507682A0/es
Publication of ES8300099A1 publication Critical patent/ES8300099A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
ES507682A 1980-12-04 1981-12-03 Procedimiento para preparar esteres de acidos n-pirimidinilcarbamicos. Expired ES8300099A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803045720 DE3045720A1 (de) 1980-12-04 1980-12-04 N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
ES507682A0 true ES507682A0 (es) 1982-10-01
ES8300099A1 ES8300099A1 (es) 1982-10-01

Family

ID=6118292

Family Applications (1)

Application Number Title Priority Date Filing Date
ES507682A Expired ES8300099A1 (es) 1980-12-04 1981-12-03 Procedimiento para preparar esteres de acidos n-pirimidinilcarbamicos.

Country Status (12)

Country Link
US (1) US4386084A (es)
EP (1) EP0053695A3 (es)
JP (1) JPS57122068A (es)
AU (1) AU7821981A (es)
DE (1) DE3045720A1 (es)
DK (1) DK535781A (es)
ES (1) ES8300099A1 (es)
FI (1) FI813845L (es)
GR (1) GR75115B (es)
NO (1) NO814138L (es)
PT (1) PT74077B (es)
ZA (1) ZA818370B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5707996A (en) * 1995-11-06 1998-01-13 Macleod Pharmaceuticals, Inc. Pharmaceutical solution and methods for preparation thereof
AU2003281340B2 (en) * 2002-07-02 2009-04-09 Southern Research Institute Inhibitors of FtsZ and uses thereof
PT1725540E (pt) 2004-03-05 2012-11-29 Hoffmann La Roche Diaminopirimidinas como antagonistas de p2x3 e p2x2/3
CN101296907B (zh) * 2005-09-01 2013-03-27 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3调节剂的二氨基嘧啶类
CA2620129C (en) * 2005-09-01 2014-12-23 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
AU2006286576B2 (en) * 2005-09-01 2012-06-14 F. Hoffmann-La Roche Ag Diaminopyrimidines as P2X3 and P3X2/3 modulators

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3919229A (en) * 1973-07-19 1975-11-11 Labaz Pyrimidine derivatives and process for preparing the same
BE850974A (fr) * 1977-02-01 1977-05-31 Andreu Sa Dr Nouveaux imides de trimethoprim et leur obtention
DE2709634A1 (de) * 1977-03-05 1978-09-07 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2730468A1 (de) * 1977-07-06 1979-01-18 Basf Ag Neue n-pyrimidinyl-imidsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2730467A1 (de) * 1977-07-06 1979-01-18 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2732029A1 (de) * 1977-07-15 1979-02-01 Basf Ag Neue amidino-benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
JPS57122068A (en) 1982-07-29
PT74077B (de) 1983-05-11
DK535781A (da) 1982-06-05
AU7821981A (en) 1982-06-10
ZA818370B (en) 1982-11-24
GR75115B (es) 1984-07-13
US4386084A (en) 1983-05-31
NO814138L (no) 1982-06-07
FI813845L (fi) 1982-06-05
EP0053695A2 (de) 1982-06-16
DE3045720A1 (de) 1982-07-08
EP0053695A3 (de) 1982-12-15
ES8300099A1 (es) 1982-10-01
PT74077A (de) 1982-01-01

Similar Documents

Publication Publication Date Title
ES497979A0 (es) Procedimiento para preparar esteres de acidos ciclopropano- carboxilicos
ES490764A0 (es) Procedimiento para preparar esteres de acil-carnitinas
ES506386A0 (es) Procedimiento para la preparacion de mono-esteres amonio-al-cohilicos de acidos alcanol-fosforicos
AR231277A1 (es) Un procedimiento para la preparacion de esteres de insulina
ES514699A0 (es) Procedimiento para preparar esteres de acidos quinolina-car boxilicos.
ES495404A0 (es) Procedimiento para preparar esteres
ES2025122B3 (es) Procedimiento para obtencion de esteres de acidos alquencarboxilicos.
ES501021A0 (es) Un procedimiento para la preparacion de esteres de sililalquilo.
ES507682A0 (es) Procedimiento para preparar esteres de acidos n-pirimidinilcarbamicos.
ES492367A0 (es) Un procedimiento para la preparacion de esteres de acidos ciclohexencarboxilicos
ES520528A0 (es) Procedimiento para la obtencion de esteres de acido piridincarboxilico.
ES478785A0 (es) Procedimiento para preparar esteres de m-fenoxibencilo de a-cido 2-haloalquil (oxi-,tio-,sulfinil-o sulfonil) fenilalcanoicos.
MX5368E (es) Procedimiento para la preparacion de esteres de acidos ciclopropancarboxilicos
MX5905E (es) Procedimiento para la preparacion de esteres de acidos ciclopropancarboxilicos
MX5705E (es) Procedimiento para preparar esteres de(s) alfa-ciano-3-fenoxibencilo
ES509185A0 (es) Procedimiento para la obtencion de esteres de 4-fluor-3-halofenoxibencilo.
ES519679A0 (es) Procedimiento para la preparacion de acidos fenilamino-oxo-aceticos y sus esteres.
ES521311A0 (es) Procedimiento para preparar esteres fosfato trisustituidos.
AR221386A1 (es) Procedimiento para la preparacion de esteres basicos de acidos hidroxiciclohexancarboxilicos sustituidos
AR226118A1 (es) Procedimiento para la produccion de esteres de acidos 3-acil-azopropionicos
ES497743A0 (es) Procedimiento para la preparacion de esteres alquinilicos deacido ciclopropancarboxilico
ES498526A0 (es) Procedimiento para preparar esteres de acidos piperidina carboxilicos.
ES493355A0 (es) Un procedimiento para la preparacion de acido 1-etil-1,4-di-hidro-6-(2-naftil)-4-oxonicontinico y sus esteres
ES494168A0 (es) Un procedimiento para la preparacion de acidos alfa-aril- propionicos
ES494472A0 (es) Metodo de preparar esteres tion- y tiolcarbamicos

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20000201