DK452178A - R fremgangsmaade til fremstilling af phenylethanolamin-derivate - Google Patents
R fremgangsmaade til fremstilling af phenylethanolamin-derivateInfo
- Publication number
- DK452178A DK452178A DK452178A DK452178A DK452178A DK 452178 A DK452178 A DK 452178A DK 452178 A DK452178 A DK 452178A DK 452178 A DK452178 A DK 452178A DK 452178 A DK452178 A DK 452178A
- Authority
- DK
- Denmark
- Prior art keywords
- preparing
- procedure
- phenylethanolamine derivatives
- phenylethanolamine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/64—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C43/00—Ethers; Compounds having groups, groups or groups
- C07C43/02—Ethers
- C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
- C07C43/23—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing hydroxy or O-metal groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP12203477 | 1977-10-12 | ||
| JP12203477A JPS5473751A (en) | 1977-10-12 | 1977-10-12 | Phenyl ethanolamine derivatives and their preparation |
| JP12843677A JPS5463048A (en) | 1977-10-26 | 1977-10-26 | Novel phenyl ethanolamine derivatives and their preparation |
| JP12843677 | 1977-10-26 | ||
| JP15535277A JPS5495544A (en) | 1977-12-23 | 1977-12-23 | Phenylethanolamine derivative and its preparation |
| JP15535277 | 1977-12-23 | ||
| JP7496478A JPS552639A (en) | 1978-06-21 | 1978-06-21 | Phenylethanolamine derivative and its preparation |
| JP7496478 | 1978-06-21 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK452178A true DK452178A (da) | 1979-04-13 |
| DK168484B1 DK168484B1 (da) | 1994-04-05 |
Family
ID=27465764
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK452178A DK168484B1 (da) | 1977-10-12 | 1978-10-11 | Analogifremgangsmåde til fremstilling af phenylethanolaminderivater eller fysiologisk accetable syreadditionssalte deraf |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4217305A (da) |
| AT (1) | AT363457B (da) |
| AU (1) | AU526715B2 (da) |
| CA (1) | CA1147342A (da) |
| CH (1) | CH639948A5 (da) |
| DE (1) | DE2843016A1 (da) |
| DK (1) | DK168484B1 (da) |
| ES (2) | ES474149A1 (da) |
| FR (1) | FR2405931A1 (da) |
| GB (1) | GB2006772B (da) |
| GR (1) | GR65337B (da) |
| IT (1) | IT1160853B (da) |
| NO (1) | NO147148C (da) |
| PT (1) | PT68624A (da) |
| SE (1) | SE448232B (da) |
| SU (2) | SU982537A3 (da) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55124742A (en) * | 1979-03-20 | 1980-09-26 | Kyowa Hakko Kogyo Co Ltd | Novel aminoalcohol derivative |
| US4206125A (en) * | 1979-05-04 | 1980-06-03 | Richardson-Merrell Inc. | 5-[2-[(2,3-Dihydro-1,4-benzodioxan-2-ylmethyl)amino]-1-hydroxyethyl]-2-hydroxybenzoic acid derivatives |
| DD157796A5 (de) * | 1979-12-04 | 1982-12-08 | Ciba Geigy Ag | Verfahren zur herstellung neuer derivate des 2-amino-aethanols |
| JPS56110665A (en) * | 1980-02-08 | 1981-09-01 | Yamanouchi Pharmaceut Co Ltd | Sulfamoyl-substituted phenetylamine derivative and its preparation |
| US4558156A (en) * | 1980-02-08 | 1985-12-10 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl-substituted phenethylamine derivatives |
