DK23677A - PROCEDURE FOR THE PREPARATION OF OXIMI DERIVATIVES OF 7-AMINOTHIAZOLYL-ACETAMIDOCEPHALOSPORANIC ACID - Google Patents
PROCEDURE FOR THE PREPARATION OF OXIMI DERIVATIVES OF 7-AMINOTHIAZOLYL-ACETAMIDOCEPHALOSPORANIC ACIDInfo
- Publication number
- DK23677A DK23677A DK23677A DK23677A DK23677A DK 23677 A DK23677 A DK 23677A DK 23677 A DK23677 A DK 23677A DK 23677 A DK23677 A DK 23677A DK 23677 A DK23677 A DK 23677A
- Authority
- DK
- Denmark
- Prior art keywords
- oximi
- aminothiazolyl
- derivatives
- procedure
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DK242483A DK160872C (en) | 1976-01-23 | 1983-05-30 | 2-AMINO-4-THIAZOLYL-OXYIMINO ACETIC ACID DERIVATIVES USED AS INTERMEDIATES FOR THE PREPARATION OF SIMILAR CEPHALOSPORINE DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF |
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7601834A FR2346014A1 (en) | 1976-01-23 | 1976-01-23 | Amino-thiazolyl-hydroxyimino-acetamido-cephalosporanic acids - with antibacterial activity |
FR7617743A FR2361893A2 (en) | 1976-01-23 | 1976-06-11 | Amino-thiazolyl-hydroxyimino-acetamido-cephalosporanic acids - with antibacterial activity |
FR7601834 | 1976-07-11 | ||
FR7625051 | 1976-08-18 | ||
FR7625051A FR2361894A2 (en) | 1976-01-23 | 1976-08-18 | Amino-thiazolyl-hydroxyimino-acetamido-cephalosporanic acids - with antibacterial activity |
FR7617743 | 1979-08-18 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK23677A true DK23677A (en) | 1977-07-24 |
DK161082B DK161082B (en) | 1991-05-27 |
DK161082C DK161082C (en) | 1991-11-04 |
Family
ID=27250574
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK023677A DK161082C (en) | 1976-01-23 | 1977-01-21 | ANALOGY PROCEDURE FOR PREPARING SYN-ISOMER OXIMER DERIVATIVES OF 7-AMINOTHIAZOLYLACETAMIDOCEPHALOSPORANIC ACID |
Country Status (31)
Country | Link |
---|---|
JP (3) | JPS52102293A (en) |
AR (1) | AR231985A1 (en) |
AT (2) | AT355205B (en) |
AU (1) | AU511680B2 (en) |
BE (1) | BE850662A (en) |
CA (1) | CA1319682C (en) |
CH (1) | CH622264A5 (en) |
CY (1) | CY1123A (en) |
DD (2) | DD132869A5 (en) |
DE (3) | DE2702501C2 (en) |
DK (1) | DK161082C (en) |
ES (2) | ES455089A1 (en) |
GB (2) | GB1580621A (en) |
GE (1) | GEP19970783B (en) |
GR (1) | GR70302B (en) |
HK (1) | HK50381A (en) |
HU (1) | HU173110B (en) |
IE (1) | IE45015B1 (en) |
IL (2) | IL51192A (en) |
IT (1) | IT1104601B (en) |
KE (1) | KE3365A (en) |
LU (1) | LU76624A1 (en) |
MX (1) | MX4407E (en) |
MY (1) | MY8500417A (en) |
NL (1) | NL7700706A (en) |
NZ (1) | NZ183150A (en) |
PL (1) | PL122698B1 (en) |
PT (1) | PT66099B (en) |
SE (2) | SE440655B (en) |
SU (1) | SU822754A3 (en) |
YU (3) | YU41060B (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK152213B (en) * | 1977-08-17 | 1988-02-08 | Roussel Uclaf | METHOD FOR PREPARING A CRYSTALLINE FORM OF THE SODIUM SALT OF AN OXIME DERIVATIVE OF 7-AMINOTHIAZOLYLACETAMIDOCEPHALOSPORANIC ACID |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2408613A2 (en) * | 1977-07-19 | 1979-06-08 | Roussel Uclaf | NEW OXIMES DERIVED FROM 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC ACID, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS |
GB1576625A (en) * | 1976-04-12 | 1980-10-08 | Fujisawa Pharmaceutical Co | Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof |
DK162391C (en) * | 1976-04-12 | 1992-03-09 | Fujisawa Pharmaceutical Co | ANALOGY PROCEDURE FOR PREPARING SYN-ISOMERS OF 3,7-DISUBSTITUTED 3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS |
DE2760484C2 (en) * | 1976-04-14 | 1992-12-03 | Takeda Chemical Industries, Ltd., Osaka, Jp | |
