DK182585A - Fosfomycinderivat og fremgangsmaade til fremstilling deraf - Google Patents
Fosfomycinderivat og fremgangsmaade til fremstilling deraf Download PDFInfo
- Publication number
- DK182585A DK182585A DK182585A DK182585A DK182585A DK 182585 A DK182585 A DK 182585A DK 182585 A DK182585 A DK 182585A DK 182585 A DK182585 A DK 182585A DK 182585 A DK182585 A DK 182585A
- Authority
- DK
- Denmark
- Prior art keywords
- phosphomycine
- procedures
- derivatives
- preparing
- compounds
- Prior art date
Links
- 238000000034 method Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 description 3
- 241000894006 Bacteria Species 0.000 description 1
- YMDXZJFXQJVXBF-STHAYSLISA-N fosfomycin Chemical class C[C@@H]1O[C@@H]1P(O)(O)=O YMDXZJFXQJVXBF-STHAYSLISA-N 0.000 description 1
- 150000002460 imidazoles Chemical class 0.000 description 1
- 208000015181 infectious disease Diseases 0.000 description 1
- 238000007911 parenteral administration Methods 0.000 description 1
- 239000008194 pharmaceutical composition Substances 0.000 description 1
- 238000001556 precipitation Methods 0.000 description 1
- 150000003839 salts Chemical class 0.000 description 1
- 239000002904 solvent Substances 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/655—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
- C07F9/65502—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a three-membered ring
- C07F9/65505—Phosphonic acids containing oxirane groups; esters thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Saccharide Compounds (AREA)
Description
den med det tilsvarende imidazolderivat efterfulgt af udfældning med et opløsningsmiddel. De fremstillede forbindelser anvendes i farmaceutiske præparater til oral og parenteral administrering. Forbindelserne er aktive overfor gram-positive og gram-negative bakterier og derfor nyttige til behandling af infektioner forårsaget af disse organismer. De fremstillede forbindelser har større biotilgængelighed end hidtil kendte salte af fosfomycin, og de kan indgives intramuskulært med mindre ubehag for patienten.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB08410502A GB2158828B (en) | 1984-04-25 | 1984-04-25 | Salts of fosfomycin |
| GB8410502 | 1984-04-25 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK182585D0 DK182585D0 (da) | 1985-04-24 |
| DK182585A true DK182585A (da) | 1985-10-26 |
Family
ID=10560028
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK182585A DK182585A (da) | 1984-04-25 | 1985-04-24 | Fosfomycinderivat og fremgangsmaade til fremstilling deraf |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4675315A (da) |
| EP (1) | EP0161843A1 (da) |
| JP (1) | JPS615088A (da) |
| AU (1) | AU4166985A (da) |
| DK (1) | DK182585A (da) |
| ES (1) | ES8603903A1 (da) |
| FI (1) | FI851618L (da) |
| GB (1) | GB2158828B (da) |
| NO (1) | NO851603L (da) |
| PT (1) | PT80343B (da) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1124610B (it) * | 1979-10-18 | 1986-05-07 | Zambo Spa | Mono(2-ammonio-2-idrossimetil-1,3-propandiolo) (2r-cis)-(o-metilossiranil)fosfonato |
| ES2239536B1 (es) * | 2004-03-05 | 2007-02-01 | Labiana Development, S.L. | Procedimiento de obtencion de la sal de metiloxiranilfosfonato de trometamina con una relacion molar de 1:1. |
| CN105963244A (zh) | 2016-01-15 | 2016-09-28 | 赵鸣 | 注射用青蒿琥酯制剂及其应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2801243A (en) * | 1956-06-05 | 1957-07-30 | American Home Prod | Imidazole salts of penicillin |
| US2750379A (en) * | 1952-10-06 | 1956-06-12 | American Home Prod | Imidazolidine salts of penicillin |
| US3914231A (en) * | 1970-09-04 | 1975-10-21 | Merck & Co Inc | ({31 )(Cis-1,2-epoxypropyl)-phosphonic acid and salts thereof |
| IT1161974B (it) * | 1978-02-02 | 1987-03-18 | Italchemi Spa | Derivti dell acido cis.i 2 epossipropilfosfonico loro procedimento di preparazione e composizioni farmaceutiche che li contengono |
-
1984
- 1984-04-25 GB GB08410502A patent/GB2158828B/en not_active Expired
-
1985
- 1985-04-17 US US06/724,093 patent/US4675315A/en not_active Expired - Fee Related
- 1985-04-22 NO NO851603A patent/NO851603L/no unknown
- 1985-04-24 AU AU41669/85A patent/AU4166985A/en not_active Abandoned
- 1985-04-24 ES ES542522A patent/ES8603903A1/es not_active Expired
- 1985-04-24 DK DK182585A patent/DK182585A/da not_active Application Discontinuation
- 1985-04-24 FI FI851618A patent/FI851618L/fi not_active Application Discontinuation
- 1985-04-24 PT PT80343A patent/PT80343B/pt unknown
- 1985-04-24 EP EP85302877A patent/EP0161843A1/en not_active Ceased
- 1985-04-25 JP JP60089884A patent/JPS615088A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| FI851618A0 (fi) | 1985-04-24 |
| GB2158828A (en) | 1985-11-20 |
| US4675315A (en) | 1987-06-23 |
| ES542522A0 (es) | 1986-01-01 |
| ES8603903A1 (es) | 1986-01-01 |
| GB2158828B (en) | 1987-12-09 |
| AU4166985A (en) | 1986-10-30 |
| FI851618L (fi) | 1985-10-26 |
| NO851603L (no) | 1985-10-28 |
| PT80343A (en) | 1985-05-01 |
| GB8410502D0 (en) | 1984-05-31 |
| PT80343B (en) | 1986-11-20 |
| EP0161843A1 (en) | 1985-11-21 |
| JPS615088A (ja) | 1986-01-10 |
| DK182585D0 (da) | 1985-04-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |