DK169674B1 - 1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser - Google Patents

1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser Download PDF

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Publication number
DK169674B1
DK169674B1 DK157686D DK157686D DK169674B1 DK 169674 B1 DK169674 B1 DK 169674B1 DK 157686 D DK157686 D DK 157686D DK 157686 D DK157686 D DK 157686D DK 169674 B1 DK169674 B1 DK 169674B1
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DK
Denmark
Prior art keywords
indole
fluorophenyl
tetrahydropyridin
methyl
formula
Prior art date
Application number
DK157686D
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Danish (da)
English (en)
Other versions
DK157686D0 (da
Inventor
Jens Kristian Perregaard
Original Assignee
Lundbeck & Co As H
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25673246&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK169674(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB858509164A external-priority patent/GB8509164D0/en
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of DK157686D0 publication Critical patent/DK157686D0/da
Application granted granted Critical
Publication of DK169674B1 publication Critical patent/DK169674B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/40—Nitrogen atoms, not forming part of a nitro radical, e.g. isatin semicarbazone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
DK157686D 1985-04-10 1986-04-08 1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser DK169674B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8509164 1985-04-10
GB858509164A GB8509164D0 (en) 1985-04-10 1985-04-10 Heterocyclic compounds
CA0616585A CA1338327B (en) 1985-04-10 1993-03-11 1-(4'-Fluorophenyl)-3,5-Substituted Indoles Useful in the Treatment of Psychic Disorders
CA616585 1993-03-11

Publications (2)

Publication Number Publication Date
DK157686D0 DK157686D0 (da) 1986-04-08
DK169674B1 true DK169674B1 (da) 1995-01-09

Family

ID=25673246

Family Applications (2)

Application Number Title Priority Date Filing Date
DK157686D DK169674B1 (da) 1985-04-10 1986-04-08 1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser
DK157686A DK157686A (da) 1985-04-10 1986-04-08 Indolderivater

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK157686A DK157686A (da) 1985-04-10 1986-04-08 Indolderivater

Country Status (11)

Country Link
US (2) US4710500A (ja)
EP (1) EP0200322B1 (ja)
JP (1) JPH064587B2 (ja)
AU (1) AU583607B2 (ja)
CA (2) CA1256437A (ja)
DK (2) DK169674B1 (ja)
FI (1) FI90976C (ja)
HK (1) HK116793A (ja)
IE (1) IE58370B1 (ja)
LU (1) LU90218I2 (ja)
NL (1) NL970016I2 (ja)

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FI90976B (fi) 1994-01-14
JPS61236764A (ja) 1986-10-22
LU90218I2 (fr) 1998-04-27
DK157686A (da) 1986-10-11
DK157686D0 (da) 1986-04-08
US4710500A (en) 1987-12-01
CA1256437A (en) 1989-06-27
FI90976C (fi) 1994-04-25
IE860618L (en) 1986-10-10
HK116793A (en) 1993-11-05
EP0200322B1 (en) 1990-02-28
NL970016I1 (nl) 1997-06-02
IE58370B1 (en) 1993-09-08
NL970016I2 (nl) 1997-09-01
USRE34299E (en) 1993-06-29
JPH064587B2 (ja) 1994-01-19
EP0200322A1 (en) 1986-11-05
FI861505A (fi) 1986-10-11
AU5590186A (en) 1986-10-16
CA1338327B (en) 1996-05-14
FI861505A0 (fi) 1986-04-09
AU583607B2 (en) 1989-05-04

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