ECSP003721A - Una composicion farmaceutica para ser usada como anticonceptivo - Google Patents

Una composicion farmaceutica para ser usada como anticonceptivo

Info

Publication number
ECSP003721A
ECSP003721A EC2000003721A ECSP003721A ECSP003721A EC SP003721 A ECSP003721 A EC SP003721A EC 2000003721 A EC2000003721 A EC 2000003721A EC SP003721 A ECSP003721 A EC SP003721A EC SP003721 A ECSP003721 A EC SP003721A
Authority
EC
Ecuador
Prior art keywords
composition
daily
active agent
dosage units
pharmaceutical composition
Prior art date
Application number
EC2000003721A
Other languages
English (en)
Inventor
Ralph Lipp
Wolfgang Heil
Jurgen Hilman
Renate Heithecker
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8240592&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP003721(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Ag filed Critical Schering Ag
Publication of ECSP003721A publication Critical patent/ECSP003721A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La invención se relaciona con una composición farmacéutica que comprende con un primer agente activo, 6B, 7B; 15B, 16B dimetilen-3-oxo-17a pregn-4-en-21, 17-carbolactona (drospirenona) en una cantidad correspondiente a una dosis diaria, a ser administrada con la composición, de desde aproximadamente 2mg a aproximadamente 4mg, y, como un segundo agente activo, 17 a-etinilestradiol (etinilestradiol) en una cantidad correspondiente a una dosis diaria desde aproximadamente 0.01mg a aproximadamente 0,05mg conjuntamente con uno o mas soportes o excipientes farmacéuticamente aceptables. En una realización específica, la composición consiste de un número de unidades de dosificación diarias colocadas en una unidad de empauqe, empaquetadas separadamente y separables individualmente, y proporcionadas para la administarción oral durante un periodo de al menos 21 días consecutivos, comprendiendo dichas unidades de dosificación diaria la combinación de drospirenona y etilestradiol. La composición puede comprender admés 7 o menos unidades de dosificación diaria que no contienen agente activo o que contienen solo etinilestradiol.
EC2000003721A 1999-08-31 2000-10-18 Una composicion farmaceutica para ser usada como anticonceptivo ECSP003721A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99202826 1999-08-31

Publications (1)

Publication Number Publication Date
ECSP003721A true ECSP003721A (es) 2002-05-23

Family

ID=8240592

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2000003721A ECSP003721A (es) 1999-08-31 2000-10-18 Una composicion farmaceutica para ser usada como anticonceptivo

Country Status (6)

Country Link
CN (1) CN1879632A (es)
AR (2) AR025443A1 (es)
CO (1) CO5200771A1 (es)
EC (1) ECSP003721A (es)
PE (1) PE20010665A1 (es)
ZA (2) ZA200201668B (es)

Also Published As

Publication number Publication date
AR043470A2 (es) 2005-07-27
ZA200404083B (en) 2006-02-22
AR025443A1 (es) 2002-11-27
CO5200771A1 (es) 2002-09-27
PE20010665A1 (es) 2001-06-19
ZA200201668B (en) 2004-06-24
CN1879632A (zh) 2006-12-20

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