DK138496B - Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. - Google Patents
Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.Info
- Publication number
- DK138496B DK138496B DK34572AA DK34572A DK138496B DK 138496 B DK138496 B DK 138496B DK 34572A A DK34572A A DK 34572AA DK 34572 A DK34572 A DK 34572A DK 138496 B DK138496 B DK 138496B
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- acid addition
- addition salts
- imidazoline derivatives
- analogous process
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000002462 imidazolines Chemical class 0.000 title 1
- 229940083254 peripheral vasodilators imidazoline derivative Drugs 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB332771 | 1971-01-27 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK138496B true DK138496B (da) | 1978-09-18 |
| DK138496C DK138496C (cs) | 1979-02-26 |
Family
ID=9756227
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK34572AA DK138496B (da) | 1971-01-27 | 1972-01-26 | Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US3818035A (cs) |
| JP (1) | JPS4938273B1 (cs) |
| AT (1) | AT311336B (cs) |
| BE (1) | BE777689A (cs) |
| CA (1) | CA962273A (cs) |
| CH (1) | CH535254A (cs) |
| DE (1) | DE2203373C3 (cs) |
| DK (1) | DK138496B (cs) |
| FI (1) | FI55841C (cs) |
| GB (1) | GB1333471A (cs) |
| HU (1) | HU162823B (cs) |
| NL (1) | NL150454B (cs) |
| NO (1) | NO134115C (cs) |
| SE (1) | SE378426B (cs) |
| SU (1) | SU474145A3 (cs) |
| YU (1) | YU34694B (cs) |
| ZA (1) | ZA72286B (cs) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3927023A (en) * | 1974-05-24 | 1975-12-16 | Warner Lambert Co | Imidazolyl benzofurans |
| DE3049542A1 (de) * | 1980-12-31 | 1982-07-29 | Basf Ag, 6700 Ludwigshafen | Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung |
| ZA825413B (en) * | 1981-08-26 | 1983-06-29 | Pfizer | Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them |
| US4851554A (en) * | 1987-04-06 | 1989-07-25 | University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4806663A (en) * | 1987-04-06 | 1989-02-21 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4831156A (en) * | 1987-09-30 | 1989-05-16 | The University Of Tennessee Research Corp. | 3-substituted 2-alkyl indole derivatives |
| ZA9811672B (en) * | 1997-12-19 | 2000-06-19 | Lilly Co Eli | Hypoglycemic imidazoline compounds. |
| US7777035B2 (en) | 2005-06-22 | 2010-08-17 | Chemocentryx, Inc. | Azaindazole compounds and methods of use |
| BRPI0707315A2 (pt) * | 2006-01-27 | 2011-05-03 | Hoffmann La Roche | uso de 2-imidazol substituìdo de derivados de imidazolina |
| AU2007312389B2 (en) * | 2006-10-19 | 2012-02-23 | F. Hoffmann-La Roche Ag | Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors |
| CN101528710B (zh) * | 2006-10-19 | 2012-11-07 | 弗·哈夫曼-拉罗切有限公司 | 氨基甲基-4-咪唑类 |
| CA2668454A1 (en) * | 2006-11-02 | 2008-05-08 | F. Hoffmann-La Roche Ag | Substituted 2-imidazoles |
| CA2669112A1 (en) * | 2006-11-16 | 2008-05-22 | F. Hoffmann-La Roche Ag | Substituted 4-imidazoles |
| ATE509628T1 (de) * | 2006-12-13 | 2011-06-15 | Hoffmann La Roche | Neue 2-imidazole als liganden für trace amine associated receptors (taar) |
| US20080146523A1 (en) * | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
| KR101174191B1 (ko) * | 2007-02-02 | 2012-08-14 | 에프. 호프만-라 로슈 아게 | 중추 신경계 장애의 치료용 ｔａａｒ1 리간드로서 2-아미노옥사졸린 |
| AU2008214774A1 (en) * | 2007-02-15 | 2008-08-21 | F. Hoffmann-La Roche Ag | 2-aminooxazolines as TAAR1 ligands |
