DK1404667T3 - Piperidinderivater, der er anvendelige som modulatorer af chemokinreceptoraktivitet - Google Patents

Piperidinderivater, der er anvendelige som modulatorer af chemokinreceptoraktivitet

Info

Publication number
DK1404667T3
DK1404667T3 DK02747793T DK02747793T DK1404667T3 DK 1404667 T3 DK1404667 T3 DK 1404667T3 DK 02747793 T DK02747793 T DK 02747793T DK 02747793 T DK02747793 T DK 02747793T DK 1404667 T3 DK1404667 T3 DK 1404667T3
Authority
DK
Denmark
Prior art keywords
modulators
chemokine receptor
receptor activity
derivatives useful
piperidine derivatives
Prior art date
Application number
DK02747793T
Other languages
English (en)
Inventor
Matthew Perry
Richard Evans
Brian Springthorpe
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0116179A external-priority patent/GB0116179D0/en
Priority claimed from GB0123037A external-priority patent/GB0123037D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK1404667T3 publication Critical patent/DK1404667T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/96—Sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/08—Antibacterial agents for leprosy
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
DK02747793T 2001-07-02 2002-07-01 Piperidinderivater, der er anvendelige som modulatorer af chemokinreceptoraktivitet DK1404667T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0116179A GB0116179D0 (en) 2001-07-02 2001-07-02 Chemical compounds
GB0123037A GB0123037D0 (en) 2001-09-25 2001-09-25 Chemical compounds

Publications (1)

Publication Number Publication Date
DK1404667T3 true DK1404667T3 (da) 2006-07-10

Family

ID=26246268

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02747793T DK1404667T3 (da) 2001-07-02 2002-07-01 Piperidinderivater, der er anvendelige som modulatorer af chemokinreceptoraktivitet

Country Status (26)

Country Link
US (1) US7307090B2 (da)
EP (2) EP1604982A1 (da)
JP (1) JP3857270B2 (da)
KR (1) KR20040013090A (da)
CN (1) CN1545509A (da)
AR (1) AR042401A1 (da)
AT (1) ATE319703T1 (da)
BR (1) BR0210733A (da)
CA (1) CA2452597A1 (da)
CO (1) CO5540307A2 (da)
CY (1) CY1106095T1 (da)
DE (1) DE60209736T2 (da)
DK (1) DK1404667T3 (da)
ES (1) ES2258642T3 (da)
HK (1) HK1062559A1 (da)
HU (1) HUP0401886A2 (da)
IL (1) IL159256A0 (da)
IS (1) IS7094A (da)
MX (1) MXPA03011722A (da)
NO (1) NO20035729L (da)
NZ (1) NZ530202A (da)
PL (1) PL368041A1 (da)
PT (1) PT1404667E (da)
RU (1) RU2004100839A (da)
SA (1) SA02230184B1 (da)
WO (1) WO2003004487A1 (da)

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SE0302956D0 (sv) * 2003-11-07 2003-11-07 Astrazeneca Ab Chemical compounds
SE0400925D0 (sv) * 2004-04-06 2004-04-06 Astrazeneca Ab Chemical compounds
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CN112105353B (zh) 2018-01-08 2024-04-19 凯莫森特里克斯股份有限公司 Ccr2拮抗剂治疗实体瘤的方法
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CA2452597A1 (en) 2003-01-16
AR042401A1 (es) 2005-06-22
IS7094A (is) 2003-12-30
HUP0401886A2 (hu) 2004-12-28
EP1404667B1 (en) 2006-03-08
CN1545509A (zh) 2004-11-10
ATE319703T1 (de) 2006-03-15
EP1604982A1 (en) 2005-12-14
RU2004100839A (ru) 2005-06-20
EP1404667A1 (en) 2004-04-07
NO20035729L (no) 2004-02-23
US7307090B2 (en) 2007-12-11
PL368041A1 (en) 2005-03-21
KR20040013090A (ko) 2004-02-11
PT1404667E (pt) 2006-07-31
CO5540307A2 (es) 2005-07-29
DE60209736T2 (de) 2006-11-02
JP2004536112A (ja) 2004-12-02
HK1062559A1 (en) 2004-11-12
SA02230184B1 (ar) 2007-03-25
JP3857270B2 (ja) 2006-12-13
CY1106095T1 (el) 2011-06-08
BR0210733A (pt) 2004-07-20
MXPA03011722A (es) 2004-03-19
US20040235894A1 (en) 2004-11-25
ES2258642T3 (es) 2006-09-01
IL159256A0 (en) 2004-06-01
NO20035729D0 (no) 2003-12-19
WO2003004487A1 (en) 2003-01-16
NZ530202A (en) 2005-06-24
DE60209736D1 (de) 2006-05-04

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