ZA781502B (en) * | 1977-03-14 | 1979-09-26 | Fujisawa Pharmaceutical Co | New cephem and cepham compounds and processes for preparation thereof |
PH17188A (en) | 1977-03-14 | 1984-06-14 | Fujisawa Pharmaceutical Co | New cephem and cepham compounds and their pharmaceutical compositions and method of use |
DE2714880A1 (en) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION |
JPS5444695A (en) * | 1977-09-13 | 1979-04-09 | Fujisawa Pharmaceut Co Ltd | 3,7-disubstituted-3-cephem-4-carboxylic acid and its salt and their preparation |
FR2410655A1 (en) * | 1977-12-05 | 1979-06-29 | Roussel Uclaf | NEW OXIMES DERIVED FROM 3-SUBSTITUTE 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR METHOD OF PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS |
JPS5498795A (en) * | 1978-01-13 | 1979-08-03 | Takeda Chem Ind Ltd | Cephalosporin derivative and its preparation |
FR2387235A1 (en) * | 1978-01-23 | 1978-11-10 | Fujisawa Pharmaceutical Co | PROCESS FOR THE PREPARATION OF COMPOUNDS OF 3,7-DISUBSTITUE-3-CEPHEM-4-CARBOXYLIC ACID AND NEW PRODUCTS THUS OBTAINED, HAVING A STRONG ANTIBACTERIAL ACTIVITY |
FR2432521A1 (en) * | 1978-03-31 | 1980-02-29 | Roussel Uclaf | NOVEL O-SUBSTITUTED OXIMES DERIVED FROM 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC ACID, THEIR PREPARATION PROCESS AND THEIR USE AS MEDICAMENTS |
SE445350B (en) * | 1978-04-14 | 1986-06-16 | Roussel Uclaf | OXIMO DERIVATIVES OF 3-AZIDOMETHYL-7-AMINO-THIAZOLYL-ACETAMIDO-CEPHALOSPORANIC ACID AND ITS USE AS ANTIBIOTICS |
US4284631A (en) * | 1978-07-31 | 1981-08-18 | Fujisawa Pharmaceutical Co., Ltd. | 7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them |
FR2448543A1 (en) * | 1979-02-09 | 1980-09-05 | Roussel Uclaf | NOVEL OXIMES O-SUBSTITUTED BY A RADICAL COMPRISING A QUATERNARY AMMONIUM AND DERIVATIVES OF 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS |
FR2461713A1 (en) * | 1979-07-19 | 1981-02-06 | Roussel Uclaf | SUBSTITUTED ALKYLOXIMIC NEWS DERIVED FROM 7- (2-AMINO 4-THIAZOLYL) ACETAMIDO CEPHALOSPORANIC ACID, PROCESS FOR PREPARING THEM AND THEIR APPLICATION AS MEDICAMENTS |
FR2461712A1 (en) * | 1979-07-23 | 1981-02-06 | Hoechst Ag | 2-Oximino-acylamino cephem cpds. prodn. - by acylating 7-amino-cephem cpds. with complexes of 2-syn-oximino-acyl halide(s) and N,N-di:substd. amide(s) |
JPS57154175A (en) * | 1981-03-16 | 1982-09-22 | Mitsui Toatsu Chem Inc | 2-thiazoleamine derivative, its preparation, and drug composition comprising it |
FR2506307A1 (en) * | 1981-05-22 | 1982-11-26 | Roussel Uclaf | 7-thiazolyl-acetamido-cephalosporin oxime derivs. - useful as broad spectrum antibacterials and disinfectants (BE 1.10.79) |
JPS57163386A (en) * | 1981-08-13 | 1982-10-07 | Takeda Chem Ind Ltd | Cephalosporin derivative and its production |
CA1296012C (en) | 1986-03-19 | 1992-02-18 | Susumu Nakagawa | 6,7-dihydroxy-isoquinoline derivatives |
HUT53892A (en) * | 1989-04-07 | 1990-12-28 | Technologishen Kom Za Promy Mi | Process for producing synaminothiazolyl and synaminooxazolyl derivatives |
CN112457271A (en) * | 2020-11-18 | 2021-03-09 | 河北合佳医药科技集团股份有限公司 | Continuous flow synthesis method of aminothiazoly loximate intermediate |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1399086A (en) * | 1971-05-14 | 1975-06-25 | Glaxo Lab Ltd | Cephalosporin compounds |
DK154939C (en) | 1974-12-19 | 1989-06-12 | Takeda Chemical Industries Ltd | METHOD OF ANALOGUE FOR THE PREPARATION OF THIAZOLYLACETAMIDO-CEPHEM COMPOUNDS OR PHARMACEUTICAL ACCEPTABLE SALTS OR ESTERS THEREOF |
