DK413180A - PROCEDURE FOR THE PREPARATION OF N- (5-TETRAZOLYL) -1-OXO-1H-THIAZOLO (3,2-A) - Google Patents
PROCEDURE FOR THE PREPARATION OF N- (5-TETRAZOLYL) -1-OXO-1H-THIAZOLO (3,2-A)Info
- Publication number
- DK413180A DK413180A DK413180A DK413180A DK413180A DK 413180 A DK413180 A DK 413180A DK 413180 A DK413180 A DK 413180A DK 413180 A DK413180 A DK 413180A DK 413180 A DK413180 A DK 413180A
- Authority
- DK
- Denmark
- Prior art keywords
- thiazolo
- tetrazolyl
- oxo
- procedure
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK13184A DK13184A (en) | 1979-11-23 | 1984-01-12 | METHOD OF ANALOGUE FOR THE PREPARATION OF 1-OXO-1H-THIAZOLO (3,2-A) PYRIMIDINE-2-CARBOXYLIC ACID OR PHARMACEUTICALLY ACCEPTABLE ANTI-CEREAL ESTATE (3-OXO-2H-THIAZOLYE) -2-THIAZOLYE (3,2-A-THIAZOLYE) AS INTERMEDIATES BY THE PROCEDURE |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US9663179A | 1979-11-23 | 1979-11-23 | |
US9663179 | 1979-11-23 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK413180A true DK413180A (en) | 1981-05-24 |
DK151811B DK151811B (en) | 1988-01-04 |
DK151811C DK151811C (en) | 1988-06-06 |
Family
ID=22258306
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK413180A DK151811C (en) | 1979-11-23 | 1980-09-30 | ANALOGY PROCEDURE FOR THE PREPARATION OF N- (5-TETRAZOLYL) -1-OXO-1H-THIAZOLOOE3,2-AAA-PYRIMIDIN-2-CARBOXAMIDES OR PHARMACEUTICALLY ACCEPTABLE COATAL SALTS THEREOF AND 1-OXO-2XO-OXO-2-OXO2 FOR USE AS THE INITIAL MATERIALS IN THE PROCEDURE |
Country Status (35)
Country | Link |
---|---|
JP (1) | JPS5687586A (en) |
KR (1) | KR830004322A (en) |
AR (2) | AR228859A1 (en) |
AT (1) | AT380883B (en) |
AU (1) | AU520995B2 (en) |
BE (1) | BE886319A (en) |
CA (1) | CA1143731A (en) |
CH (1) | CH649299A5 (en) |
CS (1) | CS241476B2 (en) |
DD (1) | DD154608A5 (en) |
DE (2) | DE3043979C2 (en) |
DK (1) | DK151811C (en) |
EG (1) | EG14929A (en) |
ES (1) | ES497066A0 (en) |
FI (1) | FI67706C (en) |
FR (1) | FR2470132A1 (en) |
GB (1) | GB2063862B (en) |
GR (1) | GR72132B (en) |
GT (1) | GT198066458A (en) |
HU (1) | HU179091B (en) |
IE (1) | IE50404B1 (en) |
IL (1) | IL61535A (en) |
IN (1) | IN154926B (en) |
IT (1) | IT1209373B (en) |
LU (1) | LU82950A1 (en) |
NL (1) | NL182565C (en) |
NO (1) | NO803521L (en) |
NZ (1) | NZ195596A (en) |
PH (1) | PH16666A (en) |
PL (1) | PL132354B1 (en) |
PT (1) | PT72090B (en) |
SE (1) | SE448732B (en) |
SU (1) | SU1042620A3 (en) |
YU (1) | YU41953B (en) |
ZA (1) | ZA807293B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8300728D0 (en) * | 1983-01-12 | 1983-02-16 | Erba Farmitalia | Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives |
US4457932A (en) * | 1983-07-22 | 1984-07-03 | Bristol-Myers Company | Anti-ulcer agents |
GB8422916D0 (en) * | 1984-09-11 | 1984-10-17 | May & Baker Ltd | Compositions of matter |
JP2690742B2 (en) * | 1987-03-30 | 1997-12-17 | 第一製薬株式会社 | Heterocyclic amine derivative |
ES2087072T3 (en) * | 1988-03-28 | 1996-07-16 | Janssen Pharmaceutica Nv | AGENTS TO PRESERVE OR RESTORE SKIN HEALTH. |
TWI500623B (en) * | 2009-10-13 | 2015-09-21 | Torrent Pharmaceuticals Ltd | Novel fused thiazolo and oxazolo pyrimidinones |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1331059A (en) * | 1971-04-19 | 1973-09-19 | Lilly Industries Ltd | Pyrimidotriazinone compounds |
US4041163A (en) * | 1976-03-29 | 1977-08-09 | Pfizer Inc. | N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents |
DE2810863A1 (en) * | 1978-03-13 | 1979-09-27 | Boehringer Mannheim Gmbh | 1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
US4223031A (en) * | 1978-05-05 | 1980-09-16 | Mead Johnson & Company | Azolopyrimidinones |
-
1980
- 1980-09-30 DK DK413180A patent/DK151811C/en not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/en active
- 1980-11-18 HU HU80802755A patent/HU179091B/en not_active IP Right Cessation
- 1980-11-18 CS CS807820A patent/CS241476B2/en unknown
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-18 AR AR283276A patent/AR228859A1/en active
- 1980-11-19 CH CH8567/80A patent/CH649299A5/en not_active IP Right Cessation
