DK157686A - Indolderivater - Google Patents

Indolderivater Download PDF

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Publication number
DK157686A
DK157686A DK157686A DK157686A DK157686A DK 157686 A DK157686 A DK 157686A DK 157686 A DK157686 A DK 157686A DK 157686 A DK157686 A DK 157686A DK 157686 A DK157686 A DK 157686A
Authority
DK
Denmark
Prior art keywords
indole derivatives
indole
derivatives
Prior art date
Application number
DK157686A
Other languages
Danish (da)
English (en)
Inventor
Jens Kristian Perregaard
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25673246&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK157686(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB858509164A external-priority patent/GB8509164D0/en
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of DK157686A publication Critical patent/DK157686A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/40—Nitrogen atoms, not forming part of a nitro radical, e.g. isatin semicarbazone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
DK157686A 1985-04-10 1986-04-08 Indolderivater DK157686A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB858509164A GB8509164D0 (en) 1985-04-10 1985-04-10 Heterocyclic compounds
CA0616585A CA1338327B (en) 1985-04-10 1993-03-11 1-(4'-Fluorophenyl)-3,5-Substituted Indoles Useful in the Treatment of Psychic Disorders

Publications (1)

Publication Number Publication Date
DK157686A true DK157686A (da) 1986-10-11

Family

ID=25673246

Family Applications (2)

Application Number Title Priority Date Filing Date
DK157686D DK169674B1 (da) 1985-04-10 1986-04-08 1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser
DK157686A DK157686A (da) 1985-04-10 1986-04-08 Indolderivater

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK157686D DK169674B1 (da) 1985-04-10 1986-04-08 1-Aryl-3-tetrahydropyridyl-, 1-aryl-3-piperidyl- eller 1-aryl-3-piperazinyl-indolderivater, fremgangsmåde til deres fremstilling og farmaceutiske kompositioner, der indeholder disse forbindelser

Country Status (11)

Country Link
US (2) US4710500A (de)
EP (1) EP0200322B1 (de)
JP (1) JPH064587B2 (de)
AU (1) AU583607B2 (de)
CA (2) CA1256437A (de)
DK (2) DK169674B1 (de)
FI (1) FI90976C (de)
HK (1) HK116793A (de)
IE (1) IE58370B1 (de)
LU (1) LU90218I2 (de)
NL (1) NL970016I2 (de)

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DE2322470A1 (de) * 1973-05-04 1974-11-21 Boehringer Sohn Ingelheim Neue indolyl-piperidino-(bzw. 1,2,5,6tetrahydro-pyridyl-)butyrophenone und verfahren zu ihrer herstellung
IL48508A (en) * 1974-12-09 1979-10-31 Roussel Uclaf Pharmaceutical compositions comprising piperidylindole derivatives
FR2349331A1 (fr) * 1976-04-30 1977-11-25 Roussel Uclaf Nouveaux derives de 2,3 dihydro a/4-(3-indolyl) 1-piperidinyl/methyl 1,4-benzodioxin-2-methanol, un procede pour leur preparation et leur application comme medicaments
FR2362628A1 (fr) * 1976-08-26 1978-03-24 Roussel Uclaf Nouveaux derives du piperidyl-indole et leurs sels, procede de preparation et application a titre de medicaments
FR2421900A1 (fr) * 1977-03-17 1979-11-02 Sauba Lab Piperazino-3-indoles, leur procede de preparation et leurs applications therapeutiques
FR2426465B1 (de) * 1978-01-16 1983-04-29 Roussel Uclaf
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FR2444678A2 (fr) * 1978-12-22 1980-07-18 Roussel Uclaf Nouveau procede de preparation de derives du piperidyl-indole et de leurs sels
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SE8004129L (sv) * 1979-07-13 1981-01-14 Roussel Uclaf Nya tetrahydropyridin-4-yl-indolderivat samt salter derav, framstellning och anvendning derav sasom lekemedel samt kompositioner innehallande dessa foreningar
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IE58370B1 (en) 1993-09-08
CA1256437A (en) 1989-06-27
NL970016I2 (nl) 1997-09-01
HK116793A (en) 1993-11-05
FI90976B (fi) 1994-01-14
CA1338327B (en) 1996-05-14
EP0200322A1 (de) 1986-11-05
AU5590186A (en) 1986-10-16
DK169674B1 (da) 1995-01-09
FI861505A0 (fi) 1986-04-09
JPH064587B2 (ja) 1994-01-19
AU583607B2 (en) 1989-05-04
FI90976C (fi) 1994-04-25
DK157686D0 (da) 1986-04-08
EP0200322B1 (de) 1990-02-28
FI861505A (fi) 1986-10-11
IE860618L (en) 1986-10-10
JPS61236764A (ja) 1986-10-22
US4710500A (en) 1987-12-01
LU90218I2 (fr) 1998-04-27
USRE34299E (en) 1993-06-29
NL970016I1 (nl) 1997-06-02

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