| US5391825A (en) * | 1980-02-08 | 1995-02-21 | Yamanouchi Pharmaceutical Co., Ltd. | Sulfamoyl substituted phenethylamine intermediates |
| DE3128117A1 (de) * | 1980-07-29 | 1982-03-11 | Yamanouchi Pharmaceutical Co., Ltd., Tokyo | Neue phenyl-aethylaminderivate, verfahren zu ihrer herstellung |
| CA1219865A (en) * | 1982-05-14 | 1987-03-31 | Leo Alig | Aziridine phenethanolamine derivatives |
| PT78388B (en) * | 1983-04-12 | 1986-09-15 | Smithkline Beckman Corp | Dopamine-beta-hydroxylase inhibitors |
| JPS6051106A (ja) * | 1983-08-31 | 1985-03-22 | Yamanouchi Pharmaceut Co Ltd | 塩酸アモスラロ−ル持続性製剤 |
| EP0162404B1 (en) * | 1984-05-15 | 1988-08-24 | Seitetsu Kagaku Co., Ltd. | Process for preparing 2-alkyl-5-haloacetylbenzenesulfonamide |
| US4678855A (en) * | 1985-10-09 | 1987-07-07 | Merck & Co., Inc. | Substituted benzenesulfonamides |
| JPS62114952A (ja) * | 1985-11-13 | 1987-05-26 | Yamanouchi Pharmaceut Co Ltd | 置換フエネチルアミン誘導体の製造法 |
| EP0317206B1 (en) * | 1987-11-13 | 1993-04-28 | Glaxo Group Limited | Phenethanolamine derivatives |
| ES2137260T3 (es) * | 1992-05-22 | 1999-12-16 | Senju Pharma Co | Composicion farmaceutica para uso en el tratamiento del glaucoma. |
| FR2737494B1 (fr) * | 1995-08-04 | 1997-08-29 | Synthelabo | Derives de benzenesulfonamide, leur preparation et leur application en therapeutique |
| AU715233B2 (en) * | 1996-01-10 | 2000-01-20 | Asahi Kasei Kogyo Kabushiki Kaisha | Novel tricyclic compounds and drug compositions containing the same |
| WO1999057131A1 (en) * | 1998-05-06 | 1999-11-11 | Duke University | Method of treating bladder and lower urinary tract syndromes |
| FR2791675B1 (fr) * | 1999-03-30 | 2001-05-04 | Synthelabo | Derives de n-[2-(4-aminophenyl) ethyl] -2,3-dihydro-1,4- benzodioxinne-2-methanamine, leur preparation et leur application en therapeutique |
| US6835853B2 (en) * | 2001-10-31 | 2004-12-28 | Synthon Bv | Process for resolution of tamsulosin and compounds, compositions, and processes associated therewith |
| ES2362998T3 (es) | 2002-08-19 | 2011-07-18 | Pfizer Inc. | Terapia de combinación para enfermedades hiperproliferativas. |
| GEP20084406B (en) | 2003-05-30 | 2008-06-25 | Ranbaxy Lab Ltd | Substituted pyrrole derivatives and their use as hmg-co inhibitors |
| WO2005056521A1 (en) * | 2003-12-09 | 2005-06-23 | Cj Corporation | Method of preparing optically pure phenethylamine derivatives |
| AU2005308575A1 (en) * | 2004-11-23 | 2006-06-01 | Warner-Lambert Company Llc | 7-(2h-pyrazol-3-yl)-3, 5-dihyroxy-heptanoic acid derivatives as HMG Co-A reductase inhibitors for the treatment of lipidemia |
| GT200600381A (es) | 2005-08-25 | 2007-03-28 | Compuestos organicos | |
| US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
| AU2006313430B2 (en) | 2005-11-08 | 2012-09-06 | Ranbaxy Laboratories Limited | Process for (3R,5R)-7-[2-(4-fluorophenyl)-5-isopropyl-3-phenyl-4- [(4-hydroxy methyl phenyl amino) carbonyl]-pyrrol-1-yl]-3, 5-dihydroxy-heptanoic acid hemi calcium salt |
| US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| WO2007131804A1 (en) | 2006-05-17 | 2007-11-22 | Synthon B.V. | Tablet composition with a prolonged release of tamsulosin |