- 1980-11-19 EG EG723/80A patent/EG14929A/en active
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/en unknown
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-21 JP JP16450280A patent/JPS5687586A/en active Granted
- 1980-11-21 NO NO803521A patent/NO803521L/en unknown
- 1980-11-21 SE SE8008189A patent/SE448732B/en not_active IP Right Cessation
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 GT GT198066458A patent/GT198066458A/en unknown
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/en not_active IP Right Cessation
- 1980-11-21 FR FR8024822A patent/FR2470132A1/en active Granted
- 1980-11-21 IT IT8026176A patent/IT1209373B/en active
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/en not_active Expired
- 1980-11-21 PT PT72090A patent/PT72090B/en not_active IP Right Cessation
- 1980-11-21 AT AT0570780A patent/AT380883B/en not_active IP Right Cessation
- 1980-11-21 FI FI803628A patent/FI67706C/en not_active IP Right Cessation
- 1980-11-21 IL IL61535A patent/IL61535A/en unknown
- 1980-11-21 DE DE3050491A patent/DE3050491C2/en not_active Expired
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/en unknown
- 1980-11-21 ES ES497066A patent/ES497066A0/en active Granted
- 1980-11-21 LU LU82950A patent/LU82950A1/en unknown
- 1980-11-21 DD DD80225391A patent/DD154608A5/en not_active IP Right Cessation
- 1980-11-21 CA CA000365258A patent/CA1143731A/en not_active Expired
- 1980-11-22 PL PL1980228008A patent/PL132354B1/en unknown
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/en unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/en not_active IP Right Cessation
-
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/en active
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK29681A (en) | PROCEDURE FOR THE PREPARATION OF IMMUNOGAMMAGLOBULIN | |
NO803851L (en) | PROCEDURE FOR THE PREPARATION OF 4,1`, 6`-TRICLOR-4,1`, 6`-TRIDEOXY-GALACTOSUCROSE | |
NO802913L (en) | PROCEDURE FOR THE PREPARATION OF CEPHALOSPOR CONNECTION | |
DK311580A (en) | PROCEDURE FOR THE PREPARATION OF OXOALKYLXANTHINES | |
DK222980A (en) | PROCEDURE FOR THE PREPARATION OF SULPHONAMIDE DERIVATIVES | |
DK274580A (en) | PROCEDURE FOR THE PREPARATION OF TRIPEPTIDAMIDES | |
DK149623C (en) | PROCEDURE FOR THE PREPARATION OF ALFA-HYDROXYCARBOXYLIC ACIDAMIDS | |
DK4280A (en) | PROCEDURE FOR THE PREPARATION OF PLEUROMUTIL INGREDIENTS | |
DK289480A (en) | PROCEDURE FOR THE PREPARATION OF O-SUBSTITUTED KETOXIMS | |
DK153791C (en) | PROCEDURE FOR THE PREPARATION OF 7-HYDROXYCUMARANES | |
MX6160E (en) | PROCEDURE FOR THE PREPARATION OF N- (2-PHENYL 2-HYDROXYETHYL) -1,1-DIMETHYL-3- (4-PHENYL SUBSTITUTED) PROPYLAMINS | |
DK149856C (en) | PROCEDURE FOR THE PREPARATION OF 1,3-DI- OR 1,3,8-TRISUBSTITUTED XANTHINES OR PHYSIOLOGICALLY ACCEPTABLE SALTS THEREOF | |
DK341281A (en) | PROCEDURE FOR THE PREPARATION OF 3,3-DIALKYDENZODIAZEPINE DERIVATIVES OR ACID ADDITION SALTS AND THE PROCEDURE USED AS INTERMEDIATES | |
DK481280A (en) | PROCEDURE FOR THE PREPARATION OF PIPERIDYLBENZIMIDAZOLINE UNDERTIVES | |
DK117779A (en) | PROCEDURE FOR THE PREPARATION OF 2,6-DIALCOXYBENZAMIDES | |
DK215980A (en) | PROCEDURE FOR THE PREPARATION OF SULPHONAMIDE DERIVATIVES | |
DK262180A (en) | PROCEDURE FOR THE PREPARATION OF ALKYL-2-CHLORO PROPRIATORS | |
DK274680A (en) | PROCEDURE FOR THE PREPARATION OF TRIPEPTIDAMIDES | |
NO820281L (en) | PROCEDURE FOR THE PREPARATION OF N- (HALOGENMETHYL) -ACYLAMIDES | |
DK134580A (en) | PROCEDURE FOR THE PREPARATION OF 2,6-DIAMINONEBULARIN OR ACID ADDITION SALTS THEREOF | |
ES491238A0 (en) | A PROCEDURE FOR THE PREPARATION OF PIRIDO (1,2-A) PIRI-MIDINAS SUBSTITUTED | |
DK413180A (en) | PROCEDURE FOR THE PREPARATION OF N- (5-TETRAZOLYL) -1-OXO-1H-THIAZOLO (3,2-A) | |
NO150601C (en) | PROCEDURE FOR THE PREPARATION OF 2`-6`-DIALKYL-N-ALCOXYMETHYL-2-CHLORO-ACETANILIDES. | |
DK338480A (en) | PROCEDURE FOR THE PREPARATION OF PYRROLIDE INGREDIENTS | |
NO153100C (en) | PROCEDURE FOR THE PREPARATION OF N- (HALOGENMETHYL) -ACYLAMIDES. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PBP | Patent lapsed |