DK1848406T3 - Fast, penoral lægemiddelform til kontraception, der indeholder dienogest og ethynylestradiol - Google Patents

Fast, penoral lægemiddelform til kontraception, der indeholder dienogest og ethynylestradiol

Info

Publication number
DK1848406T3
DK1848406T3 DK06706961T DK06706961T DK1848406T3 DK 1848406 T3 DK1848406 T3 DK 1848406T3 DK 06706961 T DK06706961 T DK 06706961T DK 06706961 T DK06706961 T DK 06706961T DK 1848406 T3 DK1848406 T3 DK 1848406T3
Authority
DK
Denmark
Prior art keywords
dienogest
solid
penal
formulation
ethinyl estradiol
Prior art date
Application number
DK06706961T
Other languages
English (en)
Inventor
Sabine Fricke
Hagen Gerecke
Ralf Ladwig
Alexander Buske
Harald Raethe
Original Assignee
Jenapharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP05003181A external-priority patent/EP1690529A1/de
Priority claimed from EP05003179A external-priority patent/EP1690543A1/de
Application filed by Jenapharm Gmbh filed Critical Jenapharm Gmbh
Application granted granted Critical
Publication of DK1848406T3 publication Critical patent/DK1848406T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Organic Chemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK06706961T 2005-02-15 2006-02-15 Fast, penoral lægemiddelform til kontraception, der indeholder dienogest og ethynylestradiol DK1848406T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05003181A EP1690529A1 (de) 2005-02-15 2005-02-15 Feste perorale Arzneiform zur Kontrazeption, die Dienogest und Ethinylestradiol enthält
EP05003179A EP1690543A1 (de) 2005-02-15 2005-02-15 Pharmazeutisches Präparat zur Kontrazeption
PCT/EP2006/001358 WO2006087177A2 (de) 2005-02-15 2006-02-15 Feste perorale arzneiform zur kontrazeption, die dienogest und ethinylestradiol enthält

Publications (1)

Publication Number Publication Date
DK1848406T3 true DK1848406T3 (da) 2008-09-15

Family

ID=37951746

Family Applications (1)

Application Number Title Priority Date Filing Date
DK06706961T DK1848406T3 (da) 2005-02-15 2006-02-15 Fast, penoral lægemiddelform til kontraception, der indeholder dienogest og ethynylestradiol

Country Status (20)

Country Link
EP (1) EP1848406B1 (da)
JP (1) JP2008527019A (da)
KR (1) KR20070087141A (da)
AT (1) ATE395047T1 (da)
AU (1) AU2006215822B2 (da)
BR (1) BRPI0606297A2 (da)
CA (1) CA2594939A1 (da)
CY (1) CY1108265T1 (da)
DE (1) DE502006000771D1 (da)
DK (1) DK1848406T3 (da)
EA (1) EA200701389A1 (da)
ES (1) ES2310907T3 (da)
HR (1) HRP20080394T3 (da)
IL (1) IL184257A0 (da)
NO (1) NO20072893L (da)
PL (1) PL1848406T3 (da)
PT (1) PT1848406E (da)
RS (1) RS50597B (da)
SI (1) SI1848406T1 (da)
WO (1) WO2006087177A2 (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010529063A (ja) * 2007-07-31 2010-08-26 バイエル・シエーリング・ファーマ アクチエンゲゼルシャフト 血圧の調節のための経口治療のための、単相医薬複合調製物（ジエノゲスト（ｄｉｅｎｏｇｅｓｔ）およびエチニルエストラジオール）
EP2170347A1 (de) * 2007-07-31 2010-04-07 Bayer Schering Pharma Aktiengesellschaft Einphasisches pharmazeutisches kombinationspräparat (dienogest und ethinylestradiol) zur oralen therapie der regulierung des blutdruckes
JP6759478B2 (ja) * 2019-02-13 2020-09-23 富士製薬工業株式会社 経口固形組成物、その製造方法、及びその製造方法によって得られた経口用錠剤
EP3954364A1 (en) 2020-08-14 2022-02-16 Chemo Research, S.L. New modified release oral contraceptive composition

