BE875247A - Nouveaux antibiotiques du type beta-lactame, leur procede de production et medicament les contenant - Google Patents

Nouveaux antibiotiques du type beta-lactame, leur procede de production et medicament les contenant

Info

Publication number
BE875247A
BE875247A BE0/194349A BE194349A BE875247A BE 875247 A BE875247 A BE 875247A BE 0/194349 A BE0/194349 A BE 0/194349A BE 194349 A BE194349 A BE 194349A BE 875247 A BE875247 A BE 875247A
Authority
BE
Belgium
Prior art keywords
beta
production process
product containing
medicinal product
new antibiotics
Prior art date
Application number
BE0/194349A
Other languages
English (en)
Inventor
R Cundall
D Walker
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of BE875247A publication Critical patent/BE875247A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BE0/194349A 1978-04-03 1979-03-30 Nouveaux antibiotiques du type beta-lactame, leur procede de production et medicament les contenant BE875247A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/893,092 US4322347A (en) 1978-04-03 1978-04-03 2-Carbamoyloxymethyl-penicillin derivatives

Publications (1)

Publication Number Publication Date
BE875247A true BE875247A (fr) 1979-10-01

Family

ID=25401020

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/194349A BE875247A (fr) 1978-04-03 1979-03-30 Nouveaux antibiotiques du type beta-lactame, leur procede de production et medicament les contenant

Country Status (15)

Country Link
US (1) US4322347A (fr)
JP (1) JPS54132594A (fr)
BE (1) BE875247A (fr)
CA (1) CA1140915A (fr)
CH (1) CH642080A5 (fr)
DE (1) DE2912483A1 (fr)
DK (1) DK129779A (fr)
FR (1) FR2421903B1 (fr)
GB (1) GB2017705B (fr)
IE (1) IE49046B1 (fr)
IT (1) IT1116851B (fr)
LU (1) LU81108A1 (fr)
NL (1) NL7902443A (fr)
SE (3) SE448239B (fr)
YU (5) YU41860B (fr)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9108999B2 (en) 2011-12-20 2015-08-18 Riboscience Llc 2′, 4′-difluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9249176B2 (en) 2013-05-16 2016-02-02 Riboscience Llc 4′-azido, 3′-deoxy-3′-fluoro substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9708357B2 (en) 2011-12-20 2017-07-18 Riboscience, LLC 4′-azido, 3′-fluoro substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9895442B2 (en) 2013-05-16 2018-02-20 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US10682369B2 (en) 2017-09-21 2020-06-16 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US10953030B2 (en) 2013-05-16 2021-03-23 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4374982A (en) * 1979-11-07 1983-02-22 Bristol-Myers Company Cepham compounds
IT1148888B (it) * 1980-07-15 1986-12-03 Schiena Ricerche Di Composti antibiotici
IL92139A0 (en) * 1988-10-31 1990-07-12 Hoffmann La Roche Penicillanic acid derivatives,their manufacture and pharmaceutical compositions containing them
US5604222A (en) * 1993-12-27 1997-02-18 Lupin Laboratories, Ltd. Method for the preparation of 2-chloro sulfinyl azetidinones
US5578721A (en) * 1994-07-11 1996-11-26 Lupin Laboratories Limited Process for preparation of 3-exomethylene cepham sulfoxide esters

