HU179091B - Process for preparing antiallergenic and antiulcerogenic 1-oxo-1h-thiazolo/3,2-a/pyrimidine-2-carboxamide derivatives - Google Patents
Process for preparing antiallergenic and antiulcerogenic 1-oxo-1h-thiazolo/3,2-a/pyrimidine-2-carboxamide derivativesInfo
- Publication number
- HU179091B HU179091B HU80802755A HU275580A HU179091B HU 179091 B HU179091 B HU 179091B HU 80802755 A HU80802755 A HU 80802755A HU 275580 A HU275580 A HU 275580A HU 179091 B HU179091 B HU 179091B
- Authority
- HU
- Hungary
- Prior art keywords
- antiulcerogenic
- antiallergenic
- thiazolo
- pyrimidine
- oxo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US9663179A | 1979-11-23 | 1979-11-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
HU179091B true HU179091B (en) | 1982-08-28 |
Family
ID=22258306
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU80802755A HU179091B (en) | 1979-11-23 | 1980-11-18 | Process for preparing antiallergenic and antiulcerogenic 1-oxo-1h-thiazolo/3,2-a/pyrimidine-2-carboxamide derivatives |
Country Status (35)
Country | Link |
---|---|
JP (1) | JPS5687586A (en) |
KR (1) | KR830004322A (en) |
AR (2) | AR228859A1 (en) |
AT (1) | AT380883B (en) |
AU (1) | AU520995B2 (en) |
BE (1) | BE886319A (en) |
CA (1) | CA1143731A (en) |
CH (1) | CH649299A5 (en) |
CS (1) | CS241476B2 (en) |
DD (1) | DD154608A5 (en) |
DE (2) | DE3043979C2 (en) |
DK (1) | DK151811C (en) |
EG (1) | EG14929A (en) |
ES (1) | ES8203363A1 (en) |
FI (1) | FI67706C (en) |
FR (1) | FR2470132A1 (en) |
GB (1) | GB2063862B (en) |
GR (1) | GR72132B (en) |
GT (1) | GT198066458A (en) |
HU (1) | HU179091B (en) |
IE (1) | IE50404B1 (en) |
IL (1) | IL61535A (en) |
IN (1) | IN154926B (en) |
IT (1) | IT1209373B (en) |
LU (1) | LU82950A1 (en) |
NL (1) | NL182565C (en) |
NO (1) | NO803521L (en) |
NZ (1) | NZ195596A (en) |
PH (1) | PH16666A (en) |
PL (1) | PL132354B1 (en) |
PT (1) | PT72090B (en) |
SE (1) | SE448732B (en) |
SU (1) | SU1042620A3 (en) |
YU (1) | YU41953B (en) |
ZA (1) | ZA807293B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8300728D0 (en) * | 1983-01-12 | 1983-02-16 | Erba Farmitalia | Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives |
US4457932A (en) * | 1983-07-22 | 1984-07-03 | Bristol-Myers Company | Anti-ulcer agents |
GB8422916D0 (en) * | 1984-09-11 | 1984-10-17 | May & Baker Ltd | Compositions of matter |
JP2690742B2 (en) * | 1987-03-30 | 1997-12-17 | 第一製薬株式会社 | Heterocyclic amine derivative |
NZ228447A (en) * | 1988-03-28 | 1990-08-28 | Janssen Pharmaceutica Nv | Cosmetic or pharmaceutical composition possessing serotonin antogonistic activity |
TWI500623B (en) * | 2009-10-13 | 2015-09-21 | Torrent Pharmaceuticals Ltd | Novel fused thiazolo and oxazolo pyrimidinones |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1331059A (en) * | 1971-04-19 | 1973-09-19 | Lilly Industries Ltd | Pyrimidotriazinone compounds |
US4041163A (en) * | 1976-03-29 | 1977-08-09 | Pfizer Inc. | N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents |
DE2810863A1 (en) * | 1978-03-13 | 1979-09-27 | Boehringer Mannheim Gmbh | 1-OXO-1H-PYRIMIDO ANGLE CLAMP ON 6.1-B ANGLE CLAMP ON BENZTHIAZOLE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
US4223031A (en) * | 1978-05-05 | 1980-09-16 | Mead Johnson & Company | Azolopyrimidinones |
-
1980
- 1980-09-30 DK DK413180A patent/DK151811C/en not_active IP Right Cessation
- 1980-10-15 IN IN760/DEL/80A patent/IN154926B/en unknown
- 1980-11-17 SU SU803212053A patent/SU1042620A3/en active
- 1980-11-18 CS CS807820A patent/CS241476B2/en unknown
- 1980-11-18 HU HU80802755A patent/HU179091B/en not_active IP Right Cessation
- 1980-11-18 AR AR283276A patent/AR228859A1/en active
- 1980-11-18 GB GB8036904A patent/GB2063862B/en not_active Expired
- 1980-11-19 EG EG723/80A patent/EG14929A/en active
- 1980-11-19 CH CH8567/80A patent/CH649299A5/en not_active IP Right Cessation
- 1980-11-20 NZ NZ195596A patent/NZ195596A/en unknown
- 1980-11-20 YU YU2950/80A patent/YU41953B/en unknown
- 1980-11-20 GR GR63413A patent/GR72132B/el unknown
- 1980-11-21 NO NO803521A patent/NO803521L/en unknown
- 1980-11-21 DD DD80225391A patent/DD154608A5/en not_active IP Right Cessation
- 1980-11-21 AT AT0570780A patent/AT380883B/en not_active IP Right Cessation
- 1980-11-21 IE IE2418/80A patent/IE50404B1/en unknown
- 1980-11-21 DE DE3043979A patent/DE3043979C2/en not_active Expired
- 1980-11-21 GT GT198066458A patent/GT198066458A/en unknown
- 1980-11-21 IL IL61535A patent/IL61535A/en unknown
- 1980-11-21 AU AU64595/80A patent/AU520995B2/en not_active Ceased
- 1980-11-21 IT IT8026176A patent/IT1209373B/en active
- 1980-11-21 ES ES497066A patent/ES8203363A1/en not_active Expired
- 1980-11-21 DE DE3050491A patent/DE3050491C2/en not_active Expired
- 1980-11-21 LU LU82950A patent/LU82950A1/en unknown
- 1980-11-21 PT PT72090A patent/PT72090B/en not_active IP Right Cessation
- 1980-11-21 PH PH24891A patent/PH16666A/en unknown
- 1980-11-21 SE SE8008189A patent/SE448732B/en not_active IP Right Cessation
- 1980-11-21 JP JP16450280A patent/JPS5687586A/en active Granted
- 1980-11-21 CA CA000365258A patent/CA1143731A/en not_active Expired
- 1980-11-21 ZA ZA00807293A patent/ZA807293B/en unknown
- 1980-11-21 FI FI803628A patent/FI67706C/en not_active IP Right Cessation
- 1980-11-21 NL NLAANVRAGE8006362,A patent/NL182565C/en not_active IP Right Cessation
- 1980-11-21 FR FR8024822A patent/FR2470132A1/en active Granted
- 1980-11-22 PL PL1980228008A patent/PL132354B1/en unknown
- 1980-11-22 KR KR1019800004474A patent/KR830004322A/en unknown
- 1980-11-24 BE BE0/202915A patent/BE886319A/en not_active IP Right Cessation
-
1982
- 1982-09-13 AR AR290628A patent/AR231296A1/en active
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
HU90 | Patent valid on 900628 | ||
HMM4 | Cancellation of final prot. due to non-payment of fee |