IL61535A - 5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof - Google Patents
5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereofInfo
- Publication number
- IL61535A IL61535A IL61535A IL6153580A IL61535A IL 61535 A IL61535 A IL 61535A IL 61535 A IL61535 A IL 61535A IL 6153580 A IL6153580 A IL 6153580A IL 61535 A IL61535 A IL 61535A
- Authority
- IL
- Israel
- Prior art keywords
- thiazolo
- tetrazolyl
- pyrimidine
- oxo
- carboxylic acids
- Prior art date
Links
- FDGPDTWORUVKQX-UHFFFAOYSA-N 5-oxo-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylic acid Chemical class O=C1C(C(=O)O)=CN=C2SC=CN21 FDGPDTWORUVKQX-UHFFFAOYSA-N 0.000 title 1
- 229940053202 antiepileptics carboxamide derivative Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9663179A | 1979-11-23 | 1979-11-23 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL61535A0 IL61535A0 (en) | 1980-12-31 |
| IL61535A true IL61535A (en) | 1984-06-29 |
Family
ID=22258306
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL61535A IL61535A (en) | 1979-11-23 | 1980-11-21 | 5-oxo-5h-thiazolo(3,2-a)pyrimidine-6-carboxylic acids and n-(5-tetrazolyl)-carboxamide derivatives thereof |
Country Status (35)
| Country | Link |
|---|---|
| JP (1) | JPS5687586A (en) |
| KR (1) | KR830004322A (en) |
| AR (2) | AR228859A1 (en) |
| AT (1) | AT380883B (en) |
| AU (1) | AU520995B2 (en) |
| BE (1) | BE886319A (en) |
| CA (1) | CA1143731A (en) |
| CH (1) | CH649299A5 (en) |
| CS (1) | CS241476B2 (en) |
| DD (1) | DD154608A5 (en) |
| DE (2) | DE3050491C2 (en) |
| DK (1) | DK151811C (en) |
| EG (1) | EG14929A (en) |
| ES (1) | ES497066A0 (en) |
| FI (1) | FI67706C (en) |
| FR (1) | FR2470132A1 (en) |
| GB (1) | GB2063862B (en) |
| GR (1) | GR72132B (en) |
| GT (1) | GT198066458A (en) |
| HU (1) | HU179091B (en) |
| IE (1) | IE50404B1 (en) |
| IL (1) | IL61535A (en) |
| IN (1) | IN154926B (en) |
| IT (1) | IT1209373B (en) |
| LU (1) | LU82950A1 (en) |
| NL (1) | NL182565C (en) |
| NO (1) | NO803521L (en) |
| NZ (1) | NZ195596A (en) |
| PH (1) | PH16666A (en) |
| PL (1) | PL132354B1 (en) |
| PT (1) | PT72090B (en) |
| SE (1) | SE448732B (en) |
| SU (1) | SU1042620A3 (en) |
| YU (1) | YU41953B (en) |
| ZA (1) | ZA807293B (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8300728D0 (en) * | 1983-01-12 | 1983-02-16 | Erba Farmitalia | Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives |
| US4457932A (en) * | 1983-07-22 | 1984-07-03 | Bristol-Myers Company | Anti-ulcer agents |
| GB8422916D0 (en) * | 1984-09-11 | 1984-10-17 | May & Baker Ltd | Compositions of matter |
| JP2690742B2 (en) * | 1987-03-30 | 1997-12-17 | 第一製薬株式会社 | Heterocyclic amine derivative |
| NZ228447A (en) * | 1988-03-28 | 1990-08-28 | Janssen Pharmaceutica Nv | Cosmetic or pharmaceutical composition possessing serotonin antogonistic activity |
| TWI500623B (en) * | 2009-10-13 | 2015-09-21 | Torrent Pharmaceuticals Ltd | Novel fused thiazole and oxazolidine |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1331059A (en) | 1971-04-19 | 1973-09-19 | Lilly Industries Ltd | Pyrimidotriazinone compounds |
| US4041163A (en) * | 1976-03-29 | 1977-08-09 | Pfizer Inc. | N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents |
| DE2810863A1 (en) * | 1978-03-13 | 1979-09-27 | Boehringer Mannheim Gmbh | 1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
| US4223031A (en) * | 1978-05-05 | 1980-09-16 | Mead Johnson & Company | Azolopyrimidinones |
-
1980
- 1980-09-30 DK DK413180A patent/DK151811C/en not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/en active
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-18 HU HU80802755A patent/HU179091B/en not_active IP Right Cessation
- 1980-11-18 AR AR283276A patent/AR228859A1/en active
- 1980-11-18 CS CS807820A patent/CS241476B2/en unknown
- 1980-11-19 EG EG723/80A patent/EG14929A/en active
- 1980-11-19 CH CH8567/80A patent/CH649299A5/en not_active IP Right Cessation
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/en unknown
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/en not_active IP Right Cessation
- 1980-11-21 NO NO803521A patent/NO803521L/en unknown
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/en unknown
- 1980-11-21 CA CA000365258A patent/CA1143731A/en not_active Expired
- 1980-11-21 PT PT72090A patent/PT72090B/en not_active IP Right Cessation
- 1980-11-21 DD DD80225391A patent/DD154608A5/en not_active IP Right Cessation
- 1980-11-21 IL IL61535A patent/IL61535A/en unknown
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3050491A patent/DE3050491C2/en not_active Expired
- 1980-11-21 SE SE8008189A patent/SE448732B/en not_active IP Right Cessation
- 1980-11-21 ES ES497066A patent/ES497066A0/en active Granted
- 1980-11-21 GT GT198066458A patent/GT198066458A/en unknown
- 1980-11-21 AT AT0570780A patent/AT380883B/en not_active IP Right Cessation
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 FR FR8024822A patent/FR2470132A1/en active Granted
- 1980-11-21 JP JP16450280A patent/JPS5687586A/en active Granted
- 1980-11-21 LU LU82950A patent/LU82950A1/en unknown
- 1980-11-21 FI FI803628A patent/FI67706C/en not_active IP Right Cessation
- 1980-11-21 IT IT8026176A patent/IT1209373B/en active
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/en not_active Expired
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/en not_active Ceased
- 1980-11-22 PL PL1980228008A patent/PL132354B1/en unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/en not_active IP Right Cessation
-
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/en active
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