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275626A (en) * 1962-07-31 1966-09-27 Lilly Co Eli Penicillin conversion via sulfoxide
US3714156A (en) * 1970-06-22 1973-01-30 Univ California Lactam process
BE787618A (fr) 1971-08-17 1973-02-16 Gist Brocades Nv Procede pour preparer des composes heterocycliques
GB1425827A (en) * 1972-03-13 1976-02-18 Astra Laekemedel Ab Penicillins and cephalosporins
US4218374A (en) * 1972-10-20 1980-08-19 Fujisawa Pharmaceutical Company, Limited Penam derivatives
GB1465893A (en) * 1973-02-09 1977-03-02 Gist Brocades Nv I-carboxypropenyl-4-iminothio-azetidine-2-one derivatives methods for their preparation and use
DE2309599A1 (de) * 1973-02-26 1974-09-05 Bayer Ag Verfahren zur herstellung von 7-acylamino-desacetoxy-cephalosporansaeurederivaten
DE2320040A1 (de) 1973-04-19 1974-11-07 Bayer Ag Verfahren zur herstellung von 7acylamino-desacetoxy-cephalosporansaeureester
US4010156A (en) * 1973-04-19 1977-03-01 American Home Products Corporation Process for the rearrangement of penicillins to cephalosporins and intermediate compounds thereof
GB1467604A (en) * 1974-06-27 1977-03-16 Toyama Chemical Co Ltd Bis-type penicillins and process for producing the same
FR2340093A1 (fr) 1976-02-05 1977-09-02 Roussel Uclaf Derives de l'acide 3-carbamoyloxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
GB1573614A (en) * 1976-02-25 1980-08-28 Leo Pharm Prod Ltd Amidinopenicillanoyloxyalkyl cephalosporanates
DE2655949A1 (de) * 1976-12-10 1978-06-15 Gruenenthal Gmbh Neue cephalosporin- und penicillinderivate, verfahren zu deren herstellung und diese produkte enthaltende arzneimittel
US4182711A (en) * 1978-04-27 1980-01-08 Bristol-Myers Company Antibacterial agents of the β-lactam type
CA1125745A (fr) * 1978-11-20 1982-06-15 Joseph Kaspi Procede de preparation du -lactam

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9108999B2 (en) 2011-12-20 2015-08-18 Riboscience Llc 2′, 4′-difluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9708357B2 (en) 2011-12-20 2017-07-18 Riboscience, LLC 4′-azido, 3′-fluoro substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9249176B2 (en) 2013-05-16 2016-02-02 Riboscience Llc 4′-azido, 3′-deoxy-3′-fluoro substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9694028B2 (en) 2013-05-16 2017-07-04 Riboscience Llc 4′-azido, 3′-deoxy-3′-fluoro substituted nucleoside derivatives as inhibitors of HCV RNA replication
US9895442B2 (en) 2013-05-16 2018-02-20 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US10953030B2 (en) 2013-05-16 2021-03-23 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US10682369B2 (en) 2017-09-21 2020-06-16 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication
US11351186B2 (en) 2017-09-21 2022-06-07 Riboscience Llc 4′-fluoro-2′-methyl substituted nucleoside derivatives as inhibitors of HCV RNA replication

Also Published As

Publication number Publication date
DE2912483A1 (de) 1979-10-11
DK129779A (da) 1979-10-04
SE8402089D0 (sv) 1984-04-13
SE8402089L (sv) 1984-04-13
SE7902916L (sv) 1979-10-04
IT7948457A0 (it) 1979-03-23
IE49046B1 (en) 1985-07-24
SE448239B (sv) 1987-02-02
IE790947L (en) 1979-10-03
SE8402090D0 (sv) 1984-04-13
YU220482A (en) 1983-01-21
CH642080A5 (fr) 1984-03-30
FR2421903A1 (fr) 1979-11-02
CA1140915A (fr) 1983-02-08
JPS54132594A (en) 1979-10-15
YU220582A (en) 1983-01-21
YU220782A (en) 1983-01-21
GB2017705A (en) 1979-10-10
GB2017705B (en) 1982-10-27
LU81108A1 (de) 1979-11-07
YU41860B (en) 1988-02-29
SE8402090L (sv) 1984-04-13
NL7902443A (nl) 1979-10-05
IT1116851B (it) 1986-02-10
SE458610B (sv) 1989-04-17
SE458609B (sv) 1989-04-17
FR2421903B1 (fr) 1986-08-29
US4322347A (en) 1982-03-30
YU75679A (en) 1983-01-21
JPH0217557B2 (fr) 1990-04-20
YU42050B (en) 1988-04-30
YU220682A (en) 1983-01-21
YU42803B (en) 1988-12-31
YU42802B (en) 1988-12-31
YU43096B (en) 1989-02-28

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: BRISTOL-MYERS CY

Effective date: 19870331