DK152668C - Analogifremgangsmaade til fremstilling af 2-(1-piperidinyl)-benzophenonderivater - Google Patents

Analogifremgangsmaade til fremstilling af 2-(1-piperidinyl)-benzophenonderivater

Info

Publication number
DK152668C
DK152668C DK289382A DK289382A DK152668C DK 152668 C DK152668 C DK 152668C DK 289382 A DK289382 A DK 289382A DK 289382 A DK289382 A DK 289382A DK 152668 C DK152668 C DK 152668C
Authority
DK
Denmark
Prior art keywords
piperidinyl
preparing
benzophenone derivatives
analogy procedure
analogy
Prior art date
Application number
DK289382A
Other languages
Danish (da)
English (en)
Other versions
DK152668B (da
DK289382A (da
Inventor
Bernard Majoie
Francois Bellamy
Pierre Dodey
Jacques Robin
Original Assignee
Fournier Innovation Synergie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fournier Innovation Synergie filed Critical Fournier Innovation Synergie
Publication of DK289382A publication Critical patent/DK289382A/da
Publication of DK152668B publication Critical patent/DK152668B/da
Application granted granted Critical
Publication of DK152668C publication Critical patent/DK152668C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK289382A 1981-06-29 1982-06-28 Analogifremgangsmaade til fremstilling af 2-(1-piperidinyl)-benzophenonderivater DK152668C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8112745 1981-06-29
FR8112745A FR2508445A1 (fr) 1981-06-29 1981-06-29 Nouveaux derives de benzoyl-phenyl-piperidine, leur procede de preparation et leur application, notamment en therapeutique

Publications (3)

Publication Number Publication Date
DK289382A DK289382A (da) 1982-12-30
DK152668B DK152668B (da) 1988-04-11
DK152668C true DK152668C (da) 1988-09-19

Family

ID=9259970

Family Applications (1)

Application Number Title Priority Date Filing Date
DK289382A DK152668C (da) 1981-06-29 1982-06-28 Analogifremgangsmaade til fremstilling af 2-(1-piperidinyl)-benzophenonderivater

Country Status (26)

Country Link
US (2) US4528294A (xx)
EP (1) EP0069012B1 (xx)
JP (1) JPS588061A (xx)
KR (1) KR880001298B1 (xx)
AR (1) AR230048A1 (xx)
AT (1) ATE9795T1 (xx)
AU (1) AU550320B2 (xx)
CA (1) CA1187501A (xx)
CS (1) CS235542B2 (xx)
DD (1) DD202557A5 (xx)
DE (1) DE3260949D1 (xx)
DK (1) DK152668C (xx)
ES (1) ES513565A0 (xx)
FI (1) FI77447C (xx)
FR (1) FR2508445A1 (xx)
GR (1) GR76401B (xx)
HU (1) HU189150B (xx)
IE (1) IE53189B1 (xx)
IL (2) IL66123A (xx)
NO (1) NO160136C (xx)
OA (1) OA07133A (xx)
PH (1) PH17368A (xx)
PT (1) PT75135B (xx)
SU (1) SU1147251A3 (xx)
YU (1) YU43799B (xx)
ZA (1) ZA824536B (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL82573A0 (en) * 1986-05-30 1987-11-30 Sori Soc Rech Ind Preparation of benzoylphenyl-piperidine derivatives
FR2620027A1 (fr) * 1987-09-09 1989-03-10 Fournier Innovation Synergie Nouvelle utilisation de la (5-amino-2-(4-methyl-1-piperidinyl)phenyl)-(4-chlorophenyl)-methanone
AU4971600A (en) * 1999-05-21 2000-12-12 Eli Lilly And Company Immunopotentiator agents
EP1286984A2 (en) * 2000-03-10 2003-03-05 Pharmacia Corporation Method for the preparation of tetrahydrobenzothiepines

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3202655A (en) * 1962-04-27 1965-08-24 Yvon G Perron 6-[alpha-substituted-alpha-(2-or 3-heterocyclic) acetamido] penicillanic acid and nontoxic salts thereof
NL124621C (xx) * 1962-11-13
FR1375300A (fr) * 1962-11-13 1964-10-16 Hoffmann La Roche Dérivés de benzophénone et leur préparation
FR1403939A (fr) * 1963-06-07 1965-06-25 Hoffmann La Roche Procédé pour la préparation de dérivés de benzodiazépine
FR1526708A (fr) * 1966-06-13 1968-05-24 Upjohn Co 1.3-amino-alcools, leurs intermédiaires et dérivés et leur procédé de préparation
US3668199A (en) * 1966-06-13 1972-06-06 Upjohn Co 1,3-aminoalcohols
FR1530393A (fr) * 1966-07-11 1968-06-21 Hoffmann La Roche Procédé pour la préparation de dérivés de pipéridine
IE34545B1 (en) * 1969-10-01 1975-06-11 Continental Pharma Amino-alcohols,their salts and process for preparing the same
HU167950B (xx) * 1973-07-26 1976-01-28
US4064121A (en) * 1973-07-26 1977-12-20 Richter Gedeon Vegyeszeti Gyar Rt. Substituted nitrobenzophenone derivatives and a process for the preparation thereof
HU167949B (xx) * 1973-07-26 1976-01-28
US4021563A (en) * 1975-02-06 1977-05-03 Sven Eric Harry Hernestam Method of treating cardiac arrhythmia with γ-piperidino-butyrophenones
IE49998B1 (en) * 1979-08-06 1986-01-22 Merrell Dow Pharma 4-(naphthalenyloxy)piperidine derivatives

