DK138893B - Analogifremgangsmåde til fremstilling af 1-(indolyl-3-alkyl)-4-ureido-piperidiner eller -thioureido-piperidiner eller syreadditionssalte deraf. - Google Patents
Analogifremgangsmåde til fremstilling af 1-(indolyl-3-alkyl)-4-ureido-piperidiner eller -thioureido-piperidiner eller syreadditionssalte deraf.Info
- Publication number
- DK138893B DK138893B DK101476AA DK101476A DK138893B DK 138893 B DK138893 B DK 138893B DK 101476A A DK101476A A DK 101476AA DK 101476 A DK101476 A DK 101476A DK 138893 B DK138893 B DK 138893B
- Authority
- DK
- Denmark
- Prior art keywords
- piperidines
- thioureido
- ureido
- indolyl
- alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55660075A | 1975-03-10 | 1975-03-10 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK101476A DK101476A (id) | 1976-09-11 |
| DK138893B true DK138893B (da) | 1978-11-13 |
| DK138893C DK138893C (id) | 1979-04-23 |
Family
ID=24222029
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK101476AA DK138893B (da) | 1975-03-10 | 1976-03-09 | Analogifremgangsmåde til fremstilling af 1-(indolyl-3-alkyl)-4-ureido-piperidiner eller -thioureido-piperidiner eller syreadditionssalte deraf. |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US4073911A (id) |
| JP (1) | JPS51113878A (id) |
| AU (1) | AU1175076A (id) |
| BE (1) | BE839347A (id) |
| DD (1) | DD124386A5 (id) |
| DE (1) | DE2609289A1 (id) |
| DK (1) | DK138893B (id) |
| ES (1) | ES445874A1 (id) |
| FI (1) | FI760584A (id) |
| FR (1) | FR2303541A1 (id) |
| GB (1) | GB1534351A (id) |
| GR (1) | GR60030B (id) |
| IL (1) | IL49171A (id) |
| NL (1) | NL7602508A (id) |
| NO (1) | NO760774L (id) |
| NZ (1) | NZ180255A (id) |
| PT (1) | PT64878B (id) |
| SE (1) | SE7602729L (id) |
| ZA (2) | ZA76475B (id) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4350634A (en) | 1977-07-12 | 1982-09-21 | Sandoz Ltd. | N-Benzoyl-N'-3-indolyl-N'alkyl-1,3-diaminopropanes |
| GB1586817A (en) * | 1977-12-01 | 1981-03-25 | Wyeth John & Brother Ltd | Indole derivatives |
| US4329348A (en) * | 1979-02-26 | 1982-05-11 | Ciba-Geigy Corporation | N-Oxacyclic-alkylpiperidines as psychostimulants |
| US4359468A (en) * | 1981-02-25 | 1982-11-16 | Boehringer Ingelheim Ltd. | Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones |
| NZ216720A (en) * | 1985-07-08 | 1990-09-26 | Bristol Myers Co | Diazinylpiperidine derivatives and pharmaceutical compositions |
| JP2807577B2 (ja) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
| EP0640081B1 (en) * | 1992-03-31 | 2000-01-12 | Glaxo Group Limited | Substituted phenylcarbamates and phenylureas, their preparation and their use as 5-ht4 antagonists |
| JP3916092B2 (ja) * | 1993-09-17 | 2007-05-16 | 杏林製薬株式会社 | イミダゾリジノン誘導体とその酸付加塩及び老年性痴呆症の治療薬 |
| US6489300B1 (en) * | 1997-07-31 | 2002-12-03 | Eugene D. Thorsett | Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 |
