DK140667B - Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf.

Info

Publication number
DK140667B
DK140667B DK53174AA DK53174A DK140667B DK 140667 B DK140667 B DK 140667B DK 53174A A DK53174A A DK 53174AA DK 53174 A DK53174 A DK 53174A DK 140667 B DK140667 B DK 140667B
Authority
DK
Denmark
Prior art keywords
dihydropteridines
salts
preparation
tautomeric forms
analogous process
Prior art date
Application number
DK53174AA
Other languages
Danish (da)
English (en)
Other versions
DK140667C (enrdf_load_stackoverflow
Inventor
Hamish Christopher Swan Wood
Norman Whittaker
Irene Stirling
Kyuji Ohta
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB518673A external-priority patent/GB1468171A/en
Priority claimed from DK420173AA external-priority patent/DK138019B/da
Priority to AR252155A priority Critical patent/AR205702A1/es
Priority to FR7403214A priority patent/FR2215963A1/fr
Priority to NL7401350A priority patent/NL7401350A/xx
Priority to CH136274A priority patent/CH601300A5/xx
Priority to DD176300A priority patent/DD110499A5/xx
Priority to ZA00740657A priority patent/ZA74657B/xx
Priority to PL1974168470A priority patent/PL91643B1/pl
Priority to HU74WE00000499A priority patent/HU171384B/hu
Priority to CS7400000661A priority patent/CS183731B2/cs
Priority to DE2404593A priority patent/DE2404593A1/de
Application filed by Wellcome Found filed Critical Wellcome Found
Priority to IN208/CAL/74A priority patent/IN139181B/en
Priority to DK53174AA priority patent/DK140667B/da
Priority to IE176/74A priority patent/IE38809B1/xx
Priority to SE7401254A priority patent/SE415563B/xx
Priority to CA191,502A priority patent/CA1025855A/en
Priority to ES422825A priority patent/ES422825A1/es
Priority to FI267/74A priority patent/FI55663C/fi
Priority to JP49013252A priority patent/JPS49102695A/ja
Priority to IL44123A priority patent/IL44123A/en
Priority to BE140440A priority patent/BE810474A/xx
Priority to AU65134/74A priority patent/AU478874B2/en
Publication of DK140667B publication Critical patent/DK140667B/da
Publication of DK140667C publication Critical patent/DK140667C/da
Application granted granted Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/02Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
    • C07D475/04Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK53174AA 1973-02-01 1974-01-31 Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf. DK140667B (da)

Priority Applications (21)

Application Number Priority Date Filing Date Title
AR252155A AR205702A1 (es) 1973-02-01 1974-01-01 Metodo para producir un nuevo derivado de 2-amino-4-hidroxi-7,8-dihidropteridina-6-carboxaldehido
BE140440A BE810474A (fr) 1973-02-01 1974-01-31 Composes a activite biologique
DK53174AA DK140667B (da) 1973-02-01 1974-01-31 Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf.
CH136274A CH601300A5 (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
DD176300A DD110499A5 (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
ZA00740657A ZA74657B (en) 1973-02-01 1974-01-31 Biologically active compounds
PL1974168470A PL91643B1 (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
HU74WE00000499A HU171384B (hu) 1973-02-01 1974-01-31 Sposob poluchenija biologicheski aktivnykh proizvodnykh pteridina
CS7400000661A CS183731B2 (en) 1973-02-01 1974-01-31 Method for producing novel pteridine derivatives
DE2404593A DE2404593A1 (de) 1973-02-01 1974-01-31 Biologisch wirksame verbindungen
FR7403214A FR2215963A1 (en) 1973-02-01 1974-01-31 Pteridine antimicrobials and bacteriostats
IN208/CAL/74A IN139181B (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
NL7401350A NL7401350A (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
IE176/74A IE38809B1 (en) 1973-02-01 1974-01-31 "2-amino-4-hydroxy-7,8-dithydropteridine-6-carboxaldehyde derivatives
SE7401254A SE415563B (sv) 1973-02-01 1974-01-31 Analogiforfarande for framstellning av 2-amino-4hydroxi-7,7-dimetyl-7,8-dihydropteridin-6-karboxaldehyd
CA191,502A CA1025855A (en) 1973-02-01 1974-01-31 Pteridine derivatives
ES422825A ES422825A1 (es) 1973-02-01 1974-01-31 Un metodo de preparar derivados de pteridina.
FI267/74A FI55663C (fi) 1973-02-01 1974-01-31 Foerfarande foer framstaellning av antimikrobiskt verkande 2-amino-4-hydroxi-7,7-dimetyl-7,8-dihydropteridin-6-karboxialdehyd
JP49013252A JPS49102695A (enrdf_load_stackoverflow) 1973-02-01 1974-01-31
IL44123A IL44123A (en) 1973-02-01 1974-01-31 2-amino-4-hydroxy-7,8-dihydropteridine-6-carboxaldehyde derivatives their preparation and pharmaceutical compositions containing them
AU65134/74A AU478874B2 (en) 1973-02-01 1974-02-01 Biologically active compounds