| US8404896B2 (en) | 2006-12-01 | 2013-03-26 | Bristol-Myers Squibb Company | N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
| US8465770B2 (en) * | 2008-12-24 | 2013-06-18 | Synthon Bv | Low dose controlled release tablet |
| CN102050766B (zh) * | 2009-11-03 | 2013-08-07 | 安徽省新星药物开发有限责任公司 | 一种盐酸氨磺洛尔的合成方法 |
| AU2014255381A1 (en) | 2013-04-17 | 2015-10-08 | Pfizer Inc. | N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases |
| WO2016055901A1 (en) | 2014-10-08 | 2016-04-14 | Pfizer Inc. | Substituted amide compounds |
| MX2021008533A (es) | 2019-01-18 | 2021-08-19 | Astrazeneca Ab | Inhibidores de la pcsk9 y metodos de uso de los mismos. |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3701808A (en) * | 1967-12-21 | 1972-10-31 | Allen & Hanburys Ltd | Phenylethanolamines |
| GB1266058A (da) | 1969-07-08 | 1972-03-08 | ||
| GB1321701A (en) | 1969-10-01 | 1973-06-27 | Continental Pharma | Amino-alcohols their salts and process for prepairing the same |
| US3711545A (en) * | 1971-02-23 | 1973-01-16 | Smith Kline French Lab | Alpha-aminoalkyl-4-hydroxy-3-sulfamoylaminobenzyl alcohols |
| DE2115926C3 (de) * | 1971-04-01 | 1978-05-03 | C.H. Boehringer Sohn, 6507 Ingelheim | 1 -(4-Hydroxy-3-dimethylaminosuIfamidophenyI)-2-aminoäthanderivate, Verfahren zu ihrer Herstellung und diese enthaltende Mittel |
| US4034112A (en) * | 1973-06-22 | 1977-07-05 | Imperial Chemical Industries Limited | Ethanolamine derivatives having β-adrenergic blocking activity |
| US3860647A (en) * | 1973-08-20 | 1975-01-14 | Smithkline Corp | {60 -Aminomethyl-4-hydroxy-3-sulfamyl-benzyl alcohols and 4-hydroxy-3-sulfamyl phenethylamines |
| GB1593651A (en) * | 1977-02-03 | 1981-07-22 | Allen & Hanburys Ltd | Amides |
| DK31578A (da) * | 1977-02-03 | 1978-08-04 | Allen & Hanburys Ltd | Fremgangsmaade til fremstilling af benzenderivater |
-
1978
- 1978-09-22 CA CA000311934A patent/CA1147342A/en not_active Expired
- 1978-09-25 GR GR57301A patent/GR65337B/el unknown
- 1978-09-27 US US05/946,192 patent/US4217305A/en not_active Expired - Lifetime
- 1978-10-02 CH CH1021878A patent/CH639948A5/de not_active IP Right Cessation
- 1978-10-03 DE DE19782843016 patent/DE2843016A1/de active Granted
- 1978-10-06 PT PT68624A patent/PT68624A/pt unknown
- 1978-10-09 FR FR7828743A patent/FR2405931A1/fr active Granted
- 1978-10-11 SE SE7810613A patent/SE448232B/sv not_active IP Right Cessation
- 1978-10-11 DK DK452178A patent/DK168484B1/da active
- 1978-10-11 ES ES474149A patent/ES474149A1/es not_active Expired
- 1978-10-11 SU SU782673556A patent/SU982537A3/ru active
- 1978-10-11 AT AT0731778A patent/AT363457B/de not_active IP Right Cessation
- 1978-10-11 IT IT69350/78A patent/IT1160853B/it active
- 1978-10-11 NO NO783442A patent/NO147148C/no unknown
- 1978-10-12 GB GB7840390A patent/GB2006772B/en not_active Expired
- 1978-10-12 AU AU40642/78A patent/AU526715B2/en not_active Expired
-
1979
- 1979-06-13 ES ES481549A patent/ES481549A1/es not_active Expired