| WO2009003868A2 (en) | 2007-07-02 | 2009-01-08 | F. Hoffmann-La Roche Ag | 2 -imidazolines having a good affinity to the trace amine associated receptors (taars) |
| EP2173719A1 (en) * | 2007-07-03 | 2010-04-14 | F. Hoffmann-Roche AG | 4-imidazolines and their use as antidepressants |
| KR101133862B1 (ko) * | 2007-07-27 | 2012-04-06 | 에프. 호프만-라 로슈 아게 | Ｔａａｒ 리간드로서의 2-아제티딘메테인아민 및 2-피롤리딘메테인아민 |
| BRPI0815038A2 (pt) * | 2007-08-02 | 2015-03-17 | Hoffmann La Roche | Uso de derivados de benzamida para o tratamento de transtornos do cns |
| EP2185502A1 (en) * | 2007-08-03 | 2010-05-19 | F. Hoffmann-Roche AG | Pyridinecarboxamide and benzamide derivatives as taar1 ligands |
| PE20110215A1 (es) * | 2008-07-24 | 2011-03-31 | Hoffmann La Roche | Derivados de 4,5-dihidro-oxazol-2-ilo |
| US8242153B2 (en) * | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
| US20100311798A1 (en) * | 2009-06-05 | 2010-12-09 | Decoret Guillaume | 2-aminooxazolines as taar1 ligands |
| US8354441B2 (en) * | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
| US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| AU2017234042B2 (en) | 2016-03-17 | 2020-11-19 | F. Hoffmann-La Roche Ag | 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of TAAR |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1121054B (de) * | 1960-11-23 | 1962-01-04 | Merck Ag E | Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen |
-
1971
- 1971-01-27 GB GB332771A patent/GB1333471A/en not_active Expired
-
1972
- 1972-01-05 BE BE777689A patent/BE777689A/xx not_active IP Right Cessation
- 1972-01-06 CH CH17272A patent/CH535254A/fr not_active IP Right Cessation
- 1972-01-10 US US00216795A patent/US3818035A/en not_active Expired - Lifetime
- 1972-01-17 ZA ZA720286A patent/ZA72286B/xx unknown
- 1972-01-25 DE DE2203373A patent/DE2203373C3/de not_active Expired
- 1972-01-26 HU HULA791A patent/HU162823B/hu not_active IP Right Cessation
- 1972-01-26 NO NO192/72A patent/NO134115C/no unknown
- 1972-01-26 YU YU181/72A patent/YU34694B/xx unknown
- 1972-01-26 SE SE7200867A patent/SE378426B/xx unknown
- 1972-01-26 DK DK34572AA patent/DK138496B/da unknown
- 1972-01-27 JP JP47010207A patent/JPS4938273B1/ja active Pending
- 1972-01-27 CA CA133,337A patent/CA962273A/en not_active Expired
- 1972-01-27 SU SU1742351A patent/SU474145A3/ru active
- 1972-01-27 NL NL727201121A patent/NL150454B/xx not_active IP Right Cessation
- 1972-01-27 AT AT64772A patent/AT311336B/de not_active IP Right Cessation
- 1972-01-27 FI FI219/72A patent/FI55841C/fi active
Also Published As
| Publication number | Publication date |
|---|---|
| DE2203373A1 (de) | 1972-08-17 |
| US3818035A (en) | 1974-06-18 |
| DK138496C (cs) | 1979-02-26 |
| AT311336B (de) | 1973-11-12 |
| YU18172A (en) | 1979-07-10 |
| NO134115B (cs) | 1976-05-10 |
| FI55841B (fi) | 1979-06-29 |
| AU3817772A (en) | 1973-07-26 |
| NL7201121A (cs) | 1972-07-31 |
| CA962273A (en) | 1975-02-04 |
| NL150454B (nl) | 1976-08-16 |
| JPS4938273B1 (cs) | 1974-10-16 |
| SU474145A3 (ru) | 1975-06-14 |
| GB1333471A (en) | 1973-10-10 |
| DE2203373B2 (de) | 1977-08-11 |
| FI55841C (fi) | 1979-10-10 |
| HU162823B (cs) | 1973-04-28 |
| SE378426B (cs) | 1975-09-01 |
| DE2203373C3 (de) | 1978-04-13 |
| YU34694B (en) | 1979-12-31 |
| NO134115C (cs) | 1976-08-18 |
| BE777689A (fr) | 1972-07-05 |
| CH535254A (fr) | 1973-03-31 |
| ZA72286B (en) | 1972-09-27 |
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