Also Published As

Publication number Publication date
FI822215L (fi) 1982-12-30
EP0069012B1 (fr) 1984-10-10
PT75135B (fr) 1984-05-25
EP0069012A1 (fr) 1983-01-05
CS235542B2 (en) 1985-05-15
YU43799B (en) 1989-12-31
PH17368A (en) 1984-08-06
JPH0127062B2 (xx) 1989-05-26
FI77447C (fi) 1989-03-10
ES8304936A1 (es) 1983-03-16
IE821475L (en) 1982-12-29
JPS588061A (ja) 1983-01-18
DD202557A5 (de) 1983-09-21
KR880001298B1 (ko) 1988-07-22
AU8542982A (en) 1983-01-06
ZA824536B (en) 1983-04-27
IL66123A0 (en) 1982-09-30
OA07133A (fr) 1984-03-31
GR76401B (xx) 1984-08-10
DK152668B (da) 1988-04-11
US4680402A (en) 1987-07-14
NO160136B (no) 1988-12-05
US4528294A (en) 1985-07-09
IL76287A0 (en) 1986-01-31
KR840000514A (ko) 1984-02-22
ATE9795T1 (de) 1984-10-15
AU550320B2 (en) 1986-03-20
IL66123A (en) 1986-02-28
FI822215A0 (fi) 1982-06-21
SU1147251A3 (ru) 1985-03-23
FR2508445A1 (fr) 1982-12-31
DK289382A (da) 1982-12-30
HU189150B (en) 1986-06-30
PT75135A (fr) 1982-07-01
DE3260949D1 (en) 1984-11-15
ES513565A0 (es) 1983-03-16
IE53189B1 (en) 1988-08-17
YU141582A (en) 1985-03-20
FR2508445B1 (xx) 1984-02-10
NO160136C (no) 1989-03-15
AR230048A1 (es) 1984-02-29
NO822185L (no) 1982-12-30
CA1187501A (en) 1985-05-21
FI77447B (fi) 1988-11-30

Similar Documents

Publication Publication Date Title
DK280083D0 (da) Fremgangsmade til fremstilling af 2-(4-puridyl)-thiazolderivater
DK157019C (da) Analogifremgangsmaade til fremstilling af 2-amino-4-hydroxyquinazolinderivater
DK164593C (da) Analogifremgangsmaade til fremstilling af 1-phenyl-2-piperidinopropanolderivater
DK50779A (da) Fremgangsmaade til fremstilling af piperazinderivater
DK28282A (da) Fremgangsmaade til fremstilling af hexapyranoseforbindelser eller salte deraf
DK161024C (da) Analogifremgangsmaade til fremstilling af cephalosporinderivater
DK221182A (da) Fremgangsmaade til fremstilling af chirale 2-(2-benzyl-3-mercaptopropionyl)amino-1-alkanolderivater eller chirale 2-(2-benzyl-3-mercaptopropionyl)amino-4-methylthiosmoersyrer eller faraaaceutisk acceptable salte af syrerne
DK162991C (da) Analogifremgangsmaade til fremstilling af thiazolidinylalkylenpiperazinderivater
DK151252C (da) Analogifremgangsmaade til fremstilling af 3-alkyltio-4-oxoquinolinforbindelser
DK150070C (da) Analogifremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater
DK145698C (da) Analogifremgangsmaade til fremstilling af 2-alkoxyadeninderivater
DK152428C (da) Analogifremgangsmaade til fremstilling af 2-(aminoalkylthio)-quinolinderivater
DK152132C (da) Analogifremgangsmaade til fremstilling af derivater af 5,6,7,7a-tetrahydro-4h-thienooe3,2-caapyridin-2-on
DK312082A (da) Fremgangsmaade til fremstilling af benzothiazolsulfonamidderivater
DK156722C (da) Analogifremgangsmaade til fremstilling af 2-piperazinopyrimidinderivater
DK147145C (da) Analogifremgangsmaade til fremstilling af chlorambucilderivater
DK164403C (da) Analogifremgangsmaade til fremstilling af benzothiazolinderivater
DK157849C (da) Analogifremgangsmaade til fremstilling af 2-(hydroxyphenyl)-indoler
DK237383D0 (da) Fremgangsmade til fremstilling af piperazinderivater
DK161310C (da) Analogifremgangsmaade til fremstilling af aminopropoxyphenylderivater
DK163000C (da) Analogifremgangsmaade til fremstilling af vinylthioacetamido-1-dethia-1-oxa-cephalosporinderivater
DK154136C (da) Analogifremgangsmaade til fremstilling af 2-amino-3-benzoylphenylacetamider
DK372081A (da) Fremgangsmaade til fremstilling af fluorerede pentendiaminderivater
DK152674C (da) Analogifremgangsmaade til fremstilling af 3-metyltiometyl-4-oxo-quinolonderivater
DK4982A (da) Fremgangsmaade til fremstilling af pyridinylsubstituerede benzimidazolderivater

Legal Events

Date Code Title Description
PBP Patent lapsed