- 1979-10-18 SU SU792835396A patent/SU932982A3/ru active
Also Published As
| Publication number | Publication date |
|---|---|
| US4217305A (en) | 1980-08-12 |
| ES474149A1 (es) | 1979-10-16 |
| CA1147342A (en) | 1983-05-31 |
| NO147148B (no) | 1982-11-01 |
| SU982537A3 (ru) | 1982-12-15 |
| IT1160853B (it) | 1987-03-11 |
| AU4064278A (en) | 1980-04-17 |
| SE7810613L (sv) | 1979-04-13 |
| AU526715B2 (en) | 1983-01-27 |
| GB2006772B (en) | 1982-02-03 |
| GB2006772A (en) | 1979-05-10 |
| FR2405931A1 (fr) | 1979-05-11 |
| NO147148C (no) | 1983-02-09 |
| AT363457B (de) | 1981-08-10 |
| DE2843016C2 (da) | 1988-10-13 |
| SU932982A3 (ru) | 1982-05-30 |
| DE2843016A1 (de) | 1979-04-26 |
| NO783442L (no) | 1979-04-18 |
| SE448232B (sv) | 1987-02-02 |
| DK168484B1 (da) | 1994-04-05 |
| FR2405931B1 (da) | 1982-11-19 |
| CH639948A5 (de) | 1983-12-15 |
| IT7869350A0 (it) | 1978-10-11 |
| PT68624A (en) | 1978-11-01 |
| GR65337B (en) | 1980-08-18 |
| ES481549A1 (es) | 1980-04-01 |
| ATA731778A (de) | 1981-01-15 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK452178A (da) | R fremgangsmaade til fremstilling af phenylethanolamin-derivate | |
| DK155733C (da) | Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater | |
| DK349478A (da) | Fremgangsmaade til fremstilling af oligoimider | |
| DK195378A (da) | Fremgangsmaade til fremstilling af polyenforbindelser | |
| DK269178A (da) | Analogifremgangsmaade til fremstilling af n-alkylpiperidinderivater | |
| DK536178A (da) | Fremgangsmaade til fremstilling af stilbenderivater | |
| DK539578A (da) | Fremgangsmaade til fremstilling af pleuromutilinglycsid-derivater | |
| DK155279C (da) | Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater | |
| DK531178A (da) | Fremgangsmaade til fremstilling af phenylglycinderivater | |
| DK30578A (da) | Fremgangsmaade til fremstilling af aminoalkoxyphenylderivater | |
| DK470978A (da) | R fremgangsmaade til fremstilling af pyrazinobenzoxapinderivate | |
| DK152130C (da) | Fremgangsmaade til fremstilling af benzooebaathienopyridinderivater | |
| DK494978A (da) | Fremgangsmaade til fremstilling af 2-iminoimidazolidinderivater | |
| DK50778A (da) | Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater | |
| DK97578A (da) | Fremgangsmaade til fremstilling af benzylpyrimidin-forbindelser | |
| DK50878A (da) | Fremgangsmaade til fremstilling af oxadiazolopyrimidinderivater | |
| DK520178A (da) | Fremgangsmaade til fremstilling af phenoxyalkanolamin-derivater | |
| DK385478A (da) | Fremgangsmaade til fremstilling af dibenzocycloocteniminer | |
| DK246878A (da) | Fremgangsmaade til fremstilling af acylderivater | |
| DK61778A (da) | Fremgangsmaade til fremstilling af everninominderivater | |
| DK570578A (da) | Fremgangsmaade til fremstilling af 21-hydroxy-20-methyl-pregnan-derivater | |
| DK190178A (da) | Fremgangsmaade til fremstilling af pyranoquinolinon-derivater | |
| DK144884C (da) | Fremgangsmaade til fremstilling af 3-bromphthalid | |
| DK351478A (da) | Fremgangsmaade til fremstilling af apovincamin | |
| DK521578A (da) | Fremgangsmaade til fremstilling af phenylbutenoner |