GB1536281A (en) * | 1975-06-09 | 1978-12-20 | Takeda Chemical Industries Ltd | Cephem compounds |
DE2760123C2 (en) | 1976-01-23 | 1986-04-30 | Roussel-Uclaf, Paris | 7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporanic acids, their preparation and pharmaceutical compositions containing them |
JPS6011713B2 (en) | 1976-09-08 | 1985-03-27 | 武田薬品工業株式会社 | Cephalosporin derivatives and their production method |
-
1976
- 1976-12-29 SE SE7614678A patent/SE440655B/en not_active IP Right Cessation
- 1976-12-31 IL IL51192A patent/IL51192A/en unknown
-
1977
- 1977-01-15 ES ES455089A patent/ES455089A1/en not_active Expired
- 1977-01-18 SU SU772439818A patent/SU822754A3/en active
- 1977-01-19 AR AR266241A patent/AR231985A1/en active
- 1977-01-19 YU YU137/77A patent/YU41060B/en unknown
- 1977-01-20 IT IT47727/77A patent/IT1104601B/en active Protection Beyond IP Right Term
- 1977-01-20 MX MX775372U patent/MX4407E/en unknown
- 1977-01-21 DD DD7700200629A patent/DD132869A5/en unknown
- 1977-01-21 DE DE2702501A patent/DE2702501C2/en not_active Expired
- 1977-01-21 HU HU77RO909A patent/HU173110B/en unknown
- 1977-01-21 NZ NZ183150A patent/NZ183150A/en unknown
- 1977-01-21 DE DE2760287A patent/DE2760287C2/de not_active Expired
- 1977-01-21 CA CA000270375A patent/CA1319682C/en not_active Expired - Lifetime
- 1977-01-21 CY CY1123A patent/CY1123A/en unknown
- 1977-01-21 DK DK023677A patent/DK161082C/en active
- 1977-01-21 DE DE2759895A patent/DE2759895C2/en not_active Expired
- 1977-01-21 JP JP504977A patent/JPS52102293A/en active Granted
- 1977-01-21 BE BE174311A patent/BE850662A/en not_active IP Right Cessation
- 1977-01-21 GB GB2640/77A patent/GB1580621A/en not_active Expired
- 1977-01-21 CH CH78777A patent/CH622264A5/en not_active IP Right Cessation
- 1977-01-21 DD DD7700197036A patent/DD128594A5/en unknown
- 1977-01-21 GB GB15561/79A patent/GB1580623A/en not_active Expired
- 1977-01-21 LU LU76624A patent/LU76624A1/xx unknown
- 1977-01-21 PT PT66099A patent/PT66099B/en unknown
- 1977-01-22 PL PL1977195504A patent/PL122698B1/en unknown
- 1977-01-22 GR GR52630A patent/GR70302B/el unknown
- 1977-01-24 NL NL7700706A patent/NL7700706A/en not_active Application Discontinuation
- 1977-01-24 AT AT41277A patent/AT355205B/en not_active IP Right Cessation
- 1977-01-24 AU AU21579/77A patent/AU511680B2/en not_active Expired
- 1977-01-24 IE IE148/77A patent/IE45015B1/en not_active IP Right Cessation
-
1978
- 1978-02-01 ES ES466539A patent/ES466539A1/en not_active Expired
-
1979
- 1979-03-20 AT AT0209479A patent/AT373592B/en not_active IP Right Cessation
- 1979-05-31 IL IL57445A patent/IL57445A0/en not_active IP Right Cessation
-
1981
- 1981-10-22 HK HK503/81A patent/HK50381A/en unknown
-
1982
- 1982-08-26 SE SE8204893A patent/SE455307B/en not_active IP Right Cessation
-
1983
- 1983-01-04 YU YU11/83A patent/YU43143B/en unknown
- 1983-01-04 YU YU00012/83A patent/YU1283A/en unknown
-
1984
- 1984-01-11 KE KE3365A patent/KE3365A/en unknown
-
1985
- 1985-12-30 MY MY417/85A patent/MY8500417A/en unknown
-
1990
- 1990-04-19 JP JP2101872A patent/JPH03204868A/en active Pending
-
1993
- 1993-01-20 JP JP5023427A patent/JPH05247013A/en active Pending
- 1993-09-09 GE GEAP19931537A patent/GEP19970783B/en unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK152213B (en) * | 1977-08-17 | 1988-02-08 | Roussel Uclaf | METHOD FOR PREPARING A CRYSTALLINE FORM OF THE SODIUM SALT OF AN OXIME DERIVATIVE OF 7-AMINOTHIAZOLYLACETAMIDOCEPHALOSPORANIC ACID |
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