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19525017A1 (de) * 1995-06-28 1997-01-02 Schering Ag Pharmazeutisches Kombinatonspräparat, Kit und Methode zur hormonalen Kontrazeption
JP2000515890A (ja) * 1996-07-26 2000-11-28 アメリカン・ホーム・プロダクツ・コーポレイション プロゲスチンとエストロゲンとの混合剤からなる一相性避妊法およびキット

Also Published As

Publication number Publication date
CY1108265T1 (el) 2014-02-12
HRP20080394T3 (en) 2008-11-30
AU2006215822B2 (en) 2008-09-04
ES2310907T3 (es) 2009-01-16
WO2006087177A2 (de) 2006-08-24
RS50597B (sr) 2010-05-07
EP1848406A2 (de) 2007-10-31
ATE395047T1 (de) 2008-05-15
BRPI0606297A2 (pt) 2009-06-09
KR20070087141A (ko) 2007-08-27
IL184257A0 (en) 2007-10-31
WO2006087177B1 (de) 2007-10-11
CA2594939A1 (en) 2006-08-24
EP1848406B1 (de) 2008-05-14
DE502006000771D1 (de) 2008-06-26
PL1848406T3 (pl) 2009-06-30
NO20072893L (no) 2007-09-12
WO2006087177A8 (de) 2007-05-24
WO2006087177A3 (de) 2007-08-30
EA200701389A1 (ru) 2008-02-28
JP2008527019A (ja) 2008-07-24
PT1848406E (pt) 2008-08-21
SI1848406T1 (sl) 2008-10-31
AU2006215822A1 (en) 2006-08-24

Similar Documents

Publication Publication Date Title
HRP20070188B1 (hr) Farmaceutska kombinacija etinilestradiola i drospirenona za upotrebu kao kontracepcijskog sredstva
HRP20090418T1 (en) Pharmaceutical composition containing gestagens and/or estrogens and 5-methyl-(6s)-tetrahydrofolate
EA200900491A1 (ru) Применение эстрадиола валерата или 17в-эстрадиола в комбинации с диеногестом для перорального лечения для поддержания и/или повышения полового влечения у особи женского пола
CA2420292A1 (en) Contraception process and administration form for the same
NO327588B1 (no) Farmasoytisk sammensetning og preparat omfattende etinylostradiol og drospirenon for anvendelse som antikonsepsjonsmiddel
HRP20100513T1 (en) Multi-phase contraceptive preparation based on a natural estrogen
DK1848406T3 (da) Fast, penoral lægemiddelform til kontraception, der indeholder dienogest og ethynylestradiol
WO2005092441A3 (en) Extended cycle multiphasic oral contraceptive method
TW200638951A (en) Solid oral pharmaceutical form for contraception
UA85003C2 (ru) Твердая лекарственная форма для контрацепции
HRP20090256T1 (en) Use of estradiolvalerate and dienogest for oral treatment of dysfunctional uterine bleeding in a contraceptive method
NO20091057L (no) Oral legemiddelform for prevensjon
DK1937274T3 (da) Anvendelse af estradiolvalerat i kombination med dienogest til oral behandling af dysfunktionel uterin blødning i enhed med en oral kontraception
TH80558A (th) รูปแบบยาทางช่องปากชนิดแข็งสำหรับการคุมกำเนิด
TH80558B (th) รูปแบบยาทางช่องปากชนิดแข็งสำหรับการคุมกำเนิด
PE20091020A1 (es) Uso de un gestageno en combinacion con un estrogeno y uno o varios excipientes/portadores farmaceuticamente aceptables para la anticoncepcion oral sin lactosa
UY29378A1 (es) Preparación farmaceutica para la anticoncepción oral
ECSP003721A (es) Una composicion farmaceutica para ser usada como anticonceptivo
JO2213B1 (en) A pharmaceutical composition for use as a contraceptive method