DK514981A - METHOD FOR PREPARING 3-AMINO-SUBSTITUTED STEROID DERIVATIVES - Google Patents

METHOD FOR PREPARING 3-AMINO-SUBSTITUTED STEROID DERIVATIVES

Info

Publication number
DK514981A
DK514981A DK514981A DK514981A DK514981A DK 514981 A DK514981 A DK 514981A DK 514981 A DK514981 A DK 514981A DK 514981 A DK514981 A DK 514981A DK 514981 A DK514981 A DK 514981A
Authority
DK
Denmark
Prior art keywords
amino
preparing
steroid derivatives
substituted steroid
substituted
Prior art date
Application number
DK514981A
Other languages
Danish (da)
Other versions
DK161093C (en
DK161093B (en
Inventor
R Deraedt
V Torelli
J Benzoni
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK514981A publication Critical patent/DK514981A/en
Publication of DK161093B publication Critical patent/DK161093B/en
Application granted granted Critical
Publication of DK161093C publication Critical patent/DK161093C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J13/00Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027Azides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK514981A 1980-11-21 1981-11-20 ANALOGY PROCEDURE FOR THE PREPARATION OF 3-AMINO-SUBSTITUTED STEROID DERIVATIVES DK161093C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8024750A FR2494698A1 (en) 1980-11-21 1980-11-21 NOVEL SUBSTITUTED 3-AMINO STEROID DERIVATIVES, THEIR SALTS, PREPARATION METHOD, MEDICAMENT APPLICATION AND COMPOSITIONS COMPRISING THE SAME
FR8024750 1980-11-21

Publications (3)

Publication Number Publication Date
DK514981A true DK514981A (en) 1982-05-22
DK161093B DK161093B (en) 1991-05-27
DK161093C DK161093C (en) 1991-11-18

Family

ID=9248226

Family Applications (1)

Application Number Title Priority Date Filing Date
DK514981A DK161093C (en) 1980-11-21 1981-11-20 ANALOGY PROCEDURE FOR THE PREPARATION OF 3-AMINO-SUBSTITUTED STEROID DERIVATIVES

Country Status (23)

Country Link
JP (1) JPS57116099A (en)
KR (1) KR880001239B1 (en)
AT (1) AT389703B (en)
AU (1) AU546100B2 (en)
BE (1) BE891201A (en)
CA (1) CA1175415A (en)
CH (1) CH651056A5 (en)
DE (1) DE3146117A1 (en)
DK (1) DK161093C (en)
ES (1) ES8207195A1 (en)
FI (1) FI77871C (en)
FR (1) FR2494698A1 (en)
GB (1) GB2087894B (en)
HU (1) HU184896B (en)
IE (1) IE52188B1 (en)
IL (1) IL64224A0 (en)
IT (1) IT1172086B (en)
LU (1) LU83781A1 (en)
NL (1) NL8105260A (en)
PT (1) PT74015B (en)
SE (1) SE451456B (en)
SU (1) SU1327789A3 (en)
ZA (1) ZA817806B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9084800B2 (en) * 2011-11-07 2015-07-21 Natreon, Inc. Indolealkylamino-withasteroid conjugates and method of use

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2430467A (en) * 1944-02-11 1947-11-11 Glidden Co 3-amino-derivatives of steroids and method of making same
US2781342A (en) * 1952-05-17 1957-02-12 Upjohn Co Steroid enamines
GB962324A (en) * 1959-09-12 1964-07-01 Clin Byla Ets Steroid compounds and production thereof
FR1311761A (en) * 1959-09-12 1962-12-14 Clin Byla Ets Amino compounds of the steroid series and method of preparing such compounds
NL103735C (en) * 1961-02-17
US3503959A (en) * 1962-03-30 1970-03-31 Sterling Drug Inc 3-amino steroids
US3196168A (en) * 1964-02-18 1965-07-20 American Home Prod Aminoaroyl aminosteroids
BE647858A (en) * 1964-05-13
US3196169A (en) * 1964-11-03 1965-07-20 American Home Prod Aminoacyl aminosteroids
BE672238A (en) * 1965-11-12 1966-03-01
BE811304R (en) * 1973-10-24 1974-06-17 PREPARATION PROCEDURE FOR (20 S) 3 BETA -N-DIMETHYLAMINO
FR2463777A1 (en) * 1979-08-17 1981-02-27 Roussel Uclaf NOVEL DERIVATIVES OF 5A-PREGNAN-20-OL, PROCESS FOR PREPARING THEM AND THEIR APPLICATION AS MEDICAMENTS

Also Published As

Publication number Publication date
DK161093C (en) 1991-11-18
IT8149746A0 (en) 1981-11-20
AU7772381A (en) 1982-05-27
ATA497081A (en) 1989-06-15
SU1327789A3 (en) 1987-07-30
AU546100B2 (en) 1985-08-15
FR2494698A1 (en) 1982-05-28
HU184896B (en) 1984-10-29
BE891201A (en) 1982-05-21
AT389703B (en) 1990-01-25
CA1175415A (en) 1984-10-02
PT74015A (en) 1981-12-01
FR2494698B1 (en) 1983-06-24
GB2087894B (en) 1984-09-26
IE812732L (en) 1982-05-21
FI77871C (en) 1989-05-10
NL8105260A (en) 1982-06-16
KR830007716A (en) 1983-11-04
ES507309A0 (en) 1982-09-01
SE8105995L (en) 1982-05-22
FI77871B (en) 1989-01-31
SE451456B (en) 1987-10-12
IE52188B1 (en) 1987-08-05
CH651056A5 (en) 1985-08-30
FI813677L (en) 1982-05-22
DK161093B (en) 1991-05-27
PT74015B (en) 1983-11-30
LU83781A1 (en) 1982-06-30
GB2087894A (en) 1982-06-03
JPS57116099A (en) 1982-07-19
IT1172086B (en) 1987-06-18
ES8207195A1 (en) 1982-09-01
KR880001239B1 (en) 1988-07-12
IL64224A0 (en) 1982-02-28
JPH0247479B2 (en) 1990-10-19
DE3146117A1 (en) 1982-06-16
ZA817806B (en) 1982-10-27

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