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB518673A GB1468171A (en) 1973-02-01 1973-02-01 2-amino-4-hydroxy-7,8-dihydropteridine-6-carboxaldehyde deri vatives
DK420173AA DK138019B (da) 1972-08-01 1973-07-31 Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere eller salte deraf.
DK53174AA DK140667B (da) 1973-02-01 1974-01-31 Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf.

Publications (2)

Publication Number Publication Date
DK140667B true DK140667B (da) 1979-10-22
DK140667C DK140667C (enrdf_load_stackoverflow) 1980-03-24

Family

ID=27220757

Family Applications (1)

Application Number Title Priority Date Filing Date
DK53174AA DK140667B (da) 1973-02-01 1974-01-31 Analogifremgangsmåde til fremstilling af 7,8-dihydropteridiner eller tautomere former eller salte deraf.

Country Status (20)

Country Link
JP (1) JPS49102695A (enrdf_load_stackoverflow)
AR (1) AR205702A1 (enrdf_load_stackoverflow)
BE (1) BE810474A (enrdf_load_stackoverflow)
CA (1) CA1025855A (enrdf_load_stackoverflow)
CH (1) CH601300A5 (enrdf_load_stackoverflow)
CS (1) CS183731B2 (enrdf_load_stackoverflow)
DD (1) DD110499A5 (enrdf_load_stackoverflow)
DE (1) DE2404593A1 (enrdf_load_stackoverflow)
DK (1) DK140667B (enrdf_load_stackoverflow)
ES (1) ES422825A1 (enrdf_load_stackoverflow)
FI (1) FI55663C (enrdf_load_stackoverflow)
FR (1) FR2215963A1 (enrdf_load_stackoverflow)
HU (1) HU171384B (enrdf_load_stackoverflow)
IE (1) IE38809B1 (enrdf_load_stackoverflow)
IL (1) IL44123A (enrdf_load_stackoverflow)
IN (1) IN139181B (enrdf_load_stackoverflow)
NL (1) NL7401350A (enrdf_load_stackoverflow)
PL (1) PL91643B1 (enrdf_load_stackoverflow)
SE (1) SE415563B (enrdf_load_stackoverflow)
ZA (1) ZA74657B (enrdf_load_stackoverflow)

Also Published As

Publication number Publication date
JPS49102695A (enrdf_load_stackoverflow) 1974-09-27
AR205702A1 (es) 1976-05-31
IE38809B1 (en) 1978-06-07
ES422825A1 (es) 1976-05-01
DD110499A5 (enrdf_load_stackoverflow) 1974-12-20
IE38809L (en) 1974-08-01
NL7401350A (enrdf_load_stackoverflow) 1974-08-05
DE2404593A1 (de) 1974-08-15
FR2215963B1 (enrdf_load_stackoverflow) 1976-09-03
CH601300A5 (enrdf_load_stackoverflow) 1978-07-14
SE415563B (sv) 1980-10-13
FI55663B (fi) 1979-05-31
PL91643B1 (enrdf_load_stackoverflow) 1977-03-31
AU6513474A (en) 1975-08-07
CA1025855A (en) 1978-02-07
CS183731B2 (en) 1978-07-31
IL44123A0 (en) 1974-05-16
DK140667C (enrdf_load_stackoverflow) 1980-03-24
BE810474A (fr) 1974-07-31
FI55663C (fi) 1979-09-10
ZA74657B (en) 1975-09-24
HU171384B (hu) 1977-12-28
FR2215963A1 (en) 1974-08-30
IN139181B (enrdf_load_stackoverflow) 1976-05-15
IL44123A (en) 1977-10-31

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