| FR2803298A1 (fr) * | 1999-12-30 | 2001-07-06 | Adir | Nouvelles urees lineaires ou cycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| EP1533299A4 (en) * | 2002-07-19 | 2007-04-04 | Meiji Dairies Corp | INDOIND DERIVATIVES AND MEDICAMENTS CONTAINING THEM |
| JP4705908B2 (ja) * | 2003-04-15 | 2011-06-22 | メルク・シャープ・エンド・ドーム・コーポレイション | Ｃｇｒｐ受容体拮抗薬 |
| CA2529196A1 (en) * | 2003-06-26 | 2005-02-17 | Merck & Co., Inc. | Benzodiazepine cgrp receptor antagonists |
| AU2005208834B2 (en) * | 2004-01-29 | 2009-10-08 | Merck Sharp & Dohme Corp. | CGRP receptor antagonists |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3238215A (en) * | 1963-10-17 | 1966-03-01 | Sterling Drug Inc | 1-[(3-, 2-, and 1-indolyl)-lower-alkyl-, lower-alkenyl-, and lower-alkynyl]piperidines |
| GB1273563A (en) * | 1968-07-24 | 1972-05-10 | Wyeth John & Brother Ltd | Indoles |
-
1976
- 1976-01-28 ZA ZA760475A patent/ZA76475B/xx unknown
- 1976-02-02 US US05/654,254 patent/US4073911A/en not_active Expired - Lifetime
- 1976-02-27 SE SE7602729A patent/SE7602729L/xx unknown
- 1976-03-05 GB GB8902/76A patent/GB1534351A/en not_active Expired
- 1976-03-05 NO NO760774A patent/NO760774L/no unknown
- 1976-03-06 GR GR50261A patent/GR60030B/el unknown
- 1976-03-06 DE DE19762609289 patent/DE2609289A1/de active Pending
- 1976-03-08 AU AU11750/76A patent/AU1175076A/en not_active Expired
- 1976-03-08 ES ES445874A patent/ES445874A1/es not_active Expired
- 1976-03-08 FI FI760584A patent/FI760584A/fi not_active Application Discontinuation
- 1976-03-08 FR FR7606495A patent/FR2303541A1/fr active Granted
- 1976-03-08 IL IL49171A patent/IL49171A/xx unknown
- 1976-03-09 PT PT64878A patent/PT64878B/pt unknown
- 1976-03-09 DD DD191763A patent/DD124386A5/xx unknown
- 1976-03-09 BE BE164977A patent/BE839347A/xx unknown
- 1976-03-09 DK DK101476AA patent/DK138893B/da unknown
- 1976-03-09 NZ NZ180255A patent/NZ180255A/xx unknown
- 1976-03-09 ZA ZA761467A patent/ZA761467B/xx unknown
- 1976-03-10 NL NL7602508A patent/NL7602508A/xx unknown
- 1976-03-10 JP JP51026622A patent/JPS51113878A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| ES445874A1 (es) | 1977-06-01 |
| ZA761467B (en) | 1977-10-26 |
| PT64878B (en) | 1977-07-22 |
| US4073911A (en) | 1978-02-14 |
| AU1175076A (en) | 1977-09-15 |
| DK138893C (id) | 1979-04-23 |
| IL49171A0 (en) | 1976-05-31 |
| DE2609289A1 (de) | 1976-09-30 |
| GR60030B (en) | 1978-03-31 |
| NO760774L (id) | 1976-09-13 |
| NZ180255A (en) | 1978-07-10 |
| PT64878A (en) | 1976-04-01 |
| FR2303541A1 (fr) | 1976-10-08 |
| GB1534351A (en) | 1978-12-06 |
| IL49171A (en) | 1978-12-17 |
| SE7602729L (sv) | 1976-09-13 |
| DK101476A (id) | 1976-09-11 |
| ZA76475B (en) | 1977-08-31 |
| NL7602508A (nl) | 1976-09-14 |
| JPS51113878A (en) | 1976-10-07 |
| FR2303541B1 (id) | 1979-10-05 |
| FI760584A (id) | 1976-09-11 |
| BE839347A (fr) | 1976-09-09 |
| DD124386A5 (id) | 1977-02-16 |
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