DK165744C - Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater - Google Patents

Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater

Info

Publication number
DK165744C
DK165744C DK617184A DK617184A DK165744C DK 165744 C DK165744 C DK 165744C DK 617184 A DK617184 A DK 617184A DK 617184 A DK617184 A DK 617184A DK 165744 C DK165744 C DK 165744C
Authority
DK
Denmark
Prior art keywords
sup
carbon atoms
alkyl group
procedures
preparing
Prior art date
Application number
DK617184A
Other languages
Danish (da)
English (en)
Other versions
DK617184A (da
DK165744B (da
DK617184D0 (da
Inventor
Kunihiro Ninomiya
Issei Nitta
Akihiro Tobe
Mitsuo Egawa
Ryoji Kikumoto
Original Assignee
Mitsubishi Chem Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Chem Ind filed Critical Mitsubishi Chem Ind
Publication of DK617184D0 publication Critical patent/DK617184D0/da
Publication of DK617184A publication Critical patent/DK617184A/da
Publication of DK165744B publication Critical patent/DK165744B/da
Application granted granted Critical
Publication of DK165744C publication Critical patent/DK165744C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK617184A 1984-01-05 1984-12-20 Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater DK165744C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP59000479A JPS60146891A (ja) 1984-01-05 1984-01-05 〔２，３−ｄ〕チエノピリミジン誘導体およびその塩
JP47984 1984-01-05

Publications (4)

Publication Number Publication Date
DK617184D0 DK617184D0 (da) 1984-12-20
DK617184A DK617184A (da) 1985-07-06
DK165744B DK165744B (da) 1993-01-11
DK165744C true DK165744C (da) 1993-06-07

Family

ID=11474905

Family Applications (1)

Application Number Title Priority Date Filing Date
DK617184A DK165744C (da) 1984-01-05 1984-12-20 Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater

Country Status (8)

Country Link
US (1) US4695568A (de)
EP (1) EP0150469B1 (de)
JP (1) JPS60146891A (de)
AT (1) ATE35137T1 (de)
CA (1) CA1224782A (de)
DE (1) DE3472106D1 (de)
DK (1) DK165744C (de)
HU (1) HU191161B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4734418A (en) * 1984-12-14 1988-03-29 Mitsui Petrochemical Industries, Ltd. Quinazoline compounds and antihypertensives
US4703120A (en) * 1986-04-28 1987-10-27 Ortho Pharmaceutical Corporation Furo(3,4-d)pyrimidine-2,4-dione derivatives and intermediates thereof
GB8912335D0 (en) * 1989-05-30 1989-07-12 Smithkline Beckman Intercredit Compounds
DE19636769A1 (de) * 1996-09-10 1998-03-12 Basf Ag 3-Substituierte Pyrido [4',3':4,5]thieno[2,3-d]pyrimidin-Derivate, ihre Herstellung und Verwendung
JPH10298078A (ja) * 1997-05-06 1998-11-10 Mitsubishi Chem Corp 抗不安薬
GB0112494D0 (en) * 2001-05-22 2001-07-11 Arachnova Therapeutics Ltd New therapeutic use
GB0216027D0 (en) 2002-07-10 2002-08-21 Arachnova Therapeutics Ltd New therapeutic use
BR0312511A (pt) * 2002-07-10 2005-04-12 Arachnova Therapeutics Ltd 4- (2-fluorofenil)-6-metil-2- (1-piperazinil) tieno [2,3-d] pirimidina no tratamento de distúrbio funcional dos intestinos
DE10232750A1 (de) * 2002-07-18 2004-02-05 Basf Ag Verfahren zur Herstellung von macrocyclischen Ketonen durch Dieckmann-Kondensation in der Gasphase
KR20050058511A (ko) * 2002-08-29 2005-06-16 아라크노바 테라퓨틱스 리미티드 4-(2-플루오로페닐)-6-메틸-2-(1-피페라지닐)티에노[2,3-디]피리미딘의 새로운 치료적 용도
EP1567163B1 (de) * 2003-01-13 2007-04-11 Dynogen Pharmaceuticals Inc. Verfahren zur behandlung von übelkeit, erbrechen, würgereiz oder jede kombination daraus
EP1558081A4 (de) 2003-01-13 2006-06-14 Dynogen Pharmaceuticals Inc Verfahren zur behandlung von funktionalen darmerkrankungen
JP2006522144A (ja) * 2003-04-04 2006-09-28 ダイノゲン ファーマシューティカルズ，インコーポレイテッド 下部尿路障害の治療方法
WO2005002583A1 (en) * 2003-07-07 2005-01-13 Mitsubishi Pharma Corporation Use of thieno`2,3-d ! pyrimidines for the prophylaxis or treatment of hyperactivity disorder
US20060293309A1 (en) * 2005-03-28 2006-12-28 Dynogen Pharmaceuticals, Inc. Method of treating disorders and conditions using peripherally-restricted antagonists and inhibitors
WO2008051282A2 (en) * 2006-03-31 2008-05-02 Dynogen Pharmaceuticals, Inc. Crystalline forms of 4-(2-fluorophenyl)-6-methyl-2-(piperazin-1-yl)thieno(2,3-d)pyrimidine
US20070254899A1 (en) * 2006-03-31 2007-11-01 Dynogen Pharmaceuticals, Inc. Soluble salts of thieno[2,3-d]pyrimidine derivatives
ES2827233T3 (es) * 2013-01-18 2021-05-20 Guangzhou Maxinovel Pharmaceuticals Co Ltd Compuesto heterocíclico de cinco y seis miembros, y método de preparación, composición farmacéutica y uso del mismo

