DK152365C - Azetidinderivater til anvendelse som mellemprodukter ved fremstilling af cephalosporansyrederivater og fremgangsmaade til fremstilling af saadanne azetidinderivater - Google Patents

Azetidinderivater til anvendelse som mellemprodukter ved fremstilling af cephalosporansyrederivater og fremgangsmaade til fremstilling af saadanne azetidinderivater

Info

Publication number
DK152365C
DK152365C DK045875A DK45875A DK152365C DK 152365 C DK152365 C DK 152365C DK 045875 A DK045875 A DK 045875A DK 45875 A DK45875 A DK 45875A DK 152365 C DK152365 C DK 152365C
Authority
DK
Denmark
Prior art keywords
derivatives
azetide
azetidin
intermediates
procedure
Prior art date
Application number
DK045875A
Other languages
Danish (da)
English (en)
Other versions
DK45875A (xx
DK152365B (da
Inventor
Jan Verweij
Hong Sheng Tan
Original Assignee
Gist Brocades Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gist Brocades Nv filed Critical Gist Brocades Nv
Publication of DK45875A publication Critical patent/DK45875A/da
Publication of DK152365B publication Critical patent/DK152365B/da
Application granted granted Critical
Publication of DK152365C publication Critical patent/DK152365C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02Preparation
    • C07D501/08Preparation by forming the ring or condensed ring systems
    • C07D501/10Preparation by forming the ring or condensed ring systems from compounds containing the penicillin ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/30Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino-radical acylated by an araliphatic carboxylic acid

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Health & Medical Sciences (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK045875A 1974-02-08 1975-02-07 Azetidinderivater til anvendelse som mellemprodukter ved fremstilling af cephalosporansyrederivater og fremgangsmaade til fremstilling af saadanne azetidinderivater DK152365C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB581174 1974-02-08
GB5811/74A GB1483526A (en) 1974-02-08 1974-02-08 Azetidine derivatives

Publications (3)

Publication Number Publication Date
DK45875A DK45875A (xx) 1975-10-06
DK152365B DK152365B (da) 1988-02-22
DK152365C true DK152365C (da) 1988-08-01

Family

ID=9803053

Family Applications (2)

Application Number Title Priority Date Filing Date
DK045875A DK152365C (da) 1974-02-08 1975-02-07 Azetidinderivater til anvendelse som mellemprodukter ved fremstilling af cephalosporansyrederivater og fremgangsmaade til fremstilling af saadanne azetidinderivater
DK446978A DK151810C (da) 1974-02-08 1978-10-06 Fremgangsmaade til fremstilling af cephalosporansyrederivater

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK446978A DK151810C (da) 1974-02-08 1978-10-06 Fremgangsmaade til fremstilling af cephalosporansyrederivater

Country Status (17)

Country Link
US (1) US4007202A (xx)
JP (2) JPS5924991B2 (xx)
BE (1) BE825325A (xx)
CH (1) CH594661A5 (xx)
CS (2) CS189635B2 (xx)
DE (1) DE2505280A1 (xx)
DK (2) DK152365C (xx)
FI (1) FI63748C (xx)
FR (1) FR2260584B1 (xx)
GB (1) GB1483526A (xx)
HU (1) HU172237B (xx)
IE (1) IE40636B1 (xx)
IT (1) IT1046090B (xx)
LU (1) LU71817A1 (xx)
NL (1) NL182727C (xx)
SE (2) SE429337B (xx)
SU (2) SU577979A3 (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1465893A (en) * 1973-02-09 1977-03-02 Gist Brocades Nv I-carboxypropenyl-4-iminothio-azetidine-2-one derivatives methods for their preparation and use
US4046761A (en) * 1974-02-08 1977-09-06 Gist-Brocades N.V. Process for preparing cephalosporin derivatives
US4301278A (en) * 1974-02-26 1981-11-17 Ciba-Geigy Corporation Process for the manufacture of enol derivatives
US4147864A (en) * 1975-02-20 1979-04-03 Ciba-Geigy Corporation Process for the manufacture of 7β-amino-3-cephem-3-ol-4 carboxylic acid compounds
GB2099817B (en) * 1981-04-10 1985-05-15 Otsuka Kagaku Yakuhin Azetidinone derivatives and process for the preparation of the same
JPS5865289A (ja) * 1981-10-14 1983-04-18 Sankyo Co Ltd アゼチジノン誘導体
JPS59164771A (ja) * 1983-03-10 1984-09-17 Otsuka Chem Co Ltd 塩素化アゼチジノン誘導体の製造方法
JPH0487971A (ja) * 1990-07-13 1992-03-19 Mishima Seishi Kk 帯電防止および又は静電気シールド用包装容器
US6383773B2 (en) 1998-04-23 2002-05-07 Massachusetts Institute Of Technology Penicillin conversion

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL204361A (xx) * 1955-04-22 1900-01-01
US3843682A (en) * 1972-05-15 1974-10-22 Lilly Co Eli 2-chlorosulfinyl-3-imido-azetedin-4-ones

Also Published As

Publication number Publication date
DK45875A (xx) 1975-10-06
NL182727C (nl) 1988-05-02
FR2260584B1 (xx) 1979-02-23
SE7810147L (sv) 1978-09-27
IT1046090B (it) 1980-06-30
DK446978A (da) 1978-10-06
NL182727B (nl) 1987-12-01
JPS5924991B2 (ja) 1984-06-13
DK152365B (da) 1988-02-22
SU577979A3 (ru) 1977-10-25
BE825325A (fr) 1975-08-07
SE7501375L (xx) 1975-08-11
DK151810B (da) 1988-01-04
CS189635B2 (en) 1979-04-30
NL7501457A (nl) 1975-08-12
US4007202A (en) 1977-02-08
DE2505280A1 (de) 1975-08-14
JPS58150598A (ja) 1983-09-07
FI63748C (fi) 1983-08-10
JPS6047277B2 (ja) 1985-10-21
LU71817A1 (xx) 1975-06-24
IE40636L (en) 1975-08-08
FR2260584A1 (xx) 1975-09-05
SE429337B (sv) 1983-08-29
HU172237B (hu) 1978-07-28
CS189642B2 (en) 1979-04-30
CH594661A5 (xx) 1978-01-13
SU656526A3 (ru) 1979-04-05
JPS50108257A (xx) 1975-08-26
GB1483526A (en) 1977-08-24
DK151810C (da) 1988-06-06
FI63748B (fi) 1983-04-29
SE427842B (sv) 1983-05-09
IE40636B1 (en) 1979-07-18
FI750346A (xx) 1975-08-09

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