DK169255B1 - Analogifremgangsmåde til fremstilling af thieno-isothiazol-1,1-dioxid-derivater og farmaceutisk acceptable salte heraf - Google Patents

Analogifremgangsmåde til fremstilling af thieno-isothiazol-1,1-dioxid-derivater og farmaceutisk acceptable salte heraf Download PDF

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Publication number
DK169255B1
DK169255B1 DK270583A DK270583A DK169255B1 DK 169255 B1 DK169255 B1 DK 169255B1 DK 270583 A DK270583 A DK 270583A DK 270583 A DK270583 A DK 270583A DK 169255 B1 DK169255 B1 DK 169255B1
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Prior art keywords
formula
compound
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reacted
meanings
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Application number
DK270583A
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Danish (da)
English (en)
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DK270583A (da
DK270583D0 (da
Inventor
Guy A Schiehser
Donald P Strike
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/468,221 external-priority patent/US4490527A/en
Priority claimed from GB838311653A external-priority patent/GB8311653D0/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of DK270583D0 publication Critical patent/DK270583D0/da
Publication of DK270583A publication Critical patent/DK270583A/da
Application granted granted Critical
Publication of DK169255B1 publication Critical patent/DK169255B1/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK270583A 1983-02-22 1983-06-13 Analogifremgangsmåde til fremstilling af thieno-isothiazol-1,1-dioxid-derivater og farmaceutisk acceptable salte heraf DK169255B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/468,221 US4490527A (en) 1982-09-30 1983-02-22 Benzo-fused heterocyclic anti-ulcer agents
US46822183 1983-02-22
GB8311653 1983-04-28
GB838311653A GB8311653D0 (en) 1983-04-28 1983-04-28 Fused heterocyclic compounds

Publications (3)

Publication Number Publication Date
DK270583D0 DK270583D0 (da) 1983-06-13
DK270583A DK270583A (da) 1984-08-23
DK169255B1 true DK169255B1 (da) 1994-09-26

Family

ID=26285976

Family Applications (1)

Application Number Title Priority Date Filing Date
DK270583A DK169255B1 (da) 1983-02-22 1983-06-13 Analogifremgangsmåde til fremstilling af thieno-isothiazol-1,1-dioxid-derivater og farmaceutisk acceptable salte heraf

Country Status (12)

Country Link
EP (1) EP0120585B1 (fr)
KR (1) KR900004150B1 (fr)
AU (1) AU563007B2 (fr)
CA (1) CA1215709A (fr)
DE (1) DE3468108D1 (fr)
DK (1) DK169255B1 (fr)
FI (1) FI78107C (fr)
GB (1) GB2137197B (fr)
GR (1) GR79987B (fr)
IE (1) IE56889B1 (fr)
NZ (1) NZ207209A (fr)
PT (1) PT78134B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4588719A (en) * 1984-04-27 1986-05-13 William H. Rorer, Inc. Bicyclic benzenoid aminoalkylene ethers and thioethers, pharmaceutical compositions and use
FI862513A (fi) * 1985-07-04 1987-01-05 Chemie Linz Ag Nya tieno-1,2-tiazolderivat, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska preparat.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2534689B2 (de) * 1974-09-16 1979-03-01 Basf Ag, 6700 Ludwigshafen 23-Dihydro-3-oxo-thieno-isothiazol-1,1-dioxide
GB1565966A (en) * 1976-08-04 1980-04-23 Allen & Hanburys Ltd Aminoalkyl furan derivatives
US4165378A (en) * 1977-04-20 1979-08-21 Ici Americas Inc. Guanidine derivatives of imidazoles and thiazoles
AT364852B (de) * 1977-11-05 1981-11-25 Thomae Gmbh Dr K Verfahren zur herstellung von kondensierten isothiazol-3(2h)-on-1,1-dioxiden und von deren salzen
GB2023133B (en) * 1978-04-26 1982-09-08 Glaxo Group Ltd Heterocyclic derivatives

Also Published As

Publication number Publication date
FI78107C (fi) 1989-06-12
FI78107B (fi) 1989-02-28
FI840687A (fi) 1984-08-23
EP0120585A1 (fr) 1984-10-03
FI840687A0 (fi) 1984-02-20
AU2472584A (en) 1984-08-30
KR840007880A (ko) 1984-12-11
PT78134A (en) 1984-03-01
DE3468108D1 (en) 1988-01-28
DK270583A (da) 1984-08-23
GR79987B (fr) 1984-10-31
GB2137197B (en) 1986-07-02
CA1215709A (fr) 1986-12-23
GB2137197A (en) 1984-10-03
EP0120585B1 (fr) 1987-12-16
PT78134B (en) 1986-06-11
DK270583D0 (da) 1983-06-13
AU563007B2 (en) 1987-06-25
KR900004150B1 (ko) 1990-06-16
IE840381L (en) 1984-08-22
NZ207209A (en) 1987-04-30
IE56889B1 (en) 1992-01-15
GB8404205D0 (en) 1984-03-21

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed