DK495287D0 - 2-eller 3-arylsubstituerede imidazo(1,2-a)pyridi ner - Google Patents

2-eller 3-arylsubstituerede imidazo(1,2-a)pyridi ner

Info

Publication number
DK495287D0
DK495287D0 DK4952/87A DK495287A DK495287D0 DK 495287 D0 DK495287 D0 DK 495287D0 DK 4952/87 A DK4952/87 A DK 4952/87A DK 495287 A DK495287 A DK 495287A DK 495287 D0 DK495287 D0 DK 495287D0
Authority
DK
Denmark
Prior art keywords
pyridia
aryl
substituted imidazo
imidazo
substituted
Prior art date
Application number
DK4952/87A
Other languages
English (en)
Other versions
DK164669C (da
DK164669B (da
DK495287A (da
Inventor
B Press Jeffery
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/909,648 external-priority patent/US4727145A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of DK495287D0 publication Critical patent/DK495287D0/da
Publication of DK495287A publication Critical patent/DK495287A/da
Publication of DK164669B publication Critical patent/DK164669B/da
Application granted granted Critical
Publication of DK164669C publication Critical patent/DK164669C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK495287A 1986-09-22 1987-09-21 2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf DK164669C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US90964886 1986-09-22
US06/909,648 US4727145A (en) 1986-09-22 1986-09-22 2- Or 3- aryl substituted imidazo [1,2-a]pyridines
US07/090,111 US4791117A (en) 1986-09-22 1987-08-31 2- or 3-aryl substituted imidazo[1,2-a]pyridines and their use as calcium channel blockers
US9011187 1987-08-31

Publications (4)

Publication Number Publication Date
DK495287D0 true DK495287D0 (da) 1987-09-21
DK495287A DK495287A (da) 1988-03-23
DK164669B DK164669B (da) 1992-07-27
DK164669C DK164669C (da) 1992-12-21

Family

ID=26781926

Family Applications (1)

Application Number Title Priority Date Filing Date
DK495287A DK164669C (da) 1986-09-22 1987-09-21 2- eller 3-arylsubstituerede imidazooe1,2-aaapyridiner samt fremgangsmaader til fremstilling deraf

Country Status (5)

Country Link
US (1) US4791117A (da)
EP (1) EP0261912A3 (da)
AU (1) AU597108B2 (da)
DK (1) DK164669C (da)
IE (1) IE872541L (da)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2647451B1 (fr) * 1989-05-26 1994-08-05 Sanofi Sa Derives d'imidazo(1,2-a)pyridine, procede de preparation, compositions pharmaceutiques les contenant
DE4405378A1 (de) * 1994-02-19 1995-08-24 Merck Patent Gmbh Adhäsionsrezeptor-Antagonisten
US6541479B1 (en) * 1997-12-02 2003-04-01 Massachusetts College Of Pharmacy Calcium channel blockers
CA2311483A1 (en) 2000-06-12 2001-12-12 Gregory N Beatch IMIDAZO [1,2-A] PYRIDINIC ETHERS AND USES THEREOF
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
DE10117183A1 (de) * 2001-04-05 2002-10-10 Gruenenthal Gmbh Verwendung von substituierten Imidazo[1,2-a]-pyridinverbindungen als Arzneimittel
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
DE10247271A1 (de) * 2002-10-10 2004-08-26 Grünenthal GmbH Substituierte C-Imidazo[1,2-a]pyridin-3-yle
MXPA04008070A (es) 2003-03-10 2004-11-26 Altana Pharma Ag Novedoso proceso para la preparacion de roflumilasto.
JP5383183B2 (ja) 2005-03-16 2014-01-08 タケダ ゲゼルシャフト ミット ベシュレンクテル ハフツング ロフルミラストを含有する矯味された剤形
TW200803903A (en) * 2006-04-28 2008-01-16 Nihon Mediphysics Co Ltd Novel compound having affinity to amyloid
ES2376491T3 (es) 2006-05-19 2012-03-14 Nihon Medi-Physics Co., Ltd. Compuesto que tiene afinidad por amiloide.
EP2042501B1 (en) * 2006-06-21 2017-04-12 Nihon Medi-Physics Co., Ltd. Compound having affinity for amyloid
NZ577318A (en) * 2006-11-17 2012-04-27 Nihon Mediphysics Co Ltd Novel compounds with affinity for amyloid
TW200823211A (en) 2006-11-30 2008-06-01 Nihon Mediphysics Co Ltd Novel compound having affinity for amyloid
TWI406674B (zh) 2007-02-13 2013-09-01 Nihon Mediphysics Co Ltd Method for manufacturing diagnostic radiographic diagnostic agents
TW200918102A (en) * 2007-10-24 2009-05-01 Nihon Mediphysics Co Ltd Novel compound having affinity for amyloid
JP5313158B2 (ja) * 2007-10-26 2013-10-09 日本メジフィジックス株式会社 新規アミロイド親和性化合物
CA2704172A1 (en) * 2007-10-30 2009-05-07 Nihon Medi-Physics Co., Ltd. Use of novel compound having affinity for amyloid, and process for production of the same
JPWO2009057578A1 (ja) * 2007-10-30 2011-03-10 日本メジフィジックス株式会社 新規アミロイド親和性化合物の使用及び製造方法
EP2832234A1 (en) * 2013-07-30 2015-02-04 IMAX Discovery GmbH Imidazo[1,2-a]pyridine-ylmethyl-derivatives and their use as flavoring agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2937179A (en) * 1958-04-09 1960-05-17 Seymour L Shapiro Process for phenylimidazolino [1, 2-alpha]piperidines
GB1442707A (en) * 1973-07-07 1976-07-14 Yoshitomi Pharmaceutical Substituted phenylalkanoic acids and their derivatives and pharma ceutical compositions thereof
GB1473819A (en) * 1976-01-28 1977-05-18 Gallardo Antonio Sa Derivatives of imidazo 1,2-a pyridine
EP0068378B1 (en) * 1981-06-26 1986-03-05 Schering Corporation Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
GB8305245D0 (en) * 1983-02-25 1983-03-30 Fujisawa Pharmaceutical Co Imidazo-heterocyclic compounds
AU7928787A (en) * 1986-10-07 1988-04-14 Yamanouchi Pharmaceutical Co., Ltd. Imidazopyridine derivatives
US4831041A (en) * 1986-11-26 1989-05-16 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
ES2026666T3 (es) * 1987-03-27 1992-05-01 Synthelabo Procedimiento para preparar derivados de imidazopiridinas.

Also Published As

Publication number Publication date
US4791117A (en) 1988-12-13
IE872541L (en) 1988-03-22
EP0261912A3 (en) 1989-09-20
EP0261912A2 (en) 1988-03-30
DK164669C (da) 1992-12-21
DK164669B (da) 1992-07-27
AU7849387A (en) 1988-03-24
DK495287A (da) 1988-03-23
AU597108B2 (en) 1990-05-24

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