DK141064B - Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. - Google Patents

Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. Download PDF

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Publication number
DK141064B
DK141064B DK22277AA DK22277A DK141064B DK 141064 B DK141064 B DK 141064B DK 22277A A DK22277A A DK 22277AA DK 22277 A DK22277 A DK 22277A DK 141064 B DK141064 B DK 141064B
Authority
DK
Denmark
Prior art keywords
dihydro
formula
quinazolinone
compounds
phenyl
Prior art date
Application number
DK22277AA
Other languages
Danish (da)
English (en)
Other versions
DK141064C (pt-PT
DK22277A (pt-PT
Inventor
Michihiro Yamamoto
Hisao Yamamoto
Shigenari Katayama
Masao Koshiba
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of DK22277A publication Critical patent/DK22277A/da
Publication of DK141064B publication Critical patent/DK141064B/da
Application granted granted Critical
Publication of DK141064C publication Critical patent/DK141064C/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • C07D239/82Oxygen atoms with an aryl radical attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
DK22277AA 1976-01-23 1977-01-20 Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. DK141064B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP692076A JPS5291885A (en) 1976-01-23 1976-01-23 3,4-dihydro-2(1h)-quinazolinone derivatives
JP692076 1976-01-23

Publications (3)

Publication Number Publication Date
DK22277A DK22277A (pt-PT) 1977-07-24
DK141064B true DK141064B (da) 1980-01-07
DK141064C DK141064C (pt-PT) 1980-06-23

Family

ID=11651662

Family Applications (1)

Application Number Title Priority Date Filing Date
DK22277AA DK141064B (da) 1976-01-23 1977-01-20 Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater.

Country Status (13)

Country Link
US (1) US4048168A (pt-PT)
JP (1) JPS5291885A (pt-PT)
AT (1) AT353276B (pt-PT)
CA (1) CA1069505A (pt-PT)
CH (1) CH625231A5 (pt-PT)
DE (1) DE2702530A1 (pt-PT)
DK (1) DK141064B (pt-PT)
FR (1) FR2338934A1 (pt-PT)
GB (1) GB1525892A (pt-PT)
HU (1) HU174389B (pt-PT)
MX (1) MX3959E (pt-PT)
NL (1) NL7614574A (pt-PT)
SE (1) SE422324B (pt-PT)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5271483A (en) * 1975-12-11 1977-06-14 Sumitomo Chem Co Ltd Synthesis of 2(1h)-quinazolinone derivatives
US4282226A (en) * 1978-04-26 1981-08-04 E. R. Squibb & Sons, Inc. Thioxopyrazolo[1,5-c]quinazoline derivatives, anti-allergic compositions and methods for treating allergic conditions by parenteral administration, aerosol or insufflation
EP1394242A3 (en) * 2002-08-07 2004-04-21 Rohm And Haas Company Cyclic thioureas and their use as additives for lubricating oils
CA2513708C (en) * 2003-01-23 2011-01-04 Shire Holdings Ag Formulation and methods for the treatment of thrombocythemia
US20060030574A1 (en) * 2004-08-04 2006-02-09 Shire Holdings Ag Quinazoline derivatives useful for the treatment of peripheral arterial disease and as phosphodiesterase inhibitors
US7700608B2 (en) * 2004-08-04 2010-04-20 Shire Holdings Ag Quinazoline derivatives and their use in the treatment of thrombocythemia
US7910597B2 (en) * 2006-11-28 2011-03-22 Shire Llc Substituted quinazolines
US8304420B2 (en) 2006-11-28 2012-11-06 Shire Llc Substituted quinazolines for reducing platelet count

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3748331A (en) * 1971-05-06 1973-07-24 Sandoz Ag 1,4-disubstituted-methylenedioxy -2-(1h)-quinazolinones and quinazolinthiones

Also Published As

Publication number Publication date
SE422324B (sv) 1982-03-01
AT353276B (de) 1979-11-12
DK141064C (pt-PT) 1980-06-23
DK22277A (pt-PT) 1977-07-24
DE2702530A1 (de) 1977-07-28
CA1069505A (en) 1980-01-08
US4048168A (en) 1977-09-13
SE7700533L (sv) 1977-07-24
HU174389B (hu) 1979-12-28
ATA22777A (de) 1979-04-15
CH625231A5 (pt-PT) 1981-09-15
MX3959E (es) 1981-10-15
FR2338934A1 (fr) 1977-08-19
JPS5291885A (en) 1977-08-02
GB1525892A (en) 1978-09-20
NL7614574A (nl) 1977-07-26
AU2131477A (en) 1978-02-23
FR2338934B1 (pt-PT) 1980-12-19

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