DK142707B - Analogifremgangsmåde til fremstilling af 19-oxygenerede steroidforbindelser. - Google Patents

Analogifremgangsmåde til fremstilling af 19-oxygenerede steroidforbindelser. Download PDF

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Publication number
DK142707B
DK142707B DK438577AA DK438577A DK142707B DK 142707 B DK142707 B DK 142707B DK 438577A A DK438577A A DK 438577AA DK 438577 A DK438577 A DK 438577A DK 142707 B DK142707 B DK 142707B
Authority
DK
Denmark
Prior art keywords
group
hydroxy
formula
solution
hydrogen atom
Prior art date
Application number
DK438577AA
Other languages
Danish (da)
English (en)
Other versions
DK142707C (xx
DK438577A (xx
Inventor
Michel Biollaz
Peter Wieland
Georg Anner
Hellmut Ueberwasser
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from LU75936A external-priority patent/LU75936A1/xx
Priority claimed from LU76966A external-priority patent/LU76966A1/xx
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of DK438577A publication Critical patent/DK438577A/da
Publication of DK142707B publication Critical patent/DK142707B/da
Application granted granted Critical
Publication of DK142707C publication Critical patent/DK142707C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/007—3 membered carbocyclic rings in position 6-7
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/001—Lactones
    • C07J21/003—Lactones at position 17
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/005—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton spiro-condensed
    • C07J33/007—Cyclic thioketals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK438577AA 1976-10-05 1977-10-04 Analogifremgangsmåde til fremstilling af 19-oxygenerede steroidforbindelser. DK142707B (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
LU75936A LU75936A1 (xx) 1976-10-05 1976-10-05
LU75936 1976-10-05
LU76966 1977-03-17
LU76966A LU76966A1 (xx) 1977-03-17 1977-03-17

Publications (3)

Publication Number Publication Date
DK438577A DK438577A (xx) 1978-04-06
DK142707B true DK142707B (da) 1980-12-29
DK142707C DK142707C (xx) 1981-10-05

Family

ID=26640214

Family Applications (1)

Application Number Title Priority Date Filing Date
DK438577AA DK142707B (da) 1976-10-05 1977-10-04 Analogifremgangsmåde til fremstilling af 19-oxygenerede steroidforbindelser.

Country Status (16)

Country Link
US (1) US4150127A (xx)
JP (1) JPS5346952A (xx)
AT (1) ATA705277A (xx)
AU (1) AU512101B2 (xx)
CA (1) CA1099701A (xx)
DD (1) DD132349A5 (xx)
DE (1) DE2744255A1 (xx)
DK (1) DK142707B (xx)
ES (1) ES462882A1 (xx)
FI (1) FI58779C (xx)
FR (1) FR2367079A1 (xx)
IL (1) IL53058A0 (xx)
NL (1) NL7710939A (xx)
NO (1) NO773381L (xx)
NZ (1) NZ185341A (xx)
SE (1) SE7711094L (xx)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4259240A (en) * 1979-09-28 1981-03-31 Advance Biofactures Corporation Synthesis of furyl intermediates, and cardenolides and their isomers prepared therefrom
DE3326013A1 (de) * 1983-07-15 1985-01-24 Schering AG, 1000 Berlin und 4709 Bergkamen 15,16-methylen-17(alpha)-pregna-4,6-dien-21-carbonsaeuresalze, diese enthaltende pharmazeutische praeparate sowie verfahren zu deren herstellung
DE3330084A1 (de) * 1983-08-17 1985-03-07 Schering AG, 1000 Berlin und 4709 Bergkamen 7(alpha)-alkoxycarbonyl-3-oxo-17(alpha)-pregn-4-en-21,17-carbolactone und deren 21-carbonsaeuresalze, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
JPH0425327Y2 (xx) * 1985-11-08 1992-06-17
FR2656309B1 (fr) * 1989-12-22 1992-05-07 Roussel Uclaf Nouveaux produits sterouides comportant en position 10, un radical ethyle substitue, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant.
EP0738275B9 (en) * 1994-01-06 2001-03-21 Sri International Novel antiandrogenic agents and related pharmaceutical compositions and methods of use
WO2012107513A1 (en) * 2011-02-10 2012-08-16 Crystal Pharma, S.A.U. Process for obtaining drospirenone
EP2853958A1 (fr) 2013-09-26 2015-04-01 Montres Breguet SA Pièce d'horlogerie à niveau acoustique amélioré

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4058522A (en) * 1973-07-09 1977-11-15 Richter Gedeon Vegyeszeti Gyar Rt. Steroids effective against heavy-metal poisoning
US4028348A (en) * 1976-02-17 1977-06-07 Richter Gedeon Vegyeszeti Gyar Rt 6-Amino-5β,19-cycloandrostane derivatives

Also Published As

Publication number Publication date
AU512101B2 (en) 1980-09-25
NL7710939A (nl) 1978-04-07
NZ185341A (en) 1979-06-19
ATA705277A (de) 1981-07-15
FI772900A (fi) 1978-04-06
IL53058A0 (en) 1977-12-30
AU2932577A (en) 1979-04-12
DK142707C (xx) 1981-10-05
CA1099701A (en) 1981-04-21
US4150127A (en) 1979-04-17
DD132349A5 (de) 1978-09-20
FR2367079A1 (fr) 1978-05-05
DE2744255A1 (de) 1978-04-06
SE7711094L (sv) 1978-04-06
JPS5346952A (en) 1978-04-27
NO773381L (no) 1978-04-06
FR2367079B1 (xx) 1980-04-18
ES462882A1 (es) 1978-12-16
DK438577A (xx) 1978-04-06
FI58779C (fi) 1981-04-10
FI58779B (fi) 1980-12-31

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