DK142751B - Analogifremgangsmåde til fremstilling af 4-((2-methyl-3-hydroxy-4-hydroxymethyl)-5-pyridyl-N-methyl-N'-piperazinyl)-p-fluor-butyrophenon eller syreadditionssalte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af 4-((2-methyl-3-hydroxy-4-hydroxymethyl)-5-pyridyl-N-methyl-N'-piperazinyl)-p-fluor-butyrophenon eller syreadditionssalte heraf. Download PDF

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Publication number
DK142751B
DK142751B DK168074AA DK168074A DK142751B DK 142751 B DK142751 B DK 142751B DK 168074A A DK168074A A DK 168074AA DK 168074 A DK168074 A DK 168074A DK 142751 B DK142751 B DK 142751B
Authority
DK
Denmark
Prior art keywords
methyl
fluoro
preparation
butyrophenone
piperazinyl
Prior art date
Application number
DK168074AA
Other languages
Danish (da)
English (en)
Other versions
DK142751C (xx
Inventor
Andre Esanu
Original Assignee
Soc D Etudes Prod Chimique
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Soc D Etudes Prod Chimique filed Critical Soc D Etudes Prod Chimique
Publication of DK142751B publication Critical patent/DK142751B/da
Application granted granted Critical
Publication of DK142751C publication Critical patent/DK142751C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK168074AA 1973-03-28 1974-03-27 Analogifremgangsmåde til fremstilling af 4-((2-methyl-3-hydroxy-4-hydroxymethyl)-5-pyridyl-N-methyl-N'-piperazinyl)-p-fluor-butyrophenon eller syreadditionssalte heraf. DK142751B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB1481573 1973-03-28
GB1481573A GB1433222A (xx) 1973-03-28 1973-03-28

Publications (2)

Publication Number Publication Date
DK142751B true DK142751B (da) 1981-01-12
DK142751C DK142751C (xx) 1981-08-17

Family

ID=10047975

Family Applications (1)

Application Number Title Priority Date Filing Date
DK168074AA DK142751B (da) 1973-03-28 1974-03-27 Analogifremgangsmåde til fremstilling af 4-((2-methyl-3-hydroxy-4-hydroxymethyl)-5-pyridyl-N-methyl-N'-piperazinyl)-p-fluor-butyrophenon eller syreadditionssalte heraf.

Country Status (16)

Country Link
US (1) US3903088A (xx)
JP (1) JPS532876B2 (xx)
AR (1) AR200519A1 (xx)
AT (1) AT332569B (xx)
AU (1) AU473846B2 (xx)
BE (1) BE812558A (xx)
CA (1) CA1011337A (xx)
CH (1) CH592652A5 (xx)
DK (1) DK142751B (xx)
ES (1) ES424318A1 (xx)
FR (2) FR2223370B1 (xx)
GB (1) GB1433222A (xx)
IN (1) IN139464B (xx)
NL (1) NL7403812A (xx)
OA (1) OA04692A (xx)
ZA (1) ZA741617B (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA783521B (en) * 1977-07-12 1979-06-27 Scras New pyrimidine derivatives,their preparation and therapeutic compositions containing the same
US4175769A (en) * 1978-05-01 1979-11-27 Kazmark Eugene A Portable luggage carrier

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3557131A (en) * 1965-06-15 1971-01-19 Dainippon Pharmaceutical Co Nicotinate derivatives of vitamin b6
US3717636A (en) * 1970-01-21 1973-02-20 A Esanu Salts of pyridoxine mono-esters
CH541568A (de) * 1970-12-07 1973-10-31 Ciba Geigy Ag Verfahren zur Herstellung von neuen Imidazolidinonderivaten

Also Published As

Publication number Publication date
AT332569B (de) 1976-10-11
ES424318A1 (es) 1976-06-01
FR2223370B1 (xx) 1976-12-17
ATA256074A (de) 1976-01-15
DE2415128B2 (de) 1976-10-07
AU6670374A (en) 1975-09-18
DK142751C (xx) 1981-08-17
US3903088A (en) 1975-09-02
JPS532876B2 (xx) 1978-02-01
CH592652A5 (xx) 1977-10-31
CA1011337A (en) 1977-05-31
ZA741617B (en) 1975-02-26
IN139464B (xx) 1976-06-19
GB1433222A (xx) 1976-04-22
FR2223019B1 (xx) 1977-11-04
AR200519A1 (es) 1974-11-15
NL7403812A (xx) 1974-10-01
FR2223370A1 (xx) 1974-10-25
JPS5046679A (xx) 1975-04-25
DE2415128A1 (de) 1974-10-10
BE812558A (fr) 1974-09-20
FR2223019A1 (xx) 1974-10-25
AU473846B2 (en) 1976-07-01
OA04692A (fr) 1980-07-31

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