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883651A (en) * 1969-08-08 1975-05-13 Boehringer Sohn Ingelheim Pharmaceutical compositions containing a 2-(aminoalkylamino)-4-amino-thieno{8 3,2-d{9 pyrimidine and method of use
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
GB1570494A (en) * 1975-11-28 1980-07-02 Ici Ltd Thienopyrimidine derivatives and their use as pesticides
US4196207A (en) * 1977-05-23 1980-04-01 Ici Australia Limited Process for controlling eradicating or preventing infestations of animals by Ixodid ticks
US4471117A (en) * 1979-06-21 1984-09-11 Janssen Pharmaceutica N.V. 3,4-Dihydro-2H-pyrimido(2,1-b)benzothiazoles
JPS5692875A (en) * 1979-12-27 1981-07-27 Dainippon Pharmaceut Co Ltd 2-aminoquinazoline derivative
EP0082023A3 (de) * 1981-12-16 1983-07-20 Sankyo Company Limited Thienopyrimidinderivate, ihre Herstellung und ihre Verwendung als Arzneimittel
FR2521144A1 (fr) * 1982-02-08 1983-08-12 Sanofi Sa Nouveaux derives de la piperazinyl-2 phenyl-4 quinazoline possedant des proprietes antidepressives, methode de preparation desdits composes et medicaments en contenant

Also Published As

Publication number Publication date
DK617184A (da) 1985-07-06
ATE35137T1 (de) 1988-07-15
CA1224782A (en) 1987-07-28
EP0150469B1 (de) 1988-06-15
DK165744B (da) 1993-01-11
DE3472106D1 (en) 1988-07-21
HU191161B (en) 1987-01-28
JPH0367071B2 (de) 1991-10-21
DK617184D0 (da) 1984-12-20
EP0150469A1 (de) 1985-08-07
HUT37435A (en) 1985-12-28
US4695568A (en) 1987-09-22
JPS60146891A (ja) 1985-08-02

Similar Documents

Publication Publication Date Title
DK165744C (da) Thienopyrimidinderivater, fremgangsmaader til fremstilling deraf og farmaceutiske praeparater
EP0163599A3 (en) Pyrimidopyrimidine derivatives, processes for producing them, pharmaceutical compositions containing them and their use as anti-allergic agents
DK0667852T3 (da) Hidtil ukendte 3,3-diphenylpropylaminer samt deres anvendelse og fremstilling
DK162519C (da) Dihydropyridazinonderivater og fremgangsmaade til fremstilling deraf samt farmaceutisk praeparat indeholdende forbindelserne
HUT52059A (en) Process for producing pharmaceutical compositions and new quinoline derivatives as a group of active components
ES2000346A6 (es) Un procedimiento para la preparacion de derivados de distamicina
ES8605506A1 (es) Procedimiento para preparar derivados de piperidina
DK12087D0 (da) Decahydroquinolinderivater, deres fremstilling og anvendelse samt praeparater med indhold deraf
ES8707243A1 (es) Un procedimiento para preparar derivados de tienopiridona
ES534505A0 (es) Un procedimiento para la preparacion de compuestos de 1, 4-dihidropiridina
MY102310A (en) New 5-oxy deravatives of tetrahydrofuran
ES8604960A1 (es) Procedimiento para preparar derivados de 1,6-naftiridina
EP0272596A3 (en) Theophyllinemethyldithiolan and theophyllinemethyldithianyl derivates, a method for their preparation and pharmaceutical compositions in which they are included
ES557597A0 (es) Procedimiento para preparar acidos hexenoicos
ES8600637A1 (es) Procedimiento de preparacion de derivados de piperacina
MY104048A (en) New allylaminoethylazoles.
HUT41029A (en) Process for preparing dioxolo-benzisoxazole derivatives
NO903084D0 (no) Farmasoeytisk anvendbare thiazol-derivater og fremgangsmaate for deres fremstilling.
ES8704947A1 (es) Un procedimiento para preparar un derivado de imidazopirida-zina
IE881752L (en) New aminoacylates of glycerol acetal
SE8305362D0 (sv) Novel substituted phenylazacycloalkanes, processes for preparation and pharmaceutical preparations for such compounds
ES485333A1 (es) Procedimiento para preparar derivados 5,6,7,8-tetrahidro-4 (3h)-quinazolinonicos y sus sales
GB1510128A (en) Cyano-heterocyclic compounds

Legal Events

Date Code Title Description
PBP Patent lapsed