DK129779A - Fremgangsmaade til omdannelse af penicillinsulfoxidestere - Google Patents

Fremgangsmaade til omdannelse af penicillinsulfoxidestere

Info

Publication number
DK129779A
DK129779A DK129779A DK129779A DK129779A DK 129779 A DK129779 A DK 129779A DK 129779 A DK129779 A DK 129779A DK 129779 A DK129779 A DK 129779A DK 129779 A DK129779 A DK 129779A
Authority
DK
Denmark
Prior art keywords
sulfoxidests
penicillin
conversion
procedure
penicillin sulfoxidests
Prior art date
Application number
DK129779A
Other languages
English (en)
Inventor
R L Cundall
D Walker
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of DK129779A publication Critical patent/DK129779A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK129779A 1978-04-03 1979-03-29 Fremgangsmaade til omdannelse af penicillinsulfoxidestere DK129779A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/893,092 US4322347A (en) 1978-04-03 1978-04-03 2-Carbamoyloxymethyl-penicillin derivatives

Publications (1)

Publication Number Publication Date
DK129779A true DK129779A (da) 1979-10-04

Family

ID=25401020

Family Applications (1)

Application Number Title Priority Date Filing Date
DK129779A DK129779A (da) 1978-04-03 1979-03-29 Fremgangsmaade til omdannelse af penicillinsulfoxidestere

Country Status (15)

Country Link
US (1) US4322347A (da)
JP (1) JPS54132594A (da)
BE (1) BE875247A (da)
CA (1) CA1140915A (da)
CH (1) CH642080A5 (da)
DE (1) DE2912483A1 (da)
DK (1) DK129779A (da)
FR (1) FR2421903B1 (da)
GB (1) GB2017705B (da)
IE (1) IE49046B1 (da)
IT (1) IT1116851B (da)
LU (1) LU81108A1 (da)
NL (1) NL7902443A (da)
SE (3) SE448239B (da)
YU (5) YU41860B (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4374982A (en) * 1979-11-07 1983-02-22 Bristol-Myers Company Cepham compounds
IT1148888B (it) * 1980-07-15 1986-12-03 Schiena Ricerche Di Composti antibiotici
CA2001642A1 (en) * 1988-10-31 1990-04-30 David J. Bartkovitz Penicillanic acid derivatives
US5604222A (en) * 1993-12-27 1997-02-18 Lupin Laboratories, Ltd. Method for the preparation of 2-chloro sulfinyl azetidinones
US5578721A (en) * 1994-07-11 1996-11-26 Lupin Laboratories Limited Process for preparation of 3-exomethylene cepham sulfoxide esters
CN104011061B (zh) 2011-12-20 2017-06-13 里博科学有限责任公司 作为hcv rna复制抑制剂的2‘,4’‑二氟‑2‘‑甲基取代的核苷衍生物
EA024847B1 (ru) 2011-12-20 2016-10-31 Рибосайенс Ллк 4'-азидо,3'-фторзамещенные производные нуклеозидов в качестве ингибиторов репликации рнк вируса гепатита с
US20180200280A1 (en) 2013-05-16 2018-07-19 Riboscience Llc 4'-Fluoro-2'-Methyl Substituted Nucleoside Derivatives as Inhibitors of HCV RNA Replication
CN105307661A (zh) 2013-05-16 2016-02-03 里博科学有限责任公司 4’-叠氮基,3’-脱氧基-3’-氟取代的核苷衍生物
UA123533C2 (uk) 2013-05-16 2021-04-21 Рібосаєнс Ллс 4'-фтор-2'-метилзаміщені нуклеозидні похідні
AR112702A1 (es) 2017-09-21 2019-11-27 Riboscience Llc Derivados de nucleósidos sustituidos con 4’-fluoro-2’-metilo como inhibidores de la replicación de hcv arn

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275626A (en) * 1962-07-31 1966-09-27 Lilly Co Eli Penicillin conversion via sulfoxide
US3714156A (en) * 1970-06-22 1973-01-30 Univ California Lactam process
BE787618A (fr) 1971-08-17 1973-02-16 Gist Brocades Nv Procede pour preparer des composes heterocycliques
GB1425827A (en) * 1972-03-13 1976-02-18 Astra Laekemedel Ab Penicillins and cephalosporins
US4218374A (en) * 1972-10-20 1980-08-19 Fujisawa Pharmaceutical Company, Limited Penam derivatives
GB1465893A (en) * 1973-02-09 1977-03-02 Gist Brocades Nv I-carboxypropenyl-4-iminothio-azetidine-2-one derivatives methods for their preparation and use
DE2309599A1 (de) * 1973-02-26 1974-09-05 Bayer Ag Verfahren zur herstellung von 7-acylamino-desacetoxy-cephalosporansaeurederivaten
US4010156A (en) * 1973-04-19 1977-03-01 American Home Products Corporation Process for the rearrangement of penicillins to cephalosporins and intermediate compounds thereof
DE2320040A1 (de) 1973-04-19 1974-11-07 Bayer Ag Verfahren zur herstellung von 7acylamino-desacetoxy-cephalosporansaeureester
GB1467604A (en) * 1974-06-27 1977-03-16 Toyama Chemical Co Ltd Bis-type penicillins and process for producing the same
FR2340093A1 (fr) 1976-02-05 1977-09-02 Roussel Uclaf Derives de l'acide 3-carbamoyloxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
GB1573614A (en) * 1976-02-25 1980-08-28 Leo Pharm Prod Ltd Amidinopenicillanoyloxyalkyl cephalosporanates
DE2655949A1 (de) * 1976-12-10 1978-06-15 Gruenenthal Gmbh Neue cephalosporin- und penicillinderivate, verfahren zu deren herstellung und diese produkte enthaltende arzneimittel
US4182711A (en) * 1978-04-27 1980-01-08 Bristol-Myers Company Antibacterial agents of the β-lactam type
CA1125745A (en) * 1978-11-20 1982-06-15 Joseph Kaspi PROCESS FOR PREPARING .beta.-LACTAM ANTIBIOTICS

Also Published As

Publication number Publication date
US4322347A (en) 1982-03-30
FR2421903A1 (fr) 1979-11-02
SE8402090L (sv) 1984-04-13
SE458610B (sv) 1989-04-17
YU41860B (en) 1988-02-29
SE7902916L (sv) 1979-10-04
SE458609B (sv) 1989-04-17
YU220682A (en) 1983-01-21
YU42803B (en) 1988-12-31
SE8402089L (sv) 1984-04-13
YU42050B (en) 1988-04-30
YU220782A (en) 1983-01-21
NL7902443A (nl) 1979-10-05
YU220482A (en) 1983-01-21
BE875247A (fr) 1979-10-01
JPS54132594A (en) 1979-10-15
IE49046B1 (en) 1985-07-24
YU220582A (en) 1983-01-21
IT1116851B (it) 1986-02-10
IE790947L (en) 1979-10-03
GB2017705A (en) 1979-10-10
SE8402089D0 (sv) 1984-04-13
YU42802B (en) 1988-12-31
SE448239B (sv) 1987-02-02
GB2017705B (en) 1982-10-27
YU43096B (en) 1989-02-28
SE8402090D0 (sv) 1984-04-13
JPH0217557B2 (da) 1990-04-20
YU75679A (en) 1983-01-21
CA1140915A (en) 1983-02-08
IT7948457A0 (it) 1979-03-23
FR2421903B1 (fr) 1986-08-29
CH642080A5 (fr) 1984-03-30
LU81108A1 (de) 1979-11-07
DE2912483A1 (de) 1979-10-11

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