DK164109C - Lh-rh-antagonister og deres farmaceutisk acceptable syreadditionssalte og fremgangsmaade til fremstilling deraf samt farmaceutisk middel indeholdende disse - Google Patents

Lh-rh-antagonister og deres farmaceutisk acceptable syreadditionssalte og fremgangsmaade til fremstilling deraf samt farmaceutisk middel indeholdende disse

Info

Publication number
DK164109C
DK164109C DK392284A DK392284A DK164109C DK 164109 C DK164109 C DK 164109C DK 392284 A DK392284 A DK 392284A DK 392284 A DK392284 A DK 392284A DK 164109 C DK164109 C DK 164109C
Authority
DK
Denmark
Prior art keywords
antagonists
procedures
preparing
composition containing
acid addition
Prior art date
Application number
DK392284A
Other languages
Danish (da)
English (en)
Other versions
DK392284D0 (da
DK164109B (da
DK392284A (da
Inventor
Hubert Jan Jozef Loozen
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of DK392284D0 publication Critical patent/DK392284D0/da
Publication of DK392284A publication Critical patent/DK392284A/da
Publication of DK164109B publication Critical patent/DK164109B/da
Application granted granted Critical
Publication of DK164109C publication Critical patent/DK164109C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/13—Luteinizing hormone-releasing hormone; related peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK392284A 1983-08-16 1984-08-15 Lh-rh-antagonister og deres farmaceutisk acceptable syreadditionssalte og fremgangsmaade til fremstilling deraf samt farmaceutisk middel indeholdende disse DK164109C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
NL8302875 1983-08-16
NL8302875 1983-08-16
NL8400153 1984-01-18
NL8400153 1984-01-18

Publications (4)

Publication Number Publication Date
DK392284D0 DK392284D0 (da) 1984-08-15
DK392284A DK392284A (da) 1985-02-17
DK164109B DK164109B (da) 1992-05-11
DK164109C true DK164109C (da) 1992-10-12

Family

ID=26645882

Family Applications (1)

Application Number Title Priority Date Filing Date
DK392284A DK164109C (da) 1983-08-16 1984-08-15 Lh-rh-antagonister og deres farmaceutisk acceptable syreadditionssalte og fremgangsmaade til fremstilling deraf samt farmaceutisk middel indeholdende disse

Country Status (13)

Country Link
US (1) US4628044A (fi)
EP (1) EP0145032B1 (fi)
KR (1) KR920004824B1 (fi)
AU (1) AU566672B2 (fi)
CA (1) CA1244009A (fi)
DE (1) DE3467173D1 (fi)
DK (1) DK164109C (fi)
ES (1) ES8602617A1 (fi)
FI (1) FI89174C (fi)
GR (1) GR80108B (fi)
HU (1) HU200481B (fi)
IE (1) IE57717B1 (fi)
PT (1) PT79074B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL70888A0 (en) * 1983-03-10 1984-05-31 Salk Inst For Biological Studi Gn rh antagonist peptides and pharmaceutical compositions containing them
US4565804A (en) * 1984-09-07 1986-01-21 The Salk Institute For Biological Studies GnRH Antagonists VI
US4690916A (en) * 1984-11-13 1987-09-01 Syntex (U.S.A.) Inc. Nona and decapeptide analogs of LHRH useful as LHRH antagonists
US4661472A (en) * 1985-05-09 1987-04-28 The Salk Institute For Biological Studies GnRH antagonists IX
HU194280B (en) * 1985-10-22 1988-01-28 Richter Gedeon Vegyeszet Process for producing new gonadoliberin analogues of high effectivity and pharmaceutical compositions containing them
DE3634435A1 (de) * 1986-10-09 1988-04-14 Hoechst Ag Analoga von gonadoliberin mit verbesserter loeslichkeit, verfahren zu deren herstellung, diese enthaltende mittel und ihre verwendung
US4801577A (en) * 1987-02-05 1989-01-31 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US4800191A (en) * 1987-07-17 1989-01-24 Schally Andrew Victor LHRH antagonists
US5064939A (en) * 1990-02-06 1991-11-12 The Salk Institute For Biological Studies Cyclic gnrh antagonists
US5502035A (en) * 1993-08-06 1996-03-26 Tap Holdings Inc. N-terminus modified analogs of LHRH
US5843901A (en) * 1995-06-07 1998-12-01 Advanced Research & Technology Institute LHRH antagonist peptides
DE19911771B4 (de) * 1999-03-17 2006-03-30 Zentaris Gmbh LHRH-Antagonist, Verfahren zu seiner Herstellung und seiner Verwendung
EP2161037A3 (en) 2003-04-22 2010-05-26 Ipsen Pharma Camptothecin-Somatostatin conjugates
JP5926876B2 (ja) * 2013-12-25 2016-05-25 本田技研工業株式会社 潤滑油の熱交換装置

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3165535D1 (en) * 1980-06-02 1984-09-20 Andrew Victor Schally Lh-rh antagonists
AU9102582A (en) * 1981-12-10 1983-06-16 David Howard Coy Lh-rh antagonists
FI832053L (fi) * 1982-06-10 1983-12-11 Syntex Inc Nonapeptid- och dekapeptidanaloger av lhrh anvaendbara som lhrh-antagonister samt deras framstaellningsfoerfarande
US4444759A (en) * 1982-07-26 1984-04-24 The Salk Institute For Biological Studies GnRH Antagonists II

