DK132174C - ANALOGICAL PROCEDURE FOR THE PREPARATION OF 2,4-DIAMINO-5-BENZYLPYRIMIDINES - Google Patents

ANALOGICAL PROCEDURE FOR THE PREPARATION OF 2,4-DIAMINO-5-BENZYLPYRIMIDINES

Info

Publication number
DK132174C
DK132174C DK513771A DK513771A DK132174C DK 132174 C DK132174 C DK 132174C DK 513771 A DK513771 A DK 513771A DK 513771 A DK513771 A DK 513771A DK 132174 C DK132174 C DK 132174C
Authority
DK
Denmark
Prior art keywords
benzylpyrimidines
diamino
preparation
analogical procedure
analogical
Prior art date
Application number
DK513771A
Other languages
Danish (da)
Other versions
DK132174B (en
Inventor
B Roth
A Stuart
T Paterson
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK132174B publication Critical patent/DK132174B/en
Application granted granted Critical
Publication of DK132174C publication Critical patent/DK132174C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK513771A 1970-10-22 1971-10-21 ANALOGICAL PROCEDURE FOR THE PREPARATION OF 2,4-DIAMINO-5-BENZYLPYRIMIDINES DK132174C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB963871*[A GB1375162A (en) 1970-10-22 1970-10-22
GB963871 1971-04-16
GB4749171 1971-10-12

Publications (2)

Publication Number Publication Date
DK132174B DK132174B (en) 1975-11-03
DK132174C true DK132174C (en) 1976-03-29

Family

ID=27255400

Family Applications (1)

Application Number Title Priority Date Filing Date
DK513771A DK132174C (en) 1970-10-22 1971-10-21 ANALOGICAL PROCEDURE FOR THE PREPARATION OF 2,4-DIAMINO-5-BENZYLPYRIMIDINES

Country Status (20)

Country Link
JP (2) JPS5536662B1 (en)
AR (3) AR192588A1 (en)
AT (1) AT319948B (en)
BE (1) BE774281A (en)
BG (4) BG20364A3 (en)
CA (1) CA967158A (en)
CH (3) CH568302A5 (en)
DD (1) DD100877A5 (en)
DK (1) DK132174C (en)
ES (1) ES396219A1 (en)
FI (1) FI56175C (en)
FR (1) FR2111769B1 (en)
GB (1) GB1375162A (en)
IE (1) IE37452B1 (en)
IL (2) IL37984A (en)
LU (1) LU64129A1 (en)
MC (1) MC894A1 (en)
NL (1) NL175178C (en)
SE (2) SE384505B (en)
ZM (1) ZM14971A1 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE792096A (en) * 1971-12-01 1973-05-30 Hoffmann La Roche NEW BENZYLPYRIMIDINES
FR2397407A2 (en) * 1977-07-11 1979-02-09 Dick Pierre 2,4-DIAMINO PYRIMIDINE DERIVATIVES AND THEIR SOLUTION IN ASSOCIATION WITH SULFAMIDS
FI791638A (en) * 1978-05-24 1979-11-25 Wellcome Found BENZYLPYRIMIDINE COMPOSITIONER
JPS61156909A (en) * 1984-12-27 1986-07-16 Matsushita Electric Ind Co Ltd Current mirror circuit
JPS62145907A (en) * 1985-12-20 1987-06-30 Hitachi Ltd Transistor circuit
RU2397171C2 (en) 2004-03-26 2010-08-20 ДАЙНИППОН СУМИТОМО ФАРМА Ко., ЛТД. 9-substituted derivative of 8-oxoadenine and medicinal agent
WO2008004948A1 (en) 2006-07-05 2008-01-10 Astrazeneca Ab 8-oxoadenine derivatives acting as modulators of tlr7
TW200831105A (en) 2006-12-14 2008-08-01 Astrazeneca Ab Novel compounds
DK2132209T3 (en) 2007-03-19 2014-04-14 Astrazeneca Ab 9-SUBSTITUTED 8-OXO ADENINE COMPOUNDS AS MODULATORS OF TLR7 (TOLL-LIKE RECEPTOR 7)
JP5329444B2 (en) 2007-03-19 2013-10-30 アストラゼネカ・アクチエボラーグ 9-Substituted-8-oxo-adenine compounds as TOLL-like receptor (TLR7) modulators
US8044056B2 (en) 2007-03-20 2011-10-25 Dainippon Sumitomo Pharma Co., Ltd. Adenine compound
PE20091236A1 (en) * 2007-11-22 2009-09-16 Astrazeneca Ab PYRIMIDINE DERIVATIVES AS IMMUNOMODULATORS OF TLR7
PE20091156A1 (en) 2007-12-17 2009-09-03 Astrazeneca Ab SALTS OF (3 - {[[3- (6-AMINO-2-BUTOXY-8-OXO-7,8-DIHIDRO-9H-PURIN-9-IL) PROPYL] (3-MORFOLIN-4-ILPROPIL) AMINO] METHYL} PHENYL) METHYL ACETATE
GB0908772D0 (en) 2009-05-21 2009-07-01 Astrazeneca Ab New salts 756
WO2010133885A1 (en) 2009-05-21 2010-11-25 Astrazeneca Ab Novel pyrimidine derivatives and their use in the treatment of cancer and further diseases
CN103370317B (en) 2010-12-16 2015-10-07 阿斯利康(瑞典)有限公司 Can be used for imidazo [4, the 5-c] quinoline-1-radical derivative for the treatment of
US8895570B2 (en) 2010-12-17 2014-11-25 Astrazeneca Ab Purine derivatives
TWI619704B (en) 2012-05-18 2018-04-01 大日本住友製藥股份有限公司 Carboxylic acid compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE710100A (en) * 1967-02-02 1968-07-30
JPS511716A (en) * 1974-06-25 1976-01-08 Toray Industries HORIESUTERUMARUCHIFUIRAMENTONO SEIHO

Also Published As

Publication number Publication date
IL45422A (en) 1976-03-31
JPS53135991A (en) 1978-11-28
NL175178B (en) 1984-05-01
CH568302A5 (en) 1975-10-31
FI56175B (en) 1979-08-31
CH568301A5 (en) 1975-10-31
IL37984A (en) 1976-03-31
SE384505B (en) 1976-05-10
BG20797A3 (en) 1975-12-20
FI56175C (en) 1979-12-10
BG20364A3 (en) 1975-11-05
MC894A1 (en) 1972-06-22
BG21406A3 (en) 1976-05-20
DD100877A5 (en) 1973-10-12
SE409705B (en) 1979-09-03
CA967158A (en) 1975-05-06
AR192588A1 (en) 1973-02-28
IE37452B1 (en) 1977-08-03
CH582681A5 (en) 1976-12-15
BE774281A (en) 1972-04-21
LU64129A1 (en) 1972-06-28
NL7114494A (en) 1972-04-25
AT319948B (en) 1975-01-10
FR2111769B1 (en) 1974-10-18
NL175178C (en) 1984-10-01
DK132174B (en) 1975-11-03
BG20365A3 (en) 1975-11-05
GB1375162A (en) 1974-11-27
FR2111769A1 (en) 1972-06-09
IE37452L (en) 1972-04-22
IL37984A0 (en) 1971-12-29
JPS5536662B1 (en) 1980-09-22
AR192803A1 (en) 1973-03-14
ES396219A1 (en) 1975-09-16
ZM14971A1 (en) 1972-07-21
AR192802A1 (en) 1973-03-14

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