Also Published As

Publication number Publication date
EP0145032B1 (en) 1987-11-04
GR80108B (en) 1984-12-14
ES535120A0 (es) 1985-12-01
IE842031L (en) 1985-02-16
DK392284D0 (da) 1984-08-15
PT79074B (en) 1986-08-14
FI89174C (fi) 1993-08-25
ES8602617A1 (es) 1985-12-01
HU200481B (en) 1990-06-28
FI843221A (fi) 1985-02-17
DE3467173D1 (en) 1987-12-10
KR850001774A (ko) 1985-04-01
DK164109B (da) 1992-05-11
AU566672B2 (en) 1987-10-29
DK392284A (da) 1985-02-17
FI89174B (fi) 1993-05-14
AU3174784A (en) 1985-02-21
PT79074A (en) 1984-09-01
EP0145032A1 (en) 1985-06-19
FI843221A0 (fi) 1984-08-15
IE57717B1 (en) 1993-03-10
KR920004824B1 (ko) 1992-06-18
HUT34766A (en) 1985-04-28
CA1244009A (en) 1988-11-01
US4628044A (en) 1986-12-09

Similar Documents

Publication Publication Date Title
DK474684A (da) 1-benzylaminoalkylpyrrolidinoner, syreadditionssalte deraf, fremgangsmaade til deres fremstilling og laegemidler indeholdende disse
DK573384A (da) Sphingosinderivater, fremgangsmaade til deres fremstilling og farmaceutiske kompositioner indeholdende disse derivater
DK247084D0 (da) 7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-quinolincarboxylsyrer,fremgangsmaader til deres fremstilling samt antibakterielle midler indeholdende disse
DK170785D0 (da) 4-substituerede-piperazin-2-carboxylsyre-derivater og farmaceutisk acceptable salte deraf, fremgangsmaade til fremstilling af saadanne forbindelser og farmaceutiske praeparater indeholdende disse
DK157931C (da) 1,3-dihydro-6-methyl-7-hydroxy-furo-(3,4-c)-pyridinderivater og terapeutisk acceptable syreadditionssalte deraf samt farmaceutiske praeparater indeholdende disse
DK522983A (da) Arylphenyletherderivater og syreadditionssalte deraf samt fremgangsmaade til fremstilling deraf
DK164109C (da) Lh-rh-antagonister og deres farmaceutisk acceptable syreadditionssalte og fremgangsmaade til fremstilling deraf samt farmaceutisk middel indeholdende disse
DK157877C (da) 9-deoxo-9a-methyl-9a-aza-9a-homoerythromycin d og farmaceutisk acceptable syreadditionssalte deraf samt 9-deoxo-9a-aza-9a-homoerythromycin d til anvendelse som udgangsmateriale ved fremstilling deraf
DK158357C (da) 9-deoxo-9a-(ethyl eller n-propyl)-9a-aza-9a-homoerythromycin a og farmaceutisk acceptable syreadditionssalte deraf samt farmaceutiske praeparater indeholdende disse forbindelser
DK162600C (da) Oe4-(2-hydroxycyklohexylmethyl)phenylaaalkansyrederivater og fremgangsmaade til fremstilling deraf samt farmaceutiske midler indeholdende disse
DK66086A (da) Dihydropyridiner, fremgangsmaader til fremstilling heraf samt farmaceutiske midler indeholdende disse
DK166878C (da) Fluorallylaminer og pharmakologisk acceptable syreadditionssalte deraf samt pharmaceutisk praeparat indeholdende disse forbindelser
DK307085D0 (da) 4-phenyl-2-trifluormethyl-1,3-dioxan-5-ylheptensyrederivater, fremgangsmaade til fremstilling deraf samt farmaceutiske midler indeholdende disse
DK160873C (da) Benzoquinolizinderivater samt farmaceutisk acceptable syreadditionssalte deraf og farmaceutisk middel indeholdende saadanne forbindelser og dettes fremstilling
DK162984C (da) 1-(2-ar-2-halogen-2-ethenyl)-1h-azoler, fremgangsmaade til deres fremstilling samt farmaceutiske praeparater indeholdende disse
DK610084A (da) Imidazolderivater eller syreadditionssalte deraf, fremgangsmaade til deres fremstilling og laegemidler indeholdende disse forbindelser
DK567184D0 (da) Pyridonderivater, fremgangsmaader til fremstilling deraf samt farmaceutiske midler indeholdende disse
DK209384D0 (da) 4-phenyl-tetrahydro-furano-pyridiner og syreadditionssalte deraf,fremgangsmaade til deres fremstilling og farmaceutiske kompositioner indeholdende forbindelserne
DK158518C (da) Phenylpiperazinderivater og syreadditionssalte deraf, fremgangsmaade til fremstilling deraf samt praeparater indeholdende derivaterne
DK165444C (da) Meta- og para-isopropenyl-alfa,alfa-dimethylbenzylamin og syreadditionssalte deraf samt fremgangsmaader til fremstilling deraf
DK628086D0 (da) Pyrazinderivater og farmaceutisk acceptable salte heraf samt fremgangsmaade til fremstilling af og farmaceutisk komposition indeholdende samme
DK507684D0 (da) Thiadiazinderivater, fremgangsmaader til deres fremstilling og farmaceutiske midler indeholdende disse thiadiazinderivater
DK163247C (da) Gonadolibeinderivater, farmaceutisk acceptable syreadditionssalte og complexer heraf samt en fremgangsmaade til fremstilling af disse og et farmaceutisk praeparat indeholdende disse
DK240984A (da) 5-(4-chlor-3-sulfamoylbenzoyl)-2,3-dihydro-2-benzofurancarboxylsyrer, fremgangsmaader til deres fremstilling samt farmaceutiske praeparater indeholdende disse
DK65986D0 (da) Dihydropyridiner, fremgangsmaader til fremstilling heraf samt farmaceutiske midler indeholdende disse

Legal Events

Date Code Title Description